Evaluation of Efficacy, Biodistribution, and Inflammation for a Potent siRNA Nanoparticle: Effect of Dexamethasone Co-treatment
Abrams, Marc T, Koser, Martin L, Seitzer, Jessica, Williams, Stephanie C, DiPietro, Martha A, Wang, Weimin, Shaw, Andrew W, Mao, Xianzhi, Jadhav, Vasant, Davide, Joseph P, Burke, Paul A, Sachs, Alan B, Stirdivant, Steven M, Sepp-Lorenzino, Laura
Published in Molecular therapy (01.01.2010)
Published in Molecular therapy (01.01.2010)
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Journal Article
Mechanistically Probing Lipid-siRNA Nanoparticle-associated Toxicities Identifies Jak Inhibitors Effective in Mitigating Multifaceted Toxic Responses
Tao, Weikang, Mao, Xianzhi, Davide, Joseph P, Ng, Bruce, Cai, Mingmei, Burke, Paul A, Sachs, Alan B, Sepp-Lorenzino, Laura
Published in Molecular therapy (01.03.2011)
Published in Molecular therapy (01.03.2011)
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Paracrine Expression of a Native Soluble Vascular Endothelial Growth Factor Receptor Inhibits Tumor Growth, Metastasis, and Mortality Rate
Goldman, Corey K., Kendall, Richard L., Cabrera, Gustavo, Soroceanu, Liliana, Heike, Yuji, Gillespie, G. Yancey, Siegal, Gene P., Mao, Xianzhi, Bett, Andrew J., Huckle, William R., Thomas, Kenneth A., Curiel, David T.
Published in Proceedings of the National Academy of Sciences - PNAS (21.07.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (21.07.1998)
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Pyridyl aminothiazoles as potent Chk1 inhibitors: Optimization of cellular activity
Dudkin, Vadim Y., Wang, Cheng, Arrington, Kenneth L., Fraley, Mark E., Hartman, George D., Stirdivant, Steven M., Drakas, Robert A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Hardwick, James, Tao, Weikang, Beck, Stephen C., Mao, Xianzhi, Lobell, Robert B., Sepp-Lorenzino, Laura
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Journal Article
Dynamic Contrast-Enhanced MRI Measurements of Passive Permeability through Blood Retinal Barrier in Diabetic Rats
Berkowitz, Bruce A, Roberts, Robin, Luan, Hongmei, Peysakhov, Jamie, Mao, Xianzhi, Thomas, Kenneth A
Published in Investigative ophthalmology & visual science (01.07.2004)
Published in Investigative ophthalmology & visual science (01.07.2004)
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Journal Article
3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6
Fraley, Mark E., Steen, Justin T., Brnardic, Edward J., Arrington, Kenneth L., Spencer, Keith L., Hanney, Barbara A., Kim, Yuntae, Hartman, George D., Stirdivant, Steven M., Drakas, Bob A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Hardwick, James, Tao, Weikang, Beck, Stephen C., Mao, Xianzhi, Lobell, Robert B., Sepp-Lorenzino, Laura, Yan, Youwei, Ikuta, Mari, Munshi, Sanjeev K., Kuo, Lawrence C., Kreatsoulas, Constantine
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
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Journal Article
Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors
Brnardic, Edward J., Garbaccio, Robert M., Fraley, Mark E., Tasber, Edward S., Steen, Justin T., Arrington, Kenneth L., Dudkin, Vadim Y., Hartman, George D., Stirdivant, Steven M., Drakas, Bob A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Hardwick, James, Tao, Weikang, Beck, Stephen C., Mao, Xianzhi, Lobell, Robert B., Sepp-Lorenzino, Laura, Yan, Youwei, Ikuta, Mari, Munshi, Sanjeev K., Kuo, Lawrence C., Kreatsoulas, Constantine
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Journal Article
Development of 6-substituted indolylquinolinones as potent Chek1 kinase inhibitors
Huang, Shaei, Garbaccio, Robert M., Fraley, Mark E., Steen, Justin, Kreatsoulas, Constantine, Hartman, George, Stirdivant, Steve, Drakas, Bob, Rickert, Keith, Walsh, Eileen, Hamilton, Kelly, Buser, Carolyn A., Hardwick, James, Mao, Xianzhi, Abrams, Marc, Beck, Steve, Tao, Weikang, Lobell, Rob, Sepp-Lorenzino, Laura, Yan, Youwei, Ikuta, Mari, Murphy, Joan Zugay, Sardana, Vinod, Munshi, Sanjeev, Kuo, Lawrence, Reilly, Michael, Mahan, Elizabeth
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
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Journal Article
Potent N-(1,3-Thiazol-2-yl)pyridin-2-amine Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitors with Excellent Pharmacokinetics and Low Affinity for the hERG Ion Channel
Bilodeau, Mark T, Balitza, Adrienne E, Koester, Timothy J, Manley, Peter J, Rodman, Leonard D, Buser-Doepner, Carolyn, Coll, Kathleen E, Fernandes, Christine, Gibbs, Jackson B, Heimbrook, David C, Huckle, William R, Kohl, Nancy, Lynch, Joseph J, Mao, Xianzhi, McFall, Rosemary C, McLoughlin, Debra, Miller-Stein, Cynthia M, Rickert, Keith W, Sepp-Lorenzino, Laura, Shipman, Jennifer M, Subramanian, Raju, Thomas, Kenneth A, Wong, Bradley K, Yu, Sean, Hartman, George D
Published in Journal of medicinal chemistry (02.12.2004)
Published in Journal of medicinal chemistry (02.12.2004)
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Journal Article
Synthesis and evaluation of substituted benzoisoquinolinones as potent inhibitors of Chk1 kinase
Garbaccio, Robert M., Huang, Shaei, Tasber, Edward S., Fraley, Mark E., Yan, Youwei, Munshi, Sanjeev, Ikuta, Mari, Kuo, Lawrence, Kreatsoulas, Constanine, Stirdivant, Steve, Drakas, Bob, Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly A., Buser, Carolyn A., Hardwick, James, Mao, Xianzhi, Beck, Stephen C., Abrams, Marc T., Tao, Weikang, Lobell, Rob, Sepp-Lorenzino, Laura, Hartman, George D.
