Identification of a novel PPARγ modulator with good anti-diabetic therapeutic index via structure-based screening, optimization and biological validation
Chen, Fangyuan, Ma, Lei, Cai, Guihui, Tang, Junyuan, Wang, Yi, Liu, Qingmei, Liu, Xiawen, Hou, Ning, Zhou, Zhi, Yi, Wei
Published in Biomedicine & pharmacotherapy (01.10.2022)
Published in Biomedicine & pharmacotherapy (01.10.2022)
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Antenatal steroids elicited neurodegenerative-associated transcriptional changes in the hippocampus of preterm fetal sheep independent of lung maturation
Carter, Sean W. D, Fee, Erin L, Usuda, Haruo, Oguz, Gokce, Ramasamy, Adaikalavan, Amin, Zubair, Agnihotri, Biswas, Wei, Qin, Xiawen, Liu, Takahashi, Tsukasa, Takahashi, Yuki, Ikeda, Hideyuki, Kumagai, Yusaku, Saito, Yuya, Saito, Masatoshi, Mattar, Citra, Evans, Mark I, Illanes, Sebastián E, Jobe, Alan H, Choolani, Mahesh, Kemp, Matthew W
Published in BMC medicine (26.08.2024)
Published in BMC medicine (26.08.2024)
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Mask and Release Strategy‐Enabled Diversity‐Oriented Synthesis for DNA‐Encoded Library
Zhang, Silin, Zhang, Haiman, Liu, Xiawen, Qi, Ping, Tan, Tingting, Wang, Shengdong, Gao, Hui, Xu, Hongtao, Zhou, Zhi, Yi, Wei
Published in Advanced science (01.02.2024)
Published in Advanced science (01.02.2024)
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EGCG Inhibits Proliferation and Induces Apoptosis Through Downregulation of SIRT1 in Nasopharyngeal Carcinoma Cells
Jiang, Shisheng, Huang, Chaoming, Zheng, Guodong, Yi, Wei, Wu, Bo, Tang, Junyuan, Liu, Xiawen, Huang, Biyun, Wu, Dan, Yan, Tingdong, Li, Mingxi, Wan, Chunpeng, Cai, Yi
Published in Frontiers in nutrition (Lausanne) (25.04.2022)
Published in Frontiers in nutrition (Lausanne) (25.04.2022)
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Simulated lunar microgravity transiently arrests growth and induces osteocyte-chondrocyte lineage differentiation in human Wharton's jelly stem cells
Subramanian, Arjunan, Ip, Chelsea Han Lin, Qin, Wei, Liu, Xiawen, W D Carter, Sean, Oguz, Gokce, Ramasamy, Adaikalavan, E Illanes, Sebastian, Biswas, Arijit, G Perron, Gabriel, L Fee, Erin, W L Li, Sarah, K Y Seah, Michelle, A Choolani, Mahesh, W Kemp, Matthew
Published in NPJ microgravity (04.05.2024)
Published in NPJ microgravity (04.05.2024)
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gem‐Difluoromethylene Alkyne‐Enabled Diverse C−H Functionalization and Application to the on‐DNA Synthesis of Difluorinated Isocoumarins
Gao, Hui, Lin, Shuang, Zhang, Shuning, Chen, Weijie, Liu, Xiawen, Yang, Guang, Lerner, Richard A., Xu, Hongtao, Zhou, Zhi, Yi, Wei
Published in Angewandte Chemie (25.01.2021)
Published in Angewandte Chemie (25.01.2021)
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Journal Article
gem‐Difluoromethylene Alkyne‐Enabled Diverse C−H Functionalization and Application to the on‐DNA Synthesis of Difluorinated Isocoumarins
Gao, Hui, Lin, Shuang, Zhang, Shuning, Chen, Weijie, Liu, Xiawen, Yang, Guang, Lerner, Richard A., Xu, Hongtao, Zhou, Zhi, Yi, Wei
Published in Angewandte Chemie International Edition (25.01.2021)
Published in Angewandte Chemie International Edition (25.01.2021)
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Journal Article
Structure-based screening, optimization and biological evaluation of novel chrysin-based derivatives as selective PPARγ modulators for the treatment of T2DM and hepatic steatosis
Ma, Lei, Tang, Junyuan, Chen, Fangyuan, Liu, Qingmei, Huang, Junjun, Liu, Xiawen, Zhou, Zhi, Yi, Wei
Published in European journal of medicinal chemistry (05.10.2024)
Published in European journal of medicinal chemistry (05.10.2024)
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Journal Article
2H‑Chromene-3-carboxylic Acid Synthesis via Solvent-Controlled and Rhodium(III)-Catalyzed Redox-Neutral C–H Activation/[3 + 3] Annulation Cascade
Zhou, Zhi, Bian, Mengyao, Zhao, Lixin, Gao, Hui, Huang, Junjun, Liu, Xiawen, Yu, Xiyong, Li, Xingwei, Yi, Wei
Published in Organic letters (06.07.2018)
Published in Organic letters (06.07.2018)
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Journal Article
2 H-Chromene-3-carboxylic Acid Synthesis via Solvent-Controlled and Rhodium(III)-Catalyzed Redox-Neutral C-H Activation/[3 + 3] Annulation Cascade
