Commercial-Scale Visible Light Trifluoromethylation of 2‑Chlorothiophenol Using CF3I Gas
Harper, Kaid C, Zhang, En-Xuan, Liu, Zhi-Qing, Grieme, Timothy, Towne, Timothy B, Mack, Daniel J, Griffin, Jeremy, Zheng, Song-Yuan, Zhang, Ning-Ning, Gangula, Srinivas, Yuan, Jia-Long, Miller, Robert, Huang, Ping-Zhong, Gage, James, Diwan, Moiz, Ku, Yi-Yin
Published in Organic process research & development (18.02.2022)
Published in Organic process research & development (18.02.2022)
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Journal Article
Development of a Convergent Large-Scale Synthesis for Venetoclax, a First-in-Class BCL‑2 Selective Inhibitor
Ku, Yi-Yin, Chan, Vincent S, Christesen, Alan, Grieme, Timothy, Mulhern, Mathew, Pu, Yu-Ming, Wendt, Michael D
Published in Journal of organic chemistry (19.04.2019)
Published in Journal of organic chemistry (19.04.2019)
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Journal Article
A Highly Efficient Synthesis of a Naphthalenoid Histamine-3 Antagonist
Ku, Yi-Yin, Grieme, Tim, Pu, Yu-Ming, Bhatia, Ashok V.
Published in Advanced synthesis & catalysis (01.08.2009)
Published in Advanced synthesis & catalysis (01.08.2009)
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Journal Article
Mechanistic Evaluation and Solvent-Based Linear Free Energy Relationship in the Alkylation of ABT-199 Using Di-tert-butyl Chloromethyl Phosphate
Harper, Kaid C, Klix, Russel, Pu, Yu-Ming, Henle, Jeremy, Ji, Jianguo, Ku, Yi-Yin
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
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Journal Article
Discovery of Novel Aminotetralines and Aminochromanes as Selective and Competitive Glycine Transporter 1 (GlyT1) Inhibitors
Amberg, Willi, Lange, Udo E. W, Ochse, Michael, Pohlki, Frauke, Behl, Berthold, Relo, Ana Lucia, Hornberger, Wilfried, Hoft, Carolin, Mezler, Mario, Sydor, Jens, Wang, Ying, Zhao, Hongyu, Brewer, Jason T, Dietrich, Justin, Li, Huanqiu, Akritopoulou-Zanze, Irini, Lao, Yanbin, Hannick, Steven M, Ku, Yi-Yin, Vasudevan, Anil
Published in Journal of medicinal chemistry (13.09.2018)
Published in Journal of medicinal chemistry (13.09.2018)
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Journal Article
Expanding the Repertoire for "Large Small Molecules": Prodrug ABBV-167 Efficiently Converts to Venetoclax with Reduced Food Effect in Healthy Volunteers
Salem, Ahmed Hamed, Tao, Zhi-Fu, Bueno, Orlando F, Chen, Jie, Chen, Shuang, Edalji, Rohinton, Elmore, Steven W, Fournier, Keith M, Harper, Kaid C, Hong, Richard, Jenkins, Gary J, Ji, Jianguo, Judge, Russell A, Kalvass, John C, Klix, Russell C, Ku, Yi-Yin, Leverson, Joel D, Marks, Richard A, Marsh, Kennan C, Menon, Rajeev M, Park, Chang H, Phillips, Darren C, Pu, Yu-Ming, Rosenberg, Saul H, Sanzgiri, Yeshwant D, Sheikh, Ahmad Y, Shi, Yi, Stolarik, Deanne, Suleiman, Ahmed A, Wang, Xilu, Zhang, Geoff G Z, Catron, Nathaniel D, Souers, Andrew J
Published in Molecular cancer therapeutics (01.06.2021)
Published in Molecular cancer therapeutics (01.06.2021)
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Journal Article
Scalable Synthesis of a Cis-Substituted Cyclobutyl-Benzothiazole Pyridazinone: Process Development of an Efficient Copper Catalyzed C–N Cross-Coupling Reaction
Kallemeyn, Jeffrey M, Ku, Yi-Yin, Mulhern, Mathew M, Bishop, Richard, Pal, Agnes, Jacob, Legi
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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Journal Article
An efficient copper-catalyzed N-arylation of pyridazinones with a structurally well-defined copper complex
Pu, Yu-Ming, Ku, Yi-Yin, Grieme, Tim, Henry, Rodger, Bhatia, Ashok V.
Published in Tetrahedron letters (09.01.2006)
Published in Tetrahedron letters (09.01.2006)
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Journal Article
An efficient and convergent synthesis of the potent and selective H3 antagonist ABT-239
Ku, Yi-Yin, Pu, Yu-Ming, Grieme, Tim, Sharma, Padam, Bhatia, Ashok V., Cowart, Marlon
Published in Tetrahedron (01.05.2006)
Published in Tetrahedron (01.05.2006)
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Journal Article
An Expedient and Multikilogram Synthesis of a Naphthalenoid H3 Antagonist
Pu, Yu-Ming, Ku, Yi-Yin, Grieme, Timothy, Black, Lawrence A, Bhatia, Ashok V, Cowart, Marlon
Published in Organic process research & development (16.11.2007)
Published in Organic process research & development (16.11.2007)
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Journal Article
The Use of Lewis Acid in the Reaction of Zinc Salts of Indoles and Acyl Chloride
Yang, ChengXi, Patel, Hemantkumar H., Ku, Yi-Yin, Shah, Rajendra, Sawick, David
Published in Synthetic communications (01.06.1997)
Published in Synthetic communications (01.06.1997)
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Journal Article
A Facile and Scaleable Synthesis of ABT-239, A Benzofuranoid H3 Antagonist
Pu, Yu-Ming, Grieme, Timothy, Gupta, Ashok, Plata, Daniel, Bhatia, Ashok V, Cowart, Marlon, Ku, Yi-Yin
Published in Organic process research & development (21.01.2005)
Published in Organic process research & development (21.01.2005)
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Journal Article
4 -[6 -(2 -Aminoethyl )naphthalen -2 -yl ]benzonitriles are potent histamine H3 receptor antagonists with high CNS penetration
BLACK, Lawrence A, NERSESIAN, Diana L, SHARMA, Padam, KU, Yi-Yin, BENNANI, Youssef L, MARSH, Kennan C, MILLER, Thomas R, ESBENSHADE, Timothy A, HANCOCK, Arthur A, COWART, Marlon
Published in Bioorganic & medicinal chemistry letters (01.03.2007)
Published in Bioorganic & medicinal chemistry letters (01.03.2007)
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Journal Article
A simple one-pot procedure for the iminium salt formation: an efficient route to β-arylethylamines
Ku, Yi-Yin, Grieme, Tim, Pu, Yu-Ming, Bhatia, Ashok V., King, Steve A.
Published in Tetrahedron letters (28.02.2005)
Published in Tetrahedron letters (28.02.2005)
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Journal Article
A practical synthesis of chiral propargylic alcohols
Ku, Yi-Yin, Patel, Ramesh R., Elisseou, E Michael, Sawick, David P.
Published in Tetrahedron letters (17.04.1995)
Published in Tetrahedron letters (17.04.1995)
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Journal Article
Asymmetric Synthesis of A-240610.0 via a New Atropselective Approach for Axially Chiral Biaryls with Chirality Transfer
Ku, Yi-Yin, Grieme, Tim, Raje, Prasad, Sharma, Padam, King, Steve A, Morton, Howard E
Published in Journal of the American Chemical Society (24.04.2002)
Published in Journal of the American Chemical Society (24.04.2002)
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