Synthesis and Biological Evaluation of Fused Tricyclic Heterocycle Piperazine (Piperidine) Derivatives As Potential Multireceptor Atypical Antipsychotics
Cao, Xudong, Zhang, Yifang, Chen, Yin, Qiu, Yinli, Yu, Minquan, Xu, Xiangqing, Liu, Xin, Liu, Bi-Feng, Zhang, Liangren, Zhang, Guisen
Published in Journal of medicinal chemistry (21.11.2018)
Published in Journal of medicinal chemistry (21.11.2018)
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A novel dual serotonin transporter and M-channel inhibitor D01 for antidepression and cognitive improvement
Wei, Yaqin, Xu, Xiangqing, Guo, Qiang, Zhao, Song, Qiu, Yinli, Wang, Dongli, Yu, Wenwen, Liu, Yani, Wang, KeWei
Published in Acta pharmaceutica Sinica. B (01.03.2024)
Published in Acta pharmaceutica Sinica. B (01.03.2024)
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Carbazole and tetrahydro-carboline derivatives as dopamine D3 receptor antagonists with the multiple antipsychotic-like properties
Li, Zhongtang, Fang, Fan, Li, Yiyan, Lv, Xuehui, Zheng, Ruqiu, Jiao, Peili, Wang, Yuxi, Zhu, Guiwang, Jin, Zefang, Xu, Xiangqing, Qiu, Yinli, Zhang, Guisen, Li, Zhongjun, Liu, Zhenming, Zhang, Liangren
Published in Acta pharmaceutica Sinica. B (01.11.2023)
Published in Acta pharmaceutica Sinica. B (01.11.2023)
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Synthesis and evaluation of fluorine-substituted phenyl acetate derivatives as ultra-short recovery sedative/hypnotic agents
Zhang, Heng, Xu, Xiangqing, Chen, Yin, Qiu, Yinli, Liu, Xin, Liu, Bi-Feng, Zhang, Guisen
Published in PloS one (05.05.2014)
Published in PloS one (05.05.2014)
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Journal Article
Synthesis and Biological Investigation of Coumarin Piperazine (Piperidine) Derivatives as Potential Multireceptor Atypical Antipsychotics
Chen, Yin, Wang, Songlin, Xu, Xiangqing, Liu, Xin, Yu, Minquan, Zhao, Song, Liu, Shicheng, Qiu, Yinli, Zhang, Tan, Liu, Bi-Feng, Zhang, Guisen
Published in Journal of medicinal chemistry (13.06.2013)
Published in Journal of medicinal chemistry (13.06.2013)
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Journal Article
2,6-diazaspiro[3.4]octan-7-one derivatives as potent sigma-1 receptor antagonists that enhanced the antinociceptive effect of morphine and rescued morphine tolerance
Fu, Kequan, Xu, Wen, Yang, Ruicong, Zhao, Huimin, Xu, Huanyu, Wei, Yaqin, Liu, Hongli, Qiu, Yinli, Chen, Danqi, Guo, Dong, Xiong, Bing
Published in European journal of medicinal chemistry (05.03.2023)
Published in European journal of medicinal chemistry (05.03.2023)
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A Novel Etomidate Analog EL-0052 Retains Potent Hypnotic Effect and Stable Hemodynamics without Suppressing Adrenocortical Function
Xu, Xiangqing, Wei, Yaqin, Dong, Yingying, Qiu, Yinli, Mei, Zhanbiao, Wang, Kai, Xiu, Jingya, Wang, Tao, Zeng, Lingguo, Dong, Xiaohu, Shen, Yi, Jiang, Wengao, Li, Qingeng
Published in The Journal of pharmacology and experimental therapeutics (01.12.2021)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2021)
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Discovery of Novel and Potent N‑Methyl‑d‑aspartate Receptor Positive Allosteric Modulators with Antidepressant-like Activity in Rodent Models
Li, Zhongtang, Cai, Guanxing, Fang, Fan, Li, Wenchao, Fan, Minghua, Lian, Jingjing, Qiu, Yinli, Xu, Xiangqing, Lv, Xuehui, Li, Yiyan, Zheng, Ruqiu, Wang, Yuxi, Li, Zhongjun, Zhang, Guisen, Liu, Zhenming, Huang, Zhuo, Zhang, Liangren
Published in Journal of medicinal chemistry (13.05.2021)
Published in Journal of medicinal chemistry (13.05.2021)
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Synthesis and Biological Evaluation of Novel σ1 Receptor Ligands for Treating Neuropathic Pain: 6‑Hydroxypyridazinones
Cao, Xudong, Chen, Yin, Zhang, Yifang, Lan, Yu, Zhang, Juecheng, Xu, Xiangqing, Qiu, Yinli, Zhao, Song, Liu, Xin, Liu, Bi-Feng, Zhang, Guisen
Published in Journal of medicinal chemistry (14.04.2016)
Published in Journal of medicinal chemistry (14.04.2016)
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Journal Article
Pharmacological Characterization of H05, a Novel Serotonin and Noradrenaline Reuptake Inhibitor with Moderate 5-HT2A Antagonist Activity for the Treatment of Depression
Xu, Xiangqing, Wei, Yaqin, Guo, Qiang, Zhao, Song, Liu, Zhiqiang, Xiao, Ting, Liu, Yani, Qiu, Yinli, Hou, Yuanyuan, Zhang, Guisen, Wang, KeWei
