Pseudoirreversible inhibition elicits persistent efficacy of a sphingosine 1-phosphate receptor 1 antagonist
Maruyama, Yuya, Ohsawa, Yusuke, Suzuki, Takayuki, Yamauchi, Yuko, Ohno, Kohsuke, Inoue, Hitoshi, Yamamoto, Akitoshi, Hayashi, Morimichi, Okuhara, Yuji, Muramatsu, Wataru, Namiki, Kano, Hagiwara, Naho, Miyauchi, Maki, Miyao, Takahisa, Ishikawa, Tatsuya, Horie, Kenta, Hayama, Mio, Akiyama, Nobuko, Hirokawa, Takatsugu, Akiyama, Taishin
Published in Nature communications (19.07.2024)
Published in Nature communications (19.07.2024)
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Involvement of CYP2A6 in the Formation of a Novel Metabolite, 3-Hydroxypilocarpine, from Pilocarpine in Human Liver Microsomes
ENDO, Takuro, BAN, Masaaki, HIRATA, Kazuma, YAMAMOTO, Akitoshi, HARA, Yoshiki, MOMOSE, Yasunori
Published in Drug metabolism and disposition (01.03.2007)
Published in Drug metabolism and disposition (01.03.2007)
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Identification of N-acyl-N-indanyl-α-phenylglycinamides as selective TRPM8 antagonists designed to mitigate the risk of adverse effects
Kobayashi, Jun-ichi, Hirasawa, Hideaki, Fujimori, Yoshikazu, Nakanishi, Osamu, Kamada, Noboru, Ikeda, Tetsuya, Yamamoto, Akitoshi, Kanbe, Hiroki
Published in Bioorganic & medicinal chemistry (15.01.2021)
Published in Bioorganic & medicinal chemistry (15.01.2021)
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スフィンゴシン1-リン酸受容体-1拮抗薬は偽非可逆性の阻害作用により持続的な作用を示す
丸山, 祐哉, 大澤, 雄亮, 鈴木, 孝幸, 山内, 裕子, 大野, 孝介, 井上, 仁史, 山本, 明俊, 林, 守道, 宮内, 真紀, 広川, 貴次, 秋山, 泰身
Published in 日本薬理学会年会要旨集 (2022)
Published in 日本薬理学会年会要旨集 (2022)
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A pseudo-irreversible inhibition elicits a persistent effect of the sphingosine 1-phosphate receptor-1 antagonist
Maruyama, Yuya, Ohsawa, Yusuke, Suzuki, Takayuki, Yamauchi, Yuko, Ohno, Kohsuke, Inoue, Hitoshi, Yamamoto, Akitoshi, Hayashi, Morimichi, Miyauchi, Maki, Hirokawa, Takatsugu, Akiyama, Taishin
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2022)
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2022)
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Vibro-Fluidization of Very Fine Particles
Mori, Shigekatsu, Haruta, Takeo, Yamamoto, Akitoshi, Yamada, Ikuho, Mizutani, Eiichi
Published in KAGAKU KOGAKU RONBUNSHU (10.09.1989)
Published in KAGAKU KOGAKU RONBUNSHU (10.09.1989)
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Vibro-fluidization of very fine particles
Mori, Shigekatsu, Haruta, Takeo, Yamamoto, Akitoshi, Yamada, Ikuho, Mizutani, Eiichi
Published in Kagaku kōgaku ronbunshū (1989)
Published in Kagaku kōgaku ronbunshū (1989)
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Ferroelectricity in {N(CH3)4}2 CoCl4
Sawada, Shozo, Shiroishi, Yoshihiro, Yamamoto, Akitoshi, Takashige, Masaaki, Matsuo, Mutsumi
Published in Physics letters. A (10.07.1978)
Published in Physics letters. A (10.07.1978)
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