Formation and evolution of the South China Sea since the Late Mesozoic: A review
Li, Xue-jie, Wang, Zhe, Yao, Yong-jian, Gao, Hong-fang, Zhu, Song, Xu, Zi-ying
Published in China Geology (01.01.2023)
Published in China Geology (01.01.2023)
Get full text
Journal Article
Characteristics of gravity and magnetic fields and deep structural responses in the southern part of the Kyushu-Palau Ridge
Lin, Zhen, Lü, Wen-chao, Xu, Zi-ying, Qin, Peng-bo, Yao, Hui-qiang, Xiao, Xiao, Zhang, Xin-he, Yang, Chu-peng, Zhang, Xiang-yu, Chen, Jia-le
Published in China Geology (01.12.2021)
Published in China Geology (01.12.2021)
Get full text
Journal Article
Landslide integrated characteristics and susceptibility assessment in Rongxian county of Guangxi, China
Liao, Li-ping, Zhu, Ying-yan, Zhao, Yan-lin, Wen, Hai-tao, Yang, Yun-chuan, Chen, Li-hua, Ma, Shao-kun, Xu, Ying-zi
Published in Journal of mountain science (01.03.2019)
Published in Journal of mountain science (01.03.2019)
Get full text
Journal Article
Design and synthesis of thiophene dihydroisoquinolines as novel BACE1 inhibitors
Xu, Ying-zi, Yuan, Shendong, Bowers, Simeon, Hom, Roy K., Chan, Wayman, Sham, Hing L., Zhu, Yong L., Beroza, Paul, Pan, Hu, Brecht, Eric, Yao, Nanhua, Lougheed, Julie, Yan, Jiangli, Tam, Danny, Ren, Zhao, Ruslim, Lany, Bova, Michael P., Artis, Dean R.
Published in Bioorganic & medicinal chemistry letters (15.05.2013)
Published in Bioorganic & medicinal chemistry letters (15.05.2013)
Get full text
Journal Article
A computational and functional study elicits the ameliorating effect of the Chinese herbal formula Huo Luo Xiao Ling Dan on experimental ischemia-induced myocardial injury in rats via inhibition of apoptosis
Han, Xiang-Dong, Zhou, Zhi-Wei, Yang, Wei, Ye, Hang-Cheng, Xu, Ying-Zi, Huang, Yun-Feng, Zhang, Tong, Zhou, Shu-Feng
Published in Drug design, development and therapy (01.01.2015)
Published in Drug design, development and therapy (01.01.2015)
Get full text
Journal Article
PEG conjugates of potent α4 integrin inhibitors, maintaining sustained levels and bioactivity in vivo, following subcutaneous administration
Smith, Jenifer L., Rossiter, Kassandra I., Semko, Christopher M., Xu, Ying-Zi, Quincy, David A., Jagodzinski, Jacek, Dappen, Michael S., Konradi, Andrei W., Vandevert, Christopher, Garrido, Caroline, Mao, Wenxian, San Pablo, F. Bong, Wipke, Brian, Dofiles, Lilibeth, Wadsworth, Angie, Peterson, Eric, Lorenzana, Carlos, Simmonds, Stellanie, Messersmith, Elizabeth K., Bard, Frederique, Pleiss, Michael A., Yednock, Ted A.
