Lead identification of novel and selective TYK2 inhibitors
Liang, Jun, Tsui, Vickie, Van Abbema, Anne, Bao, Liang, Barrett, Kathy, Beresini, Maureen, Berezhkovskiy, Leo, Blair, Wade S., Chang, Christine, Driscoll, James, Eigenbrot, Charles, Ghilardi, Nico, Gibbons, Paul, Halladay, Jason, Johnson, Adam, Kohli, Pawan Bir, Lai, Yingjie, Liimatta, Marya, Mantik, Priscilla, Menghrajani, Kapil, Murray, Jeremy, Sambrone, Amy, Xiao, Yisong, Shia, Steven, Shin, Young, Smith, Jan, Sohn, Sue, Stanley, Mark, Ultsch, Mark, Zhang, Birong, Wu, Lawren C., Magnuson, Steven
Published in European journal of medicinal chemistry (01.09.2013)
Published in European journal of medicinal chemistry (01.09.2013)
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Lead Optimization of a 4‑Aminopyridine Benzamide Scaffold To Identify Potent, Selective, and Orally Bioavailable TYK2 Inhibitors
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Published in Journal of medicinal chemistry (13.06.2013)
Published in Journal of medicinal chemistry (13.06.2013)
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Identification of the KIF18A alpha-4 helix as a therapeutic target for chromosomally unstable tumor cells
Schutt, Katherine L, Queen, Katelyn A, Fisher, Kira, Budington, Olivia, Mao, Weifeng, Liu, Wei, Gu, Xiaohui, Xiao, Yisong, Aswad, Fred, Joseph, James, Stumpff, Jason
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RobustMQ: benchmarking robustness of quantized models
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Published in Visual Intelligence (15.12.2023)
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Back Pocket Flexibility Provides Group II p21-Activated Kinase (PAK) Selectivity for Type I 1/2 Kinase Inhibitors
Staben, Steven T, Feng, Jianwen A, Lyle, Karen, Belvin, Marcia, Boggs, Jason, Burch, Jason D, Chua, Ching-ching, Cui, Haifeng, DiPasquale, Antonio G, Friedman, Lori S, Heise, Christopher, Koeppen, Hartmut, Kotey, Adrian, Mintzer, Robert, Oh, Angela, Roberts, David Allen, Rouge, Lionel, Rudolph, Joachim, Tam, Christine, Wang, Weiru, Xiao, Yisong, Young, Amy, Zhang, Yamin, Hoeflich, Klaus P
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Abstract 4965: Targeting the mitotic kinesin, KIF18A, in chromosomally unstable cancers
Joseph, James D., Schutt, Katherine, Fisher, Kira, Queen, Katelyn, Budington, Olivia, Mao, Weifeng, Liu, Wei, Zhu, Zhengqing, Zhang, Xiangping, Xiao, Yisong, Lai, Kunmin, Gu, Xiaohui, Stumpff, Jason, Aswad, Fred
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Identification of C‑2 Hydroxyethyl Imidazopyrrolopyridines as Potent JAK1 Inhibitors with Favorable Physicochemical Properties and High Selectivity over JAK2
Zak, Mark, Hurley, Christopher A, Ward, Stuart I, Bergeron, Philippe, Barrett, Kathy, Balazs, Mercedesz, Blair, Wade S, Bull, Richard, Chakravarty, Paroma, Chang, Christine, Crackett, Peter, Deshmukh, Gauri, DeVoss, Jason, Dragovich, Peter S, Eigenbrot, Charles, Ellwood, Charles, Gaines, Simon, Ghilardi, Nico, Gibbons, Paul, Gradl, Stefan, Gribling, Peter, Hamman, Chris, Harstad, Eric, Hewitt, Peter, Johnson, Adam, Johnson, Tony, Kenny, Jane R, Koehler, Michael F. T, Bir Kohli, Pawan, Labadie, Sharada, Lee, Wyne P, Liao, Jiangpeng, Liimatta, Marya, Mendonca, Rohan, Narukulla, Raman, Pulk, Rebecca, Reeve, Austin, Savage, Scott, Shia, Steven, Steffek, Micah, Ubhayakar, Savita, van Abbema, Anne, Aliagas, Ignacio, Avitabile-Woo, Barbara, Xiao, Yisong, Yang, Jing, Kulagowski, Janusz J