Zhou, Zhi, Bian, Mengyao, Zhao, Lixin, Gao, Hui, Huang, Junjun, Liu, Xiawen, Yu, Xiyong, Li, Xingwei, Yi, Wei
Published in Organic letters (06.07.2018)
Published in Organic letters (06.07.2018)
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Journal Article
Naftopidil enantiomers suppress androgen accumulation and induce cell apoptosis via the UDP-glucuronosyltransferase 2B15 in benign prostate hyperplasia
Zhan, Haoxin, Zhang, Silin, Li, Lirong, Chen, Zikai, Cai, Yi, Huang, Junjun, Wu, Dan, Huang, Biyun, Wu, Bo, Liu, Xiawen
Published in The Journal of steroid biochemistry and molecular biology (01.07.2022)
Published in The Journal of steroid biochemistry and molecular biology (01.07.2022)
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Baicalin inhibits pressure overload-induced cardiac fibrosis through regulating AMPK/TGF-β/Smads signaling pathway
Xiao, Yichuan, Ye, Jiantao, Zhou, Ying, Huang, Junjun, Liu, Xiawen, Huang, Biyun, Zhu, Liu, Wu, Bo, Zhang, Genshui, Cai, Yi
Published in Archives of biochemistry and biophysics (15.02.2018)
Published in Archives of biochemistry and biophysics (15.02.2018)
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Methazolamide Attenuates the Development of Diabetic Cardiomyopathy by Promoting β-Catenin Degradation in Type 1 Diabetic Mice
Chen, Xiaoqing, Li, Yilang, Yuan, Xun, Yuan, Wenchang, Li, Conglin, Zeng, Yue, Lian, Yuling, Qiu, Xiaoxia, Qin, Yuan, Zhang, Guiping, Liu, Xiawen, Luo, Chengfeng, Luo, Jian-Dong, Hou, Ning
Published in Diabetes (New York, N.Y.) (01.04.2022)
Published in Diabetes (New York, N.Y.) (01.04.2022)
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Journal Article
Structure-based screening and biological validation of the anti-thrombotic drug-dicoumarol as a novel and potent PPARγ-modulating ligand
Ma, Lei, Tang, Junyuan, Cai, Guihui, Chen, Fangyuan, Liu, Qingmei, Zhou, Zhi, Zhang, Silin, Liu, Xiawen, Hou, Ning, Yi, Wei
Published in Bioorganic chemistry (01.12.2022)
Published in Bioorganic chemistry (01.12.2022)
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Journal Article
Abstract 576: Nrf2 is a Key Regulator on Puerarin Preventing Cardiac Hypertrophy and Upregulating Metabolic Enzymes Ugt1a1 and Ugt1a9 in Rats
Hou, Ning, Zhao, Ganjian, Cai, Shaoai, Liu, Xiawen, Li, Aiqun, Huang, Yin, Li, Lirong, Luo, Chengfeng
Published in Circulation research (03.08.2018)
Published in Circulation research (03.08.2018)
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Journal Article
Novel naftopidil-related derivatives and their biological effects as alpha(1)-adrenoceptors antagonists and antiproliferative agents
Huang, Junjun, He, Fei, Huang, Minyi, Liu, Xiawen, Xiong, Yan, Huang, Yajian, Zhu, Liu, Yang, Ya, Xu, Xingjie, Yuan, Mu
Published in European journal of medicinal chemistry (26.05.2015)
Published in European journal of medicinal chemistry (26.05.2015)
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Journal Article
Novel naftopidil-related derivatives and their biological effects as alpha1-adrenoceptors antagonists and antiproliferative agents
Huang, Junjun, He, Fei, Huang, Minyi, Liu, Xiawen, Xiong, Yan, Huang, Yajian, Zhu, Liu, Yang, Ya, Xu, Xingjie, Yuan, Mu
Published in European journal of medicinal chemistry (26.05.2015)
Published in European journal of medicinal chemistry (26.05.2015)
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Journal Article
Determination of naftopidil enantiomers in rat plasma using chiral solid phases and pre-column derivatization high-performance liquid chromatography
Liu, Xiawen, Zhang, Yunying, Yuan, Mu, Sun, Yinxiang
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.10.2012)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.10.2012)
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Enantiospecific determination of naftopidil by RRLC–MS/MS reveals stereoselective pharmacokinetics and tissue distributions in rats
Liu, Xiawen, Zhang, Xingfei, Huang, Junjun, Rong, Yi, Luo, Chengfeng, Guo, Jiewen, Zhu, Liu, Huang, Biyun, Yuan, Mu
Published in Journal of pharmaceutical and biomedical analysis (10.08.2015)
Published in Journal of pharmaceutical and biomedical analysis (10.08.2015)
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