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Get full text
Journal Article
Discovery of ( R )-4-Cyclopropyl-7,8-difluoro-5-(4-(trifluoromethyl)phenylsulfonyl)-4,5-dihydro-1 H -pyrazolo[4,3- c ]quinoline (ELND006) and ( R )-4-Cyclopropyl-8-fluoro-5-(6-(trifluoromethyl)pyridin-3-ylsulfonyl)-4,5-dihydro-2 H -pyrazolo[4,3- c ]quinoline (ELND007): Metabolically Stable γ-Secretase Inhibitors that Selectively Inhibit the Production of Amyloid-β over Notch
Probst, Gary, Aubele, Danielle L., Bowers, Simeon, Dressen, Darren, Garofalo, Albert W., Hom, Roy K., Konradi, Andrei W., Marugg, Jennifer L., Mattson, Matthew N., Neitzel, Martin L., Semko, Chris M., Sham, Hing L., Smith, Jenifer, Sun, Minghua, Truong, Anh P., Ye, Xiaocong M., Xu, Ying-zi, Dappen, Michael S., Jagodzinski, Jacek J., Keim, Pamela S., Peterson, Brian, Latimer, Lee H., Quincy, David, Wu, Jing, Goldbach, Erich, Ness, Daniel K., Quinn, Kevin P., Sauer, John-Michael, Wong, Karina, Zhang, Hongbin, Zmolek, Wes, Brigham, Elizabeth F., Kholodenko, Dora, Hu, Kang, Kwong, Grace T., Lee, Michael, Liao, Anna, Motter, Ruth N., Sacayon, Patricia, Santiago, Pamela, Willits, Christopher, Bard, Frédérique, Bova, Michael P., Hemphill, Susanna S., Nguyen, Lam, Ruslim, Lany, Tanaka, Kevin, Tanaka, Pearl, Wallace, William, Yednock, Ted A., Basi, Guriqbal S.
Published in Journal of medicinal chemistry (11.07.2013)
Published in Journal of medicinal chemistry (11.07.2013)
Get full text
Journal Article
Thermodynamic and kinetic characterization of hydroxyethylamine β-secretase-1 inhibitors
Mondal, Kalyani, Regnstrom, Karin, Morishige, Winse, Barbour, Robin, Probst, Gary, Xu, Ying-Zi, Artis, Dean R., Yao, Nanhua, Beroza, Paul, Bova, Michael P.
Published in Biochemical and biophysical research communications (15.11.2013)
Published in Biochemical and biophysical research communications (15.11.2013)
Get full text
Journal Article
Structure-based design of novel dihydroisoquinoline BACE-1 inhibitors that do not engage the catalytic aspartates
Bowers, Simeon, Xu, Ying-zi, Yuan, Shendong, Probst, Gary D., Hom, Roy K., Chan, Wayman, Konradi, Andrei W., Sham, Hing L., Zhu, Yong L., Beroza, Paul, Pan, Hu, Brecht, Eric, Yao, Nanhua, Lougheed, Julie, Tam, Danny, Ren, Zhao, Ruslim, Lany, Bova, Michael P., Artis, Dean R.
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
Get full text
Journal Article
Arylsulfonamide pyrimidines as VLA-4 antagonists
Xu, Ying-zi, Konradi, Andrei W., Bard, Frederique, Dappen, Michael, Dofiles, Lilibeth, Dreyer, Mark, Gallager, Ian, Garrido, Caroline, Krimm, Mike, Liao, Zhenmei, Messersmith, Elizabeth, Mutter, Linda, Pleiss, Michael A., Samant, Bhushan, Semko, Christopher M., Smith, Jennifer, Stappenbeck, Frank, Stupi, Brian, Vandervert, Chris, Welch, Brent, Wipke, Brian, Yednock, Ted
Published in Bioorganic & medicinal chemistry letters (15.05.2013)
Published in Bioorganic & medicinal chemistry letters (15.05.2013)
Get full text
Journal Article
Discovery of a novel [3.2.1] benzo fused bicyclic sulfonamide-pyrazoles as potent, selective and efficacious γ-secretase inhibitors
Ye, Xiaocong M., Konradi, Andrei W., Sun, Minghua, Yuan, Shendong, Aubele, Danielle L., Dappen, Michael, Dressen, Darren, Garofalo, Albert W., Jagodzinski, Jacek J., Latimer, Lee, Probst, Gary D., Sham, Hing L., Wone, David, Xu, Ying-zi, Ness, Daniel, Brigham, Elizabeth, Kwong, Grace T., Willtis, Chris, Tonn, George, Goldbach, Erich, Quinn, Kevin P., Zhang, Hongbin H., Sauer, John-Michael, Bova, Michael, Basi, Guriqbal S.
