Search Results - "YAMAKI, Susumu" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery of ASP6918, a KRAS G12C inhibitor: Synthesis and structure-activity relationships of 1-{2,7-diazaspiro[3.5]non-2-yl} prop-2-en-1-one derivatives as covalent inhibitors with good potency and oral activity for the treatment of solid tumors

Discovery of ASP6918, a KRAS G12C inhibitor: Synthesis and structure-activity relationships of 1-{2,7-diazaspiro[3.5]non-2-yl} prop-2-en-1-one derivatives as covalent inhibitors with good potency and oral activity for the treatment of solid tumors

by Imaizumi, Tomoyoshi, Shimada, Itsuro, Satake, Yoshiki, Yamaki, Susumu, Koike, Takanori, Nigawara, Takahiro, Kaneko, Osamu, Amano, Yasushi, Mori, Kenichi, Yamanaka, Yosuke, Nakayama, Ayako, Nishizono, Yoshihiro, Shimazaki, Masashi, Nagashima, Takeyuki, Kuramoto, Kazuyuki
Published in Bioorganic & medicinal chemistry (15.01.2024)

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Journal Article

Synthesis and pharmacological evaluation of glycine amide derivatives as novel vascular adhesion protein-1 inhibitors without CYP3A4 and CYP2C19 inhibition

Synthesis and pharmacological evaluation of glycine amide derivatives as novel vascular adhesion protein-1 inhibitors without CYP3A4 and CYP2C19 inhibition

by Yamaki, Susumu, Koga, Yuji, Nagashima, Akira, Kondo, Mitsuhiro, Shimada, Yoshiaki, Kadono, Keitaro, Moritomo, Ayako, Yoshihara, Kosei
Published in Bioorganic & medicinal chemistry (01.08.2017)

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Journal Article

Discovery and biological evaluation of novel pyrazolopyridine derivatives as potent and orally available PI3Kδ inhibitors

Discovery and biological evaluation of novel pyrazolopyridine derivatives as potent and orally available PI3Kδ inhibitors

by Hamajima, Toshihiro, Takahashi, Fumie, Kato, Koji, Mukoyoshi, Koichiro, Yoshihara, Kousei, Yamaki, Susumu, Sugano, Yukihito, Moritomo, Ayako, Yamagami, Kaoru, Yokoo, Koji, Fukahori, Hidehiko
Published in Bioorganic & medicinal chemistry (15.05.2018)

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Journal Article

Synthesis and structure activity relationships of carbamimidoylcarbamate derivatives as novel vascular adhesion protein-1 inhibitors

Synthesis and structure activity relationships of carbamimidoylcarbamate derivatives as novel vascular adhesion protein-1 inhibitors

by Yamaki, Susumu, Yamada, Hiroyoshi, Nagashima, Akira, Kondo, Mitsuhiro, Shimada, Yoshiaki, Kadono, Keitaro, Yoshihara, Kosei
Published in Bioorganic & medicinal chemistry (01.11.2017)

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Journal Article

Synthesis and structure activity relationships of glycine amide derivatives as novel Vascular Adhesion Protein-1 inhibitors

Synthesis and structure activity relationships of glycine amide derivatives as novel Vascular Adhesion Protein-1 inhibitors

by Yamaki, Susumu, Suzuki, Daisuke, Fujiyasu, Jiro, Neya, Masahiro, Nagashima, Akira, Kondo, Mitsuhiro, Akabane, Takafumi, Kadono, Keitaro, Moritomo, Ayako, Yoshihara, Kosei
Published in Bioorganic & medicinal chemistry (01.01.2017)

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Journal Article

Optimization and in vivo evaluation of pyrazolopyridines as a potent and selective PI3Kδ inhibitor

