A Survey of the Role of Noncovalent Sulfur Interactions in Drug Design
Beno, Brett R, Yeung, Kap-Sun, Bartberger, Michael D, Pennington, Lewis D, Meanwell, Nicholas A
Published in Journal of medicinal chemistry (11.06.2015)
Published in Journal of medicinal chemistry (11.06.2015)
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Journal Article
meta‐Selective C−H Arylation of Fluoroarenes and Simple Arenes
Liu, Luo‐Yan, Qiao, Jennifer X., Yeung, Kap‐Sun, Ewing, William R., Yu, Jin‐Quan
Published in Angewandte Chemie International Edition (10.08.2020)
Published in Angewandte Chemie International Edition (10.08.2020)
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Journal Article
Ligand-accelerated non-directed C-H functionalization of arenes
Wang, Peng, Verma, Pritha, Xia, Guoqin, Shi, Jun, Qiao, Jennifer X, Tao, Shiwei, Cheng, Peter T W, Poss, Michael A, Farmer, Marcus E, Yeung, Kap-Sun, Yu, Jin-Quan
Published in Nature (London) (23.11.2017)
Published in Nature (London) (23.11.2017)
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Journal Article
Diverse ortho-C(sp2)–H Functionalization of Benzaldehydes Using Transient Directing Groups
Liu, Xi-Hai, Park, Hojoon, Hu, Jun-Hao, Hu, Yan, Zhang, Qun-Liang, Wang, Bao-Long, Sun, Bing, Yeung, Kap-Sun, Zhang, Fang-Lin, Yu, Jin-Quan
Published in Journal of the American Chemical Society (18.01.2017)
Published in Journal of the American Chemical Society (18.01.2017)
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Journal Article
Ligand‐Enabled β‐C(sp3)−H Lactamization of Tosyl‐Protected Aliphatic Amides Using a Practical Oxidant
Zhuang, Zhe, Liu, Shuang, Cheng, Jin‐Tang, Yeung, Kap‐Sun, Qiao, Jennifer X., Meanwell, Nicholas A., Yu, Jin‐Quan
Published in Angewandte Chemie International Edition (22.08.2022)
Published in Angewandte Chemie International Edition (22.08.2022)
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Journal Article
A General Amino Acid Synthesis Enabled by Innate Radical Cross‐Coupling
Ni, Shengyang, Garrido‐Castro, Alberto F., Merchant, Rohan R., de Gruyter, Justine N., Schmitt, Daniel C., Mousseau, James J., Gallego, Gary M., Yang, Shouliang, Collins, Michael R., Qiao, Jennifer X., Yeung, Kap‐Sun, Langley, David R., Poss, Michael A., Scola, Paul M., Qin, Tian, Baran, Phil S.
Published in Angewandte Chemie International Edition (26.10.2018)
Published in Angewandte Chemie International Edition (26.10.2018)
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Journal Article
Rational Development of Remote C−H Functionalization of Biphenyl: Experimental and Computational Studies
Fan, Zhoulong, Bay, Katherine L., Chen, Xiangyang, Zhuang, Zhe, Park, Han Seul, Yeung, Kap‐Sun, Houk, K. N., Yu, Jin‐Quan
Published in Angewandte Chemie International Edition (16.03.2020)
Published in Angewandte Chemie International Edition (16.03.2020)
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Journal Article
Remote C−H Olefination of Heterocyclic Biaryls Enabled by Reversibly Bound Templates
Liu, Luo‐Yan, Fan, Zhoulong, Hoque, Md Emdadul, Qian, Shaoqun, Meng, Guangrong, Chekshin, Nikita, Tanaka, Keita, Qiao, Jennifer X., Yeung, Kap‐Sun, Yu, Jin‐Quan
Published in Angewandte Chemie International Edition (11.09.2023)
Published in Angewandte Chemie International Edition (11.09.2023)
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Journal Article
Special issue of Medicinal Chemistry Research in honor of Dr. Nicholas A. Meanwell
Kadow, John F., Yeung, Kap-Sun, Murali Dhar, T. G.