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
Get full text
Journal Article
Orally available and efficacious α4β1/α4β7 integrin inhibitors
Xu, Ying-zi, Smith, Jenifer L., Semko, Christopher M., Rossiter, Kassandra I., Fukuda, Juri Y., Dappen, Michael S., Quincy, David A., Konradi, Andrei W., Mao, Wenxian, Welch, Brent, Dreyer, Mark L., Samant, Bhushan, Zhang, Hongbin, Lugar, Judevin, Liao, Zhenmei, Henschel, Carrol, Petersen, Eric, Vandevert, Christopher, Shoemaker, Mark, Wehner, Nancy, Mutter, Linda, Shopp, George, Krimm, Michael, Chen, Linda, Wipke, Brian, Dofiles, Lilibeth, Gallager, Ian, Sauer, John-Michael, Messersmith, Elizabeth K., Pleiss, Michael A., Bard, Frederique, Yednock, Ted A.
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
Get full text
Journal Article
Development of a novel β-secretase binding assay using the AlphaScreen platform
Ren, Zhao, Tam, Danny, Xu, Ying-Zi, Wone, David, Yuan, Shendong, Sham, Hing L, Cheung, Harry, Regnstrom, Karin, Chen, Xiaohua, Rudolph, Donald, Jobling, Michael F, Artis, Dean R, Bova, Michael P
Published in Journal of biomolecular screening (01.07.2013)
Published in Journal of biomolecular screening (01.07.2013)
Get full text
Journal Article
Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: Structure–activity relationship of the aryl region
Probst, Gary D., Bowers, Simeon, Sealy, Jennifer M., Stupi, Brian, Dressen, Darren, Jagodzinska, Barbara M., Aquino, Jose, Gailunas, Andrea, Truong, Anh P., Tso, Luke, Xu, Ying-Zi, Hom, Roy K., John, Varghese, Tung, Jay S., Pleiss, Michael A., Tucker, John A., Konradi, Andrei W., Sham, Hing L., Jagodzinski, Jacek, Toth, Gergely, Brecht, Eric, Yao, Nanhua, Pan, Hu, Lin, May, Artis, Dean R., Ruslim, Lany, Bova, Michael P., Sinha, Sukanto, Yednock, Ted A., Gauby, Shawn, Zmolek, Wes, Quinn, Kevin P., Sauer, John-Michael
Published in Bioorganic & medicinal chemistry letters (15.10.2010)
Published in Bioorganic & medicinal chemistry letters (15.10.2010)
Get full text
Journal Article
A Label-Free Approach to Identify Inhibitors of α4β7-Mediated Cell Adhesion to MadCAM
Bova, Michael P., Nguyen, Lan, Wallace, William, Garrido, Caroline, Xu, Ying-Zi, Semko, Chris, Cockcroft, Kelly, Sandberg, Eric, Bard, Frederique
Published in SLAS discovery (01.06.2011)
Published in SLAS discovery (01.06.2011)
Get full text
Journal Article
Discovery of a novel sulfonamide-pyrazolopiperidine series as potent and Efficacious γ-Secretase Inhibitors
Ye, Xiaocong M., Konradi, Andrei W., Smith, Jenifer, Xu, Ying-Zi, Dressen, Darren, Garofalo, Albert W., Marugg, Jennifer, Sham, Hing L., Truong, Anh P., Jagodzinski, Jacek, Pleiss, Michael, Zhang, Hongbin, Goldbach, Erich, Sauer, John-Michael, Brigham, Elizabeth, Bova, Michael, Basi, Guriqbal S.
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Get full text
Journal Article
Discovery of a potent, orally bioavailable pyrimidine VLA-4 antagonist effective in a sheep asthma model
Semko, Christopher M., Chen, Linda, Dressen, Darren B., Dreyer, Mark L., Dunn, Whitney, Farouz, Francine S., Freedman, Stephen B., Holsztynska, Elizabeth J., Jefferies, Michael, Konradi, Andrei W., Liao, Anna, Lugar, Judevin, Mutter, Linda, Pleiss, Michael A., Quinn, Kevin P., Thompson, Thomas, Thorsett, Eugene D., Vandevert, Christopher, Xu, Ying-Zi, Yednock, Ted A.
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Get full text
Journal Article