Published in The Journal of pharmacology and experimental therapeutics (01.06.2018)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2018)
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Journal Article
Synthesis and biological evaluation of a novel sigma-1 receptor antagonist based on 3,4-dihydro-2(1H)-quinolinone scaffold as a potential analgesic
Lan, Yu, Chen, Yin, Xu, Xiangqing, Qiu, Yinli, Liu, Shicheng, Liu, Xin, Liu, Bi-Feng, Zhang, Guisen
Published in European journal of medicinal chemistry (22.05.2014)
Published in European journal of medicinal chemistry (22.05.2014)
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Journal Article
Synthesis and Biological Evaluation of Novel Sigma‑1 Receptor Antagonists Based on Pyrimidine Scaffold As Agents for Treating Neuropathic Pain
Lan, Yu, Chen, Yin, Cao, Xudong, Zhang, Juecheng, Wang, Jie, Xu, Xiangqing, Qiu, Yinli, Zhang, Tan, Liu, Xin, Liu, Bi-Feng, Zhang, Guisen
Published in Journal of medicinal chemistry (26.12.2014)
Published in Journal of medicinal chemistry (26.12.2014)
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Journal Article
Pharmacological Characterization of H05, a Novel Serotonin and Noradrenaline Reuptake Inhibitor with Moderate 5-HT 2A Antagonist Activity for the Treatment of Depression
Xu, Xiangqing, Wei, Yaqin, Guo, Qiang, Zhao, Song, Liu, Zhiqiang, Xiao, Ting, Liu, Yani, Qiu, Yinli, Hou, Yuanyuan, Zhang, Guisen, Wang, KeWei
Published in The Journal of pharmacology and experimental therapeutics (01.06.2018)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2018)
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Journal Article
Synthesis and biological evaluation of new 6-hydroxypyridazinone benzisoxazoles: Potential multi-receptor-targeting atypical antipsychotics
Cao, Xudong, Chen, Yin, Zhang, Yifang, Qiu, Yinli, Yu, Minquan, Xu, Xiangqing, Liu, Xin, Liu, Bi-Feng, Zhang, Guisen
Published in European journal of medicinal chemistry (29.11.2016)
Published in European journal of medicinal chemistry (29.11.2016)
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Journal Article
Carbazole and tetrahydro-carboline derivatives as dopamine D 3 receptor antagonists with the multiple antipsychotic-like properties
Li, Zhongtang, Fang, Fan, Li, Yiyan, Lv, Xuehui, Zheng, Ruqiu, Jiao, Peili, Wang, Yuxi, Zhu, Guiwang, Jin, Zefang, Xu, Xiangqing, Qiu, Yinli, Zhang, Guisen, Li, Zhongjun, Liu, Zhenming, Zhang, Liangren
Published in Acta pharmaceutica Sinica. B (01.11.2023)
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Published in Acta pharmaceutica Sinica. B (01.11.2023)
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Synthesis and Biological Evaluation of Sigma‐1 (σ1) Receptor Ligands Based on Phenyl‐1,2,4‐oxadiazole Derivatives
Cao, Xudong, Yao, Zhongyuan, Dou, Fei, Zhang, Yifang, Qiu, Yinli, Zhao, Song, Xu, Xiangqing, Liu, Xin, Liu, Bi‐Feng, Chen, Yin, Zhang, Guisen
Published in Chemistry & biodiversity (01.03.2019)
Published in Chemistry & biodiversity (01.03.2019)
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Journal Article
Synthesis and Biological Evaluation of Novel σ 1 Receptor Ligands for Treating Neuropathic Pain: 6-Hydroxypyridazinones
Cao, Xudong, Chen, Yin, Zhang, Yifang, Lan, Yu, Zhang, Juecheng, Xu, Xiangqing, Qiu, Yinli, Zhao, Song, Liu, Xin, Liu, Bi-Feng, Zhang, Guisen
Published in Journal of medicinal chemistry (14.04.2016)
Published in Journal of medicinal chemistry (14.04.2016)
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Journal Article
Phenyl acetate derivatives, fluorine-substituted on the phenyl group, as rapid recovery hypnotic agents with reflex depression
Zhang, Heng, Xu, Xiangqing, Chen, Yin, Qiu, Yinli, Liu, Xin, Liu, Bi-Feng, Zhang, Guisen
Published in European journal of medicinal chemistry (07.01.2015)
Published in European journal of medicinal chemistry (07.01.2015)
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Journal Article
Pharmacological characterizations of H05, a novel potent serotonin and noradrenaline reuptake inhibitor with moderate 5-HT2A antagonist activity for anti-depression
Xu, Xiangqing, Wei, Yaqin, Guo, Qiang, Zhao, Song, Liu, Zhiqiang, Xiao, Ting, Liu, Yani, Qiu, Yinli, Hou, Yuanyuan, Zhang, Guisen, Wang, Kewei
Published in The Journal of pharmacology and experimental therapeutics (03.04.2018)
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Published in The Journal of pharmacology and experimental therapeutics (03.04.2018)
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