Published in Bioorganic & medicinal chemistry (15.11.2007)
Published in Bioorganic & medicinal chemistry (15.11.2007)
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Journal Article
Vascular Endothelial Growth Factor Receptor KDR Tyrosine Kinase Activity Is Increased by Autophosphorylation of Two Activation Loop Tyrosine Residues
Kendall, R L, Rutledge, R Z, Mao, X, Tebben, A J, Hungate, R W, Thomas, K A
Published in The Journal of biological chemistry (05.03.1999)
Published in The Journal of biological chemistry (05.03.1999)
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A novel orally bioavailable inhibitor of kinase insert domain-containing receptor induces antiangiogenic effects and prevents tumor growth in vivo
SEPP-LORENZINO, Laura, RANDS, Elaine, COLL, Kathleen, CIECKO, Patrice, FRALEY, Mark, HOFFMAN, William, HARTMAN, George, HEIMBROOK, David, GIBBS, Jackson, KOHL, Nancy, THOMAS, Kenneth, XIANZHI MAO, CONNOLLY, Brett, SHIPMAN, Jennifer, ANTANAVAGE, Joanne, HILL, Susan, DAVIS, Lenora, BECK, Stephen, RICKERT, Keith
Published in Cancer research (Chicago, Ill.) (15.01.2004)
Published in Cancer research (Chicago, Ill.) (15.01.2004)
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Enhanced hindlimb collateralization induced by acidic fibroblast growth factor is dependent upon femoral artery extraction
HERSHEY, James C, CORCORAN, Halea A, BASKIN, Elizabeth P, GILBERTO, David B, XIANZHI MAO, THOMAS, Kenneth A, COOK, Jacquelynn J
Published in Cardiovascular research (01.10.2003)
Published in Cardiovascular research (01.10.2003)
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Journal Article
Use of 99m Tc-Trodat-1 SPECT to evaluate the efficacy of deep brain stimulation in Parkinson's disease
Dongfang, Chen, Xianzhi, Mao, Cen, Lou, Zhongke, Huang
Published in Hellenic journal of nuclear medicine (01.09.2022)
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Published in Hellenic journal of nuclear medicine (01.09.2022)
Journal Article
Use of 99mTc-Trodat-1 SPECT to evaluate the efficacy of deep brain stimulation in Parkinson's disease
Dongfang, Chen, Xianzhi, Mao, Cen, Lou, Zhongke, Huang
Published in Hellenic journal of nuclear medicine (01.09.2022)
Published in Hellenic journal of nuclear medicine (01.09.2022)
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Journal Article
Vascular endothelial growth factor stimulates angiogenesis without improving collateral blood flow following hindlimb ischemia in rabbits
Hershey, James C, Baskin, Elizabeth P, Corcoran, Halea A, Bett, Andrew, Dougherty, Nancy M, Gilberto, David B, Mao, Xianzhi, Thomas, Kenneth A, Cook, Jacquelynn J
Published in Heart and vessels (01.07.2003)
Published in Heart and vessels (01.07.2003)
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Journal Article
Development of thioquinazolinones, allosteric Chk1 kinase inhibitors
Converso, Antonella, Hartingh, Timothy, Garbaccio, Robert M., Tasber, Edward, Rickert, Keith, Fraley, Mark E., Yan, Youwei, Kreatsoulas, Constantine, Stirdivant, Steve, Drakas, Bob, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Mao, Xianzhi, Abrams, Marc T., Beck, Stephen C., Tao, Weikang, Lobell, Rob, Sepp-Lorenzino, Laura, Zugay-Murphy, Joan, Sardana, Vinod, Munshi, Sanjeev K., Jezequel-Sur, Sylvie Marie, Zuck, Paul D., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Journal Article
Abstract 2888: Lipid nanoparticle-mediated delivery of siRNA to extrahepatic tumors
Davide, Joseph P., Ng, Bruce, Mao, Xianzhi, Patel, Manishkumar, Shi, Bin, Hochman, Jerome, Cunningham, James J., Sepp-Lorenzino, Laura, Tao, Weikang
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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