Initial SAR studies on apamin-displacing 2-aminothiazole blockers of calcium-activated small conductance potassium channels
Gentles, Robert G., Grant-Young, Katherine, Hu, Shuanghua, Huang, Yazhong, Poss, Michael A., Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, C. David, Harden, David G.
Published in Bioorganic & medicinal chemistry (01.10.2008)
Published in Bioorganic & medicinal chemistry (01.10.2008)
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Journal Article
Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine KCa channel blockers
GENTLES, Robert G, SHUANGHUA HU, HARDEN, David G, YAZHONG HUANG, GRANT-YOUNG, Katherine, POSS, Michael A, ANDRES, Charles, FIEDLER, Tracey, KNOX, Ronald, LODGE, Nicholas, WEAVER, C. David
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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Journal Article
Identification of a Potent and Selective 5-HT6 Antagonist: One-Step Synthesis of (E)-3-(Benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin- 4-ylidenamine from 2-(Benzenesulfonyl)-3,3- bis(methylsulfanyl)acrylonitrile
Wu, Yong-Jin, He, Huan, Hu, Shuanghua, Huang, Yazhong, Scola, Paul M, Grant-Young, Katharine, Bertekap, Robert L, Wu, Dedong, Gao, Qi, Li, Yi, Klakouski, Cheryl, Westphal, Ryan S
Published in Journal of medicinal chemistry (06.11.2003)
Published in Journal of medicinal chemistry (06.11.2003)
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Journal Article
Novel Dihydropyrazine Analogues as NPY Antagonists
Sit, Sing-Yuen, Huang, Yazhong, Antal-Zimanyi, Ildiko, Ward, Sally, Poindexter, Graham S
Published in Bioorganic & medicinal chemistry letters (11.02.2002)
Published in Bioorganic & medicinal chemistry letters (11.02.2002)
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Journal Article
Discovery of D1 Dopamine Receptor Positive Allosteric Modulators: Characterization of Pharmacology and Identification of Residues that Regulate Species Selectivity
Lewis, Martin A, Hunihan, Lisa, Watson, John, Gentles, Robert G, Hu, Shuanghua, Huang, Yazhong, Bronson, Joanne, Macor, John E, Beno, Brett R, Ferrante, Meredith, Hendricson, Adam, Knox, Ronald J, Molski, Thaddeus F, Kong, Yan, Cvijic, Mary Ellen, Rockwell, Kristin L, Weed, Michael R, Cacace, Angela M, Westphal, Ryan S, Alt, Andrew, Brown, Jeffrey M
Published in The Journal of pharmacology and experimental therapeutics (01.09.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2015)
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Journal Article
Structure activity relationship studies on chemically non-reactive glycine sulfonamide inhibitors of diacylglycerol lipase
Chupak, Louis S., Zheng, Xiaofan, Hu, Shuanghua, Huang, Yazhong, Ding, Min, Lewis, Martin A., Westphal, Ryan S., Blat, Yuval, McClure, Andrea, Gentles, Robert G.
Published in Bioorganic & medicinal chemistry (01.04.2016)
Published in Bioorganic & medicinal chemistry (01.04.2016)
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Journal Article
Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT6 antagonists
Hu, Shuanghua, Huang, Yazhong, Wu, Yong-Jin, He, Huan, Grant-Young, Katherine A., Bertekap, Robert L., Whiterock, Valerie, Brassil, Patrick, Lentz, Kimberley, Sivaprakasam, Prasanna, Langley, David R., Westphal, Ryan S., Scola, Paul M.
Published in Bioorganic & medicinal chemistry (01.03.2014)
Published in Bioorganic & medicinal chemistry (01.03.2014)
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Journal Article
Heterocyclic modification of a novel bicyclo[3.1.0]hexane NPY1 receptor antagonist
Luo, Guanglin, Chen, Ling, Hu, Shuanghua, Huang, Yazhong, Mattson, Gail, Iben, Lawrence G., Russell, John W., Clarke, Wendy J., Hogan, John B., Antal-Zimanyi, Ildiko, Poindexter, Graham S.
Published in Bioorganic & medicinal chemistry letters (01.07.2013)
Published in Bioorganic & medicinal chemistry letters (01.07.2013)
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Journal Article
Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine K Ca channel blockers
Gentles, Robert G., Hu, Shuanghua, Huang, Yazhong, Grant-Young, Katherine, Poss, Michael A., Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, C. David, Harden, David G.
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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Journal Article
Preliminary SAR studies on non-apamin-displacing 4- (aminomethylaryl)pyrrazolopyrimidine K sub(Ca) channel blockers
Gentles, Robert G, Hu, Shuanghua, Huang, Yazhong, Grant-Young, Katherine, Poss, Michael A, Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, CDavid, Harden, David G
Published in Bioorganic & medicinal chemistry (01.10.2008)
Published in Bioorganic & medicinal chemistry (01.10.2008)
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Journal Article
Discovery of a Novel Class of Bicyclo[3.1.0]hexanylpiperazines as Noncompetitive Neuropeptide Y Y1 Antagonists
Hu, Shuanghua, Huang, Yazhong, Deshpande, Milind, Luo, Guanglin, Bruce, Marc A, Chen, Ling, Mattson, Gail, Iben, Lawrence G, Zhang, Jie, Russell, John W, Clarke, Wendy J, Hogan, John B, Ortiz, Astrid, Flint, Oliver, Henwood, Andrew, Gao, Qi, Antal-Zimanyi, Ildiko, Poindexter, Graham S
Published in ACS medicinal chemistry letters (08.03.2012)
Published in ACS medicinal chemistry letters (08.03.2012)
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Journal Article
Naphthyridinone compounds useful as T cell activators
Ding, Min, Wichroski, Michael, Chupak, Louis S, Mercer, Stephen E, Velaparthi, Upender, Mcdonald, Ivar M, Martin, Scott W, Zheng, Xiaofan, Huang, Yazhong, Olson, Richard E, Gentles, Robert G
Year of Publication 09.01.2024
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Year of Publication 09.01.2024
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