Optimization and in vivo evaluation of pyrazolopyridines as a potent and selective PI3Kδ inhibitor

by Hamajima, Toshihiro, Takahashi, Fumie, Kato, Koji, Sugano, Yukihito, Yamaki, Susumu, Moritomo, Ayako, Kubo, Satoshi, Nakamura, Koji, Yamagami, Kaoru, Hamakawa, Nozomu, Yokoo, Koji, Fukahori, Hidehiko
Published in Bioorganic & medicinal chemistry (07.08.2018)

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Journal Article

Optimization of 5,6,7,8-tetrahydropyrido[4,3-d]pyrimidines to generate a highly selective PI3Kδ inhibitor

Optimization of 5,6,7,8-tetrahydropyrido[4,3-d]pyrimidines to generate a highly selective PI3Kδ inhibitor

by Hamajima, Toshihiro, Takahashi, Fumie, Kato, Koji, Sugano, Yukihito, Yamaki, Susumu, Suzuki, Daisuke, Moritomo, Ayako, Kubo, Satoshi, Nakamura, Koji, Yamagami, Kaoru, Yokoo, Koji, Fukahori, Hidehiko
Published in Bioorganic & medicinal chemistry (15.03.2019)

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Journal Article

축환 피리다진 화합물

축환 피리다진 화합물

by KURIWAKI IKUMI, NAKAMURA AKIHIKO, WASHIO TAKUYA, KURAMOTO KAZUYUKI, KAMIKUBO TAKASHI, YAMASHITA YUMI, KOIZUMI YUKA, INAGAKI YUSUKE, TOMIYAMA HIROSHI, YAMAKI SUSUMU, SABA KENGO, KOIKE TAKANORI, MAEDA JUNKO, TOYA HIROKI, IWAI YOSHINORI
Year of Publication 07.05.2024

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Patent

이고리형 1,4-디아제판온 및 이의 치료적 용도

이고리형 1,4-디아제판온 및 이의 치료적 용도

by EVANS CHRIS, SEKIOKA RYUICHI, KURIWAKI IKUMI, MORGAN BRADLEY P, COLLIBEE SCOTT, KOIZUMI YUKA, HONJO ERIKO, YAMAKI SUSUMU, TSUCHIYA KAZUYUKI, KUROSAKI TOSHIO, LU PU PING, WANG WENYUE, MAKINO TAKUYA, KATOH NAOTO, YAMASAKI MAKOTO
Year of Publication 22.08.2023

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Patent

ANNULATED PYRIDAZINE COMPOUND

ANNULATED PYRIDAZINE COMPOUND

by WASHIO, Takuya, KOIZUMI, Yuka, KURAMOTO, Kazuyuki, YAMAKI, Susumu, TOMIYAMA, Hiroshi, INAGAKI, Yusuke, KOIKE, Takanori, MAEDA, Junko, NAKAMURA, Akihiko, TOYA, Hiroki, KURIWAKI, Ikumi, IWAI, Yoshinori, SABA, Kengo, YAMASHITA, Yumi, KAMIKUBO, Takashi
Year of Publication 26.01.2023

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Patent

SUBSTITUTED PYRIDAZINE COMPOUND

SUBSTITUTED PYRIDAZINE COMPOUND

by NEGORO, Kenji, SABA, Kengo, IIDA, Maiko, KOIZUMI, Yuka, YAMAKI, Susumu, INAGAKI, Yusuke, KOIKE, Takanori, MAEDA, Junko, KAMIKUBO, Takashi, NIGAWARA, Takahiro, KURIWAKI, Ikumi, SHISHIKURA, Junichi
Year of Publication 30.09.2021

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Patent

퀴나졸린 화합물

퀴나졸린 화합물

by ARAKAWA KEISUKE, KURAMOTO KAZUYUKI, NIGAWARA TAKAHIRO, SHIMADA ITSURO, ABE TOMOAKI, SATAKE YOSHIKI, AKAIWA MICHINORI, SHIMAZAKI MASASHI, WATANABE KAZUSHI, ARAKI TAKANOBU, YAMAKI SUSUMU, KUNIKAWA SHIGEKI, KOIKE TAKANORI, IMAIZUMI TOMOYOSHI
Year of Publication 08.10.2019