Published in Journal of medicinal chemistry (13.06.2013)
Published in Journal of medicinal chemistry (13.06.2013)
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2-Amino-[1,2,4]triazolo[1,5-a]pyridines as JAK2 inhibitors
Siu, Michael, Pastor, Richard, Liu, Wendy, Barrett, Kathy, Berry, Megan, Blair, Wade S., Chang, Christine, Chen, Jacob Z., Eigenbrot, Charles, Ghilardi, Nico, Gibbons, Paul, He, Haiying, Hurley, Christopher A., Kenny, Jane R., Cyrus Khojasteh, S., Le, Hoa, Lee, Leslie, Lyssikatos, Joseph P., Magnuson, Steve, Pulk, Rebecca, Tsui, Vickie, Ultsch, Mark, Xiao, Yisong, Zhu, Bing-yan, Sampath, Deepak
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
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Discovery and Optimization of C-2 Methyl Imidazopyrrolopyridines as Potent and Orally Bioavailable JAK1 Inhibitors with Selectivity over JAK2
Zak, Mark, Mendonca, Rohan, Balazs, Mercedesz, Barrett, Kathy, Bergeron, Philippe, Blair, Wade S, Chang, Christine, Deshmukh, Gauri, DeVoss, Jason, Dragovich, Peter S, Eigenbrot, Charles, Ghilardi, Nico, Gibbons, Paul, Gradl, Stefan, Hamman, Chris, Hanan, Emily J, Harstad, Eric, Hewitt, Peter R, Hurley, Christopher A, Jin, Tian, Johnson, Adam, Johnson, Tony, Kenny, Jane R, Koehler, Michael F. T, Bir Kohli, Pawan, Kulagowski, Janusz J, Labadie, Sharada, Liao, Jiangpeng, Liimatta, Marya, Lin, Zhonghua, Lupardus, Patrick J, Maxey, Robert J, Murray, Jeremy M, Pulk, Rebecca, Rodriguez, Madeleine, Savage, Scott, Shia, Steven, Steffek, Micah, Ubhayakar, Savita, Ultsch, Mark, van Abbema, Anne, Ward, Stuart I, Xiao, Ling, Xiao, Yisong
Published in Journal of medicinal chemistry (12.07.2012)
Published in Journal of medicinal chemistry (12.07.2012)
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Benchmarking the Physical-world Adversarial Robustness of Vehicle Detection
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Zhang, Tianyuan, Wang, Lu, Li, Hainan, Xiao, Yisong, Liang, Siyuan, Liu, Aishan, Liu, Xianglong, Tao, Dacheng
Published in arXiv.org (16.07.2024)
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Year of Publication 30.06.2024
Year of Publication 30.06.2024
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RobustMQ: Benchmarking Robustness of Quantized Models
Xiao, Yisong, Liu, Aishan, Zhang, Tianyuan, Qin, Haotong, Guo, Jinyang, Liu, Xianglong
Published in arXiv.org (04.08.2023)
Published in arXiv.org (04.08.2023)
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Guo, Jun, Liu, Aishan, Zheng, Xingyu, Liang, Siyuan, Xiao, Yisong, Wu, Yichao, Liu, Xianglong
Published in arXiv.org (03.08.2023)
Published in arXiv.org (03.08.2023)
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Pre-trained Trojan Attacks for Visual Recognition
Liu, Aishan, Zhang, Xinwei, Xiao, Yisong, Zhou, Yuguang, Liang, Siyuan, Wang, Jiakai, Liu, Xianglong, Cao, Xiaochun, Tao, Dacheng
Published in arXiv.org (23.12.2023)
Published in arXiv.org (23.12.2023)
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