Published in Medicinal chemistry research (01.07.2023)
Published in Medicinal chemistry research (01.07.2023)
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Journal Article
PdII‐Catalyzed Enantioselective C(sp3)–H Arylation of Cyclobutyl Ketones Using a Chiral Transient Directing Group
Xiao, Li‐Jun, Hong, Kai, Luo, Fan, Hu, Liang, Ewing, William R., Yeung, Kap‐Sun, Yu, Jin‐Quan
Published in Angewandte Chemie International Edition (08.06.2020)
Published in Angewandte Chemie International Edition (08.06.2020)
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Journal Article
Discovery and Preclinical Characterization of the Cyclopropylindolobenzazepine BMS-791325, A Potent Allosteric Inhibitor of the Hepatitis C Virus NS5B Polymerase
Gentles, Robert G., Ding, Min, Bender, John A., Bergstrom, Carl P., Grant-Young, Katharine, Hewawasam, Piyasena, Hudyma, Thomas, Martin, Scott, Nickel, Andrew, Regueiro-Ren, Alicia, Tu, Yong, Yang, Zhong, Yeung, Kap-Sun, Zheng, Xiaofan, Chao, Sam, Sun, Jung-Hui, Beno, Brett R., Camac, Daniel M., Chang, Chong-Hwan, Gao, Mian, Morin, Paul E., Sheriff, Steven, Tredup, Jeff, Wan, John, Witmer, Mark R., Xie, Dianlin, Hanumegowda, Umesh, Knipe, Jay, Mosure, Kathy, Santone, Kenneth S., Parker, Dawn D., Zhuo, Xiaoliang, Lemm, Julie, Liu, Mengping, Pelosi, Lenore, Rigat, Karen, Voss, Stacey, Wang, Yi, Wang, Ying-Kai, Colonno, Richard J., Gao, Min, Roberts, Susan B., Gao, Qi, Ng, Alicia, Meanwell, Nicholas A, Kadow, John F.
Published in Journal of medicinal chemistry (13.03.2014)
Published in Journal of medicinal chemistry (13.03.2014)
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Journal Article
Discovery of a Hepatitis C Virus NS5B Replicase Palm Site Allosteric Inhibitor (BMS-929075) Advanced to Phase 1 Clinical Studies
Yeung, Kap-Sun, Beno, Brett R, Parcella, Kyle, Bender, John A, Grant-Young, Katherine A, Nickel, Andrew, Gunaga, Prashantha, Anjanappa, Prakash, Bora, Rajesh Onkardas, Selvakumar, Kumaravel, Rigat, Karen, Wang, Ying-Kai, Liu, Mengping, Lemm, Julie, Mosure, Kathy, Sheriff, Steven, Wan, Changhong, Witmer, Mark, Kish, Kevin, Hanumegowda, Umesh, Zhuo, Xiaoliang, Shu, Yue-Zhong, Parker, Dawn, Haskell, Roy, Ng, Alicia, Gao, Qi, Colston, Elizabeth, Raybon, Joseph, Grasela, Dennis M, Santone, Kenneth, Gao, Min, Meanwell, Nicholas A, Sinz, Michael, Soars, Matthew G, Knipe, Jay O, Roberts, Susan B, Kadow, John F
Published in Journal of medicinal chemistry (25.05.2017)
Published in Journal of medicinal chemistry (25.05.2017)
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Journal Article
Inhibitors of HIV-1 attachment. Part 7: Indole-7-carboxamides as potent and orally bioavailable antiviral agents
Yeung, Kap-Sun, Qiu, Zhilei, Xue, Quifen, Fang, Haiquan, Yang, Zheng, Zadjura, Lisa, D’Arienzo, Celia J., Eggers, Betsy J., Riccardi, Keith, Shi, Pei-Yong, Gong, Yi-Fei, Browning, Marc R., Gao, Qi, Hansel, Steven, Santone, Kenneth, Lin, Ping-Fang, Meanwell, Nicholas A., Kadow, John F.
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
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Journal Article
meta‐Selective C−H Arylation of Fluoroarenes and Simple Arenes
Liu, Luo‐Yan, Qiao, Jennifer X., Yeung, Kap‐Sun, Ewing, William R., Yu, Jin‐Quan
Published in Angewandte Chemie (10.08.2020)
Published in Angewandte Chemie (10.08.2020)
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Journal Article
Inhibitors of HIV-1 attachment. Part 8: The effect of C7-heteroaryl substitution on the potency, and in vitro and in vivo profiles of indole-based inhibitors
Yeung, Kap-Sun, Qiu, Zhilei, Yin, Zhiwei, Trehan, Ashok, Fang, Haiquan, Pearce, Bradley, Yang, Zheng, Zadjura, Lisa, D’Arienzo, Celia J., Riccardi, Keith, Shi, Pei-Yong, Spicer, Timothy P., Gong, Yi-Fei, Browning, Marc R., Hansel, Steven, Santone, Kenneth, Barker, Jonathan, Coulter, Thomas, Lin, Ping-Fang, Meanwell, Nicholas A., Kadow, John F.
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
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Journal Article
Pd(II)-Catalyzed Enantioselective C(sp3)−H Arylation of Cyclobutyl Ketones Using a Chiral Transient Directing Group
Xiao, Li-Jun, Hong, Kai, Luo, Fan, Hu, Liang, Ewing, William R., Yeung, Kap-Sun, Yu, Jin-Quan
Published in Angewandte Chemie International Edition (08.06.2020)
Published in Angewandte Chemie International Edition (08.06.2020)
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