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Patent

QUINAZOLINE COMPOUND

QUINAZOLINE COMPOUND

by ABE, Tomoaki, KURAMOTO, Kazuyuki, AKAIWA, Michinori, YAMAKI, Susumu, KOIKE, Takanori, SATAKE, Yoshiki, NIGAWARA, Takahiro, SHIMADA, Itsuro, IMAIZUMI, Tomoyoshi, ARAKI, Takanobu, ARAKAWA, Keisuke, WATANABE, Kazushi, SHIMAZAKI, Masashi, KUNIKAWA, Shigeki
Year of Publication 09.08.2018

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Patent

GUANIDINOBENZOIC ACID ESTER COMPOUND

GUANIDINOBENZOIC ACID ESTER COMPOUND

by KANEKO OSAMU, SATOU TOMOHKI, SASAMURA SATOSHI, FUJIYASU JIRO, YAMAKI SUSUMU, URANO YASUHARU, ASANO TORU, KOIKE YUKA, IMAIZUMI TOMOYOSHI
Year of Publication 23.11.2015

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Patent

테트라히드로이소퀴놀린 유도체

테트라히드로이소퀴놀린 유도체

by SATO IPPEI, MATSUSHIMA YUJI, TANAKA HIROAKI, MALIK FADY, KAMIKUBO TAKASHI, KIYOHARA HIROSHI, COLLIBEE SCOTT EMILE, ASHCRAFT LUKE, WARRINGTON JEFFREY MICHAEL, SAITO TOMOYUKI, SHIINA YASUHIRO, GARARD MARC, YAMAKI SUSUMU, MORGAN BRADLEY PAUL, OHE MUNEMICHI, LU PU PING, MIURA MASANORI, MIHARA KAYOKO
Year of Publication 06.11.2018

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Patent

GUANIDINOBENZOIC ACID COMPOUND

GUANIDINOBENZOIC ACID COMPOUND

by SATOU TOMOHKI, OHNE KAZUHIKO, HONDO TAKESHI, MATSUURA KEISUKE, SASAMURA SATOSHI, FUJIYASU JIRO, YAMAKI SUSUMU, IMAIZUMI TOMOYOSHI
Year of Publication 21.05.2014

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Patent

GUANIDINE COMPOUND

GUANIDINE COMPOUND

by MIHARA HISASHI, YAMADA HIROYOSHI, YAMAKI SUSUMU, SEKI NORIO, YOSHIHARA KOUSEI, SUZUKI DAISUKE
Year of Publication 05.02.2014

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Patent

GUANIDINOBENZOIC ACID ESTER COMPOUND

GUANIDINOBENZOIC ACID ESTER COMPOUND

by YAMAKI, SUSUMU, FUJIYASU, JIRO, URANO, YASUHARU, SASAMURA, SATOSHI, ASANO, TORU, KOIKE, YUKA, KANEKO, OSAMU, IMAIZUMI, TOMOYOSHI, SATOU, TOMOHKI
Year of Publication 18.09.2014

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Patent

GUANIDINOBENZOIC ACID COMPOUND

GUANIDINOBENZOIC ACID COMPOUND

by YAMAKI, SUSUMU, FUJIYASU, JIRO, SASAMURA, SATOSHI, HONDO, TAKESHI, OHNE, KAZUHIKO, MATSUURA, KEISUKE, IMAIZUMI, TOMOYOSHI, SATOU, TOMOHKI
Year of Publication 21.03.2013

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Patent

GUANIDINE COMPOUND

GUANIDINE COMPOUND

by YAMAKI, SUSUMU, SUZUKI, DAISUKE, YAMADA, HIROYOSHI, MIHARA, HISASHI, YOSHIHARA, KOUSEI, SEKI, NORIO
Year of Publication 20.09.2012

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Patent

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