Enantio- and Diastereoselective Michael Reaction of 1,3-Dicarbonyl Compounds to Nitroolefins Catalyzed by a Bifunctional Thiourea
Okino, Tomotaka, Hoashi, Yasutaka, Furukawa, Tomihiro, Xu, Xuenong, Takemoto, Yoshiji
Published in Journal of the American Chemical Society (12.01.2005)
Published in Journal of the American Chemical Society (12.01.2005)
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Anti-tumor activity of KNTC2 siRNA in orthotopic tumor model mice of hepatocellular carcinoma
Makita, Yukimasa, Murata, Shumpei, Katou, Yoshiki, Kikuchi, Kuniko, Uejima, Hiroshi, Teratani, Mika, Hoashi, Yasutaka, Kenjo, Eriya, Matsumoto, Satoru, Nogami, Masahiro, Otake, Kentaro, Kawamata, Yuji
Published in Biochemical and biophysical research communications (04.11.2017)
Published in Biochemical and biophysical research communications (04.11.2017)
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Thiourea-Catalyzed Asymmetric Michael Addition of Activated Methylene Compounds to α,β-Unsaturated Imides: Dual Activation of Imide by Intra- and Intermolecular Hydrogen Bonding
Inokuma, Tsubasa, Hoashi, Yasutaka, Takemoto, Yoshiji
Published in Journal of the American Chemical Society (26.07.2006)
Published in Journal of the American Chemical Society (26.07.2006)
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Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists
Kojima, Takuto, Mochizuki, Michiyo, Takai, Takafumi, Hoashi, Yasutaka, Morimoto, Sachie, Seto, Masaki, Nakamura, Minoru, Kobayashi, Katsumi, Sako, Yuu, Tanaka, Maiko, Kanzaki, Naoyuki, Kosugi, Yohei, Yano, Takahiko, Aso, Kazuyoshi
Published in Bioorganic & medicinal chemistry (15.05.2018)
Published in Bioorganic & medicinal chemistry (15.05.2018)
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Synthesis of pyrazolo[1,5-a]pyridines by thermal intramolecular cyclization
Hoashi, Yasutaka, Takai, Takafumi, Kotani, Etsuo, Koike, Tatsuki
Published in Tetrahedron letters (24.04.2013)
Published in Tetrahedron letters (24.04.2013)
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Discovery of novel 5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridine derivatives as γ-secretase modulators
Takai, Takafumi, Hoashi, Yasutaka, Tomata, Yoshihide, Morimoto, Sachie, Nakamura, Minoru, Watanabe, Tomomichi, Igari, Tomoko, Koike, Tatsuki
Published in Bioorganic & medicinal chemistry letters (01.10.2015)
Published in Bioorganic & medicinal chemistry letters (01.10.2015)
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1,6-Dihydro-2H-indeno[5,4-b]furan Derivatives: Design, Synthesis, and Pharmacological Characterization of a Novel Class of Highly Potent MT2-Selective Agonists
Koike, Tatsuki, Hoashi, Yasutaka, Takai, Takafumi, Nakayama, Masaharu, Yukuhiro, Nobuhito, Ishikawa, Takashi, Hirai, Keisuke, Uchikawa, Osamu
Published in Journal of medicinal chemistry (12.05.2011)
Published in Journal of medicinal chemistry (12.05.2011)
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Design and synthesis of piperazine derivatives as a novel class of gamma-secretase modulators that selectively lower A beta(42) production
Takai, Takafumi, Koike, Tatsuki, Honda, Eiji, Kajita, Yuichi, Nakamura, Minoru, Morimoto, Sachie, Hoashi, Yasutaka, Kamata, Makoto, Watanabe, Tomomichi, Igari, Tomoko, Terauchi, Jun
Published in Bioorganic & medicinal chemistry (01.05.2015)
Published in Bioorganic & medicinal chemistry (01.05.2015)
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Design and synthesis of piperazine derivatives as a novel class of γ-secretase modulators that selectively lower Aβ42 production
Takai, Takafumi, Koike, Tatsuki, Honda, Eiji, Kajita, Yuichi, Nakamura, Minoru, Morimoto, Sachie, Hoashi, Yasutaka, Kamata, Makoto, Watanabe, Tomomichi, Igari, Tomoko, Terauchi, Jun
Published in Bioorganic & medicinal chemistry (01.05.2015)
Published in Bioorganic & medicinal chemistry (01.05.2015)
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