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Published in Archives of toxicology (01.05.2022)
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Discovery of 5-substituent-N-arylbenzamide derivatives as potent, selective and orally bioavailable LRRK2 inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.09.2017)
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Apigenin and Temozolomide Synergistically Inhibit Glioma Growth Through the PI3K / AKT Pathway
Wang, Dong, Wang, Zhijun, Dai, Xuedong, Zhang, Liang, Li, Min
Published in Cancer biotherapy & radiopharmaceuticals (01.03.2024)
Published in Cancer biotherapy & radiopharmaceuticals (01.03.2024)
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Mild and Regioselective N‑Alkylation of 2‑Pyridones in Water
Hao, Xin, Xu, Zhongmiao, Lu, Hongfu, Dai, Xuedong, Yang, Ting, Lin, Xichen, Ren, Feng
Published in Organic letters (17.07.2015)
Published in Organic letters (17.07.2015)
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Assessing IRAK4 Functions in ABC DLBCL by IRAK4 Kinase Inhibition and Protein Degradation
Zhang, Jing, Fu, Liqiang, Shen, Bin, Liu, Yingtao, Wang, Wenqian, Cai, Xin, Kong, Linglong, Yan, Yilin, Meng, Ryan, Zhang, Zhuming, Chen, Ying-Nan P., Liu, Qian, Wan, Zhao-Kui, Zhou, Tianyuan, Wang, Xiaotao, Gavine, Paul, Del Rosario, Amanda, Ahn, Kay, Philippar, Ulrike, Attar, Ricardo, Yang, Jennifer, Xu, Yanping, Edwards, James P., Dai, Xuedong
Published in Cell chemical biology (17.12.2020)
Published in Cell chemical biology (17.12.2020)
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Discovery of Highly Potent and Selective IRAK1 Degraders to Probe Scaffolding Functions of IRAK1 in ABC DLBCL
Fu, Liqiang, Zhang, Jing, Shen, Bin, Kong, Linglong, Liu, Yingtao, Tu, Wangyang, Wang, Wenqian, Cai, Xin, Wang, Xiaotao, Cheng, Na, Xia, Mingxuan, Zhou, Tianyuan, Liu, Qian, Xu, Yanping, Yang, Jennifer, Gavine, Paul, Philippar, Ulrike, Attar, Ricardo, Edwards, James P, Venable, Jennifer D, Dai, Xuedong
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Published in Journal of medicinal chemistry (12.08.2021)
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Preclinical efficacy of the potent, selective menin-KMT2A inhibitor JNJ-75276617 (bleximenib) in KMT2A- and NPM1-altered leukemias
Kwon, Min Chul, Thuring, Jan Willem, Querolle, Olivier, Dai, Xuedong, Verhulst, Tinne, Pande, Vineet, Marien, Ann, Goffin, Dries, Wenge, Daniela V., Yue, Hong, Cutler, Jevon A., Jin, Cyrus, Perner, Florian, Hogeling, Shanna M., Shaffer, Paul L., Jacobs, Frank, Vinken, Petra, Cai, Wei, Keersmaekers, Vikki, Eyassu, Filmon, Bhogal, Balpreet, Verstraeten, Karin, El Ashkar, Sara, Perry, Jennifer A., Jayaguru, Prathiba, Barreyro, Laura, Kuchnio, Anna, Darville, Nicolas, Krosky, Daniel, Urbanietz, Gregor, Verbist, Bie, Edwards, James P., Cowley, Glenn S., Kirkpatrick, Robert, Steele, Ruth, Ferrante, Lucille, Guttke, Christina, Daskalakis, Nikki, Pietsch, E. Christine, Wilson, David M., Attar, Ricardo, Elsayed, Yusri, Fischer, Eric S., Schuringa, Jan Jacob, Armstrong, Scott A., Packman, Kathryn, Philippar, Ulrike
Published in Blood (12.09.2024)
Published in Blood (12.09.2024)
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Pharmacological Characterization of JNJ-75276617, a Menin-KMT2A Inhibitor, As Targeted Treatment for KMT2A-Altered and NPM1-Mutant Acute Leukemia
Kwon, Min Chul, Querolle, Olivier, Dai, Xuedong, Thuring, Jan Willem, Verhulst, Tinne, Marien, Ann, Goffin, Dries, Cai, Wei, Keersmaekers, Vikki, Eyassu, Filmon, Verstraeten, Karin, El Ashkar, Sara, Hogeling, Shanna M, Jacob, Frank, Vinken, Petra, Darville, Nicolas, Pande, Vineet, Krosky, Daniel, Urbanietz, Gregor, Verbist, Bie, Ferrante, Lucille A., Drenberg, Christina Diane, Wilson, David, Attar, Ricardo M., Schuringa, Jan Jacob, Daskalakis, Nikki, Packman, Kathryn, Pietsch, Christine, Elsayed, Yusri, Philippar, Ulrike
Published in Blood (15.11.2022)
Published in Blood (15.11.2022)
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5-Substituted-N-pyridazinylbenzamides as potent and selective LRRK2 inhibitors: Improved brain unbound fraction enables efficacy
Ding, Xiao, Stasi, Luigi Piero, Dai, Xuedong, Long, Kai, Peng, Cheng, Zhao, Baowei, Wang, Hailong, Sun, Changhui, Hu, Huan, Wan, Zehong, Jandu, Karamjit S., Philps, Oliver J., Chen, Yan, Wang, Lizhen, Liu, Qian, Edge, Colin, Li, Yi, Dong, Kelly, Guan, Xiaoming, Tattersall, F. David, Reith, Alastair D., Ren, Feng
Published in Bioorganic & medicinal chemistry letters (15.01.2019)
Published in Bioorganic & medicinal chemistry letters (15.01.2019)
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Lichao FANG, Liqiang FU, Tinne Ann J VERHULST, Lianzhu LIU, Wei CAI, Yanping XU, Yu SUN, Alicia Tee Fuay NG, Nicolas Freddy J DARVILLE, Min Chul KWON, Christina Diane GUTTKE, Lucille Angela FERRANTE, Sumia ALI-AHMED, Balpreet BHOGAL, Xiangjun DENG, Ulrike PHILIPPAR, Johannes Wilhelmus J. THURING, DAI, Xuedong DAI, Xuedong, Olivier Alexis Georges QUEROLLE, Yingtao LIU, Kathryn Elizabeth PACKMAN, Nikki DASKALAKIS, Eva Christine PIETSCH, Vineet PANDE, Ming LI
Year of Publication 07.06.2024
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Year of Publication 07.06.2024
Patent
3D-Pharmacophore Models for Selective A2A and A2B Adenosine Receptor Antagonists