Identification and characterization of noncalcemic, tissue-selective, nonsecosteroidal vitamin D receptor modulators
Ma, Yanfei, Khalifa, Berket, Yee, Ying K, Lu, Jianfen, Memezawa, Ai, Savkur, Rajesh S, Yamamoto, Yoko, Chintalacharuvu, Subba R, Yamaoka, Kazuyoshi, Stayrook, Keith R, Bramlett, Kelli S, Zeng, Qing Q, Chandrasekhar, Srinivasan, Yu, Xiao-Peng, Linebarger, Jared H, Iturria, Stephen J, Burris, Thomas P, Kato, Shigeaki, Chin, William W, Nagpal, Sunil
Published in The Journal of clinical investigation (01.04.2006)
Published in The Journal of clinical investigation (01.04.2006)
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Journal Article
Novel 3-Aryl Indoles as Progesterone Receptor Antagonists for Uterine Fibroids
Richardson, Timothy I, Clarke, Christian A, Yu, Kuo-Long, Yee, Ying K, Bleisch, Thomas J, Lopez, Jose E, Jones, Scott A, Hughes, Norman E, Muehl, Brian S, Lugar, Charles W, Moore, Terry L, Shetler, Pamela K, Zink, Richard W, Osborne, John J, Montrose-Rafizadeh, Chahrzad, Patel, Nita, Geiser, Andrew G, Galvin, Rachelle J. Sells, Dodge, Jeffrey A
Published in ACS medicinal chemistry letters (10.02.2011)
Published in ACS medicinal chemistry letters (10.02.2011)
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Journal Article
Vitamin D receptor modulators for inflammation and cancer
Yee, Ying K, Chintalacharuvu, Subba R, Lu, Jianfen, Nagpal, Sunil
Published in Mini reviews in medicinal chemistry (01.08.2005)
Published in Mini reviews in medicinal chemistry (01.08.2005)
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Journal Article
Vitamin D receptor as a drug discovery target
Pinette, Karen V, Yee, Ying K, Amegadzie, Bernard Y, Nagpal, Sunil
Published in Mini reviews in medicinal chemistry (01.05.2003)
Published in Mini reviews in medicinal chemistry (01.05.2003)
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Journal Article
Anthranilamide inhibitors of factor Xa
Mendel, David, Marquart, Angela L., Joseph, Sajan, Waid, Philip, Yee, Ying K., Tebbe, Anne Louise, Ratz, Andrew M., Herron, David K., Goodson, Theodore, Masters, John J., Franciskovich, Jeffry B., Tinsley, Jennifer M., Wiley, Michael R., Weir, Leonard C., Kyle, Jeffrey A., Klimkowski, Valentine J., Smith, Gerald F., Towner, Richard D., Froelich, Larry L., Buben, John, Craft, Trelia J.
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Journal Article
A novel series of selective leukotriene antagonists: exploration and optimization of the acidic region in 1,6-disubstituted indoles and indazoles
Yee, Ying K, Bernstein, Peter R, Adams, Edward J, Brown, Frederick J, Cronk, Laura A, Hebbel, Kevin C, Vacek, Edward P, Krell, Robert D, Snyder, David W
Published in Journal of medicinal chemistry (01.09.1990)
Published in Journal of medicinal chemistry (01.09.1990)
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Journal Article
Evolution of a series of peptidoleukotriene antagonists: synthesis and structure-activity relationships of 1,6-disubstituted indoles and indazoles
Brown, Frederick J, Yee, Ying K, Cronk, Laura A, Hebbel, Kevin C, Krell, Robert D, Snyder, David W
Published in Journal of medicinal chemistry (01.06.1990)
Published in Journal of medicinal chemistry (01.06.1990)
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Journal Article
N 2-Aroylanthranilamide Inhibitors of Human Factor Xa
Yee, Ying K, Tebbe, Anne Louise, Linebarger, Jared H, Beight, Douglas W, Craft, Trelia J, Gifford-Moore, Donetta, Goodson, Theodore, Herron, David K, Klimkowski, Valentine J, Kyle, Jeffrey A, Sawyer, J. Scott, Smith, Gerald F, Tinsley, Jennifer M, Towner, Richard D, Weir, Leonard, Wiley, Michael R
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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Journal Article
