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Crystal Structures of the Catalytic Domain of Phosphodiesterase 4B Complexed with AMP, 8-Br-AMP, and Rolipram
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Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPARγ partial agonist
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Ultra-potent P1 modified arylsulfonamide HIV protease inhibitors: The discovery of GW0385
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Published in Bioorganic & medicinal chemistry (15.09.2008)
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Substituted 2-[(4-Aminomethyl)phenoxy]-2-methylpropionic Acid PPARα Agonists. 1. Discovery of a Novel Series of Potent HDLc Raising Agents
Sierra, Michael L, Beneton, Véronique, Boullay, Anne-Bénédict, Boyer, Thierry, Brewster, Andrew G, Donche, Frédéric, Forest, Marie-Claire, Fouchet, Marie-Hélène, Gellibert, Françoise J, Grillot, Didier A, Lambert, Millard H, Laroze, Alain, Le Grumelec, Christelle, Linget, Jean Michel, Montana, Valerie G, Nguyen, Van-Loc, Nicodème, Edwige, Patel, Vipul, Penfornis, Annie, Pineau, Olivier, Pohin, Danig, Potvain, Florent, Poulain, Géraldine, Ruault, Cécile Bertho, Saunders, Michael, Toum, Jérôme, Xu, H. Eric, Xu, Robert X, Pianetti, Pascal M
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Solution Structure of the Amino-Terminal Fragment of Urokinase-Type Plasminogen Activator
Hansen, Andrew P, Petros, Andrew M, Meadows, Robert P, Nettesheim, David G, Mazar, Andrew P, Olejniczak, Edward T, Xu, Robert X, Pederson, Terry M, Henkin, Jack, Fesik, Stephen W
Published in Biochemistry (Easton) (01.04.1994)
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NMR Determination of the Structures of Peroxycobalt(III) Bleomycin and Cobalt(III) Bleomycin, Products of the Aerobic Oxidation of Cobalt(II) Bleomycin by Dioxygen
Xu, Robert X, Nettesheim, David, Otvos, James D, Petering, David H
Published in Biochemistry (Easton) (01.02.1994)
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Phenoxyacetic acids as PPARδ partial agonists: Synthesis, optimization, and in vivo efficacy
Evans, Karen A., Shearer, Barry G., Wisnoski, David D., Shi, Dongchuan, Sparks, Steven M., Sternbach, Daniel D., Winegar, Deborah A., Billin, Andrew N., Britt, Christy, Way, James M., Epperly, Andrea H., Leesnitzer, Lisa M., Merrihew, Raymond V., Xu, Robert X., Lambert, Millard H., Jin, Jian
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
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Crystallization of cyclic nucleotide phosphodiesterases
Ke, Hengming, Huai, Qing, Xu, Robert X
Published in Methods in molecular biology (Clifton, N.J.) (2005)
Published in Methods in molecular biology (Clifton, N.J.) (2005)
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NMR Structure of a Protein Kinase C-γ Phorbol-Binding Domain and Study of Protein−Lipid Micelle Interactions
Xu, Robert X, Pawelczyk, Tadeucz, Xia, Tai-He, Brown, Stephen C
Published in Biochemistry (Easton) (02.09.1997)
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A Structural Basis for Constitutive Activity in the Human CAR/RXRα Heterodimer
Xu, Robert X., Lambert, Millard H., Wisely, Bruce B., Warren, Erin N., Weinert, Emily E., Waitt, Gregory M., Williams, Jon D., Collins, Jon L., Moore, Linda B., Willson, Timothy M., Moore, John T.
Published in Molecular cell (22.12.2004)
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Three-dimensional structure of the FK506 binding protein/ascomycin complex in solution by heteronuclear three- and four-dimensional NMR
Meadows, Robert P, Nettesheim, David G, Xu, Robert X, Olejniczak, Edward T, Petros, Andrew M, Holzman, Thomas F, Severin, Jean, Gubbins, Earl, Smith, Harriet, Fesik, Stephen W
Published in Biochemistry (Easton) (26.01.1993)
Published in Biochemistry (Easton) (26.01.1993)
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Oxidative stress induced by a copper-thiosemicarbazone complex
Byrnes, Robert W, Mohan, Madan, Antholine, William E, Xu, Robert X, Petering, David H
Published in Biochemistry (Easton) (31.07.1990)
Published in Biochemistry (Easton) (31.07.1990)
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Corrigendum to “Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPARγ partial agonist” [Bioorg. Med. Chem. Lett. 21 (2011) 5568–5572]
Sime, Mairi, Allan, Amanda C., Chapman, Paul, Fieldhouse, Charlotte, Giblin, Gerard M.P., Healy, Mark P., Lambert, Millard H., Leesnitzer, Lisa M., Lewis, Ann, Merrihew, Raymond V., Rutter, Richard A., Sasse, Rosemary, Shearer, Barry G., Willson, Timothy M., Xu, Robert X., Virley, David J.
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
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1H, 13C, and 15N assignments and secondary structure of the FK506 binding protein when bound to ascomycin
Xu, R X, Nettesheim, D, Olejniczak, E T, Meadows, R, Gemmecker, G, Fesik, S W
Published in Biopolymers (01.04.1993)
Published in Biopolymers (01.04.1993)
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Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPAR[gamma] partial agonist
Sime, Mairi, Allan, Amanda C, Chapman, Paul, Fieldhouse, Charlotte, Giblin, Gerard MP, Healy, Mark P, Lambert, Millard H, Leesnitzer, Lisa M, Lewis, Ann, Merrihew, Raymond V, Rutter, Richard A, Sasse, Rosemary, Shearer, Barry G, Wilson, Timothy M, Xu, Robert X, Virley, David J
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
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