Collaborative virtual screening to elaborate an imidazo[1,2-]pyridine hit series for visceral leishmaniasis
Akao, Yuichiro, Canan, Stacie, Cao, Yafeng, Condroski, Kevin, Engkvist, Ola, Itono, Sachiko, Kaki, Rina, Kimura, Chiaki, Kogej, Thierry, Nagaoka, Kazuya, Naito, Akira, Nakai, Hiromi, Pairaudeau, Garry, Radu, Constantin, Roberts, Ieuan, Shimada, Mitsuyuki, Shum, David, Watanabe, Nao-aki, Xie, Huanxu, Yonezawa, Shuji, Yoshida, Osamu, Yoshida, Ryu, Mowbray, Charles, Perry, Benjamin
Published in MedChemComm (01.04.2021)
Published in MedChemComm (01.04.2021)
Get full text
Journal Article
Collaborative Virtual Screening Identifies a 2‑Aryl-4-aminoquinazoline Series with Efficacy in an In Vivo Model of Trypanosoma cruzi Infection
Tawaraishi, Taisuke, Ochida, Atsuko, Akao, Yuichiro, Itono, Sachiko, Kamaura, Masahiro, Akther, Thamina, Shimada, Mitsuyuki, Canan, Stacie, Chowdhury, Sanjoy, Cao, Yafeng, Condroski, Kevin, Engkvist, Ola, Francisco, Amanda, Ghosh, Sunil, Kaki, Rina, Kelly, John M., Kimura, Chiaki, Kogej, Thierry, Nagaoka, Kazuya, Naito, Akira, Pairaudeau, Garry, Radu, Constantin, Roberts, Ieuan, Shum, David, Watanabe, Nao-aki, Xie, Huanxu, Yonezawa, Shuji, Yoshida, Osamu, Yoshida, Ryu, Mowbray, Charles, Perry, Benjamin
Published in Journal of medicinal chemistry (26.01.2023)
Published in Journal of medicinal chemistry (26.01.2023)
Get full text
Journal Article
Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus
Klug, Dana M, Tse, Edwin G, Silva, Daniel G, Cao, Yafeng, Charman, Susan A, Chauhan, Jyoti, Crighton, Elly, Dichiara, Maria, Drake, Chris, Drewry, David, da Silva Emery, Flavio, Ferrins, Lori, Graves, Lee, Hopkins, Emily, Kresina, Thomas A C, Lorente-Macías, Álvaro, Perry, Benjamin, Phipps, Richard, Quiroga, Bruno, Quotadamo, Antonio, Sabatino, Giada N, Sama, Anthony, Schätzlein, Andreas, Simpson, Quillon J, Steele, Jonathan, Shanu-Wilson, Julia, Sjö, Peter, Stapleton, Paul, Swain, Christopher J, Vaideanu, Alexandra, Xie, Huanxu, Zuercher, William, Todd, Matthew H
Published in ACS infectious diseases (08.12.2023)
Published in ACS infectious diseases (08.12.2023)
Get full text
Journal Article