Non-Amidine-Containing 1,2-Dibenzamidobenzene Inhibitors of Human Factor Xa with Potent Anticoagulant and Antithrombotic Activity
Masters, John J, Franciskovich, Jeffry B, Tinsley, Jennifer M, Campbell, Charles, Campbell, Jack B, Craft, Trelia J, Froelich, Larry L, Gifford-Moore, Donetta S, Hay, Lynne A, Herron, David K, Klimkowski, Valentine J, Kurz, Kenneth D, Metz, James T, Ratz, Andrew M, Shuman, Robert T, Smith, Gerald F, Smith, Tommy, Towner, Richard D, Wiley, Michael R, Wilson, Alex, Yee, Ying K
Published in Journal of medicinal chemistry (01.06.2000)
Published in Journal of medicinal chemistry (01.06.2000)
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Journal Article
Hydroxyacetophenone-derived antagonists of the peptidoleukotrienes
Brown, Frederick J, Bernstein, Peter R, Cronk, Laura A, Dosset, David L, Hebbel, Kevin C, Maduskuie, Thomas P, Shapiro, Howard S, Vacek, Edward P, Yee, Ying K
Published in Journal of medicinal chemistry (01.04.1989)
Published in Journal of medicinal chemistry (01.04.1989)
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Journal Article
Identification of Essential Residues for the Catalytic Function of 85-kDa Cytosolic Phospholipase A2
Pickard, Richard T., Chiou, X. Grace, Strifler, Beth A., DeFelippis, Michael R., Hyslop, Paul A., Tebbe, Ann Louise, Yee, Ying K., Reynolds, Laure J., Dennis, Edward A., Kramer, Ruth M., Sharp, John D.
Published in The Journal of biological chemistry (09.08.1996)
Published in The Journal of biological chemistry (09.08.1996)
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Journal Article
Biochemical and pharmacological characterization of the binding of the selective peptide-leukotriene antagonist, 3H-ICI 198,615, to leukotriene D4 receptors in guinea-pig lung membranes
Aharony, D, Falcone, R C, Yee, Y K, Hesp, B, Giles, R E, Krell, R D
Published in Annals of the New York Academy of Sciences (01.04.1988)
Published in Annals of the New York Academy of Sciences (01.04.1988)
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Journal Article
Synthesis and in vitro LTD4 antagonist activity of bicyclic and monocyclic cyclopentylurethane and cyclopentylacetamide N-arylsulfonyl amides
Matassa, Victor G, Brown, Frederick J, Bernstein, Peter R, Shapiro, Howard S, Maduskuie, Thomas P, Cronk, Laura A, Vacek, Edward P, Yee, Ying K, Snyder, David W
Published in Journal of medicinal chemistry (01.09.1990)
Published in Journal of medicinal chemistry (01.09.1990)
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Journal Article
Total synthesis of dl-lycoramine
Schultz, Arthur G, Yee, Ying K, Berger, Mitchell H
Published in Journal of the American Chemical Society (01.11.1977)
Published in Journal of the American Chemical Society (01.11.1977)
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Journal Article
Identification of essential residues for the catalytic function of 85-kDa cytosolic phospholipase A2. Probing the role of histidine, aspartic acid, cysteine, and arginine
Pickard, R T, Chiou, X G, Strifler, B A, DeFelippis, M R, Hyslop, P A, Tebbe, A L, Yee, Y K, Reynolds, L J, Dennis, E A, Kramer, R M, Sharp, J D
Published in The Journal of biological chemistry (09.08.1996)
Published in The Journal of biological chemistry (09.08.1996)
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Journal Article
N(2)-Aroylanthranilamide inhibitors of human factor Xa
Yee, Y K, Tebbe, A L, Linebarger, J H, Beight, D W, Craft, T J, Gifford-Moore, D, Goodson, Jr, T, Herron, D K, Klimkowski, V J, Kyle, J A, Sawyer, J S, Smith, G F, Tinsley, J M, Towner, R D, Weir, L, Wiley, M R
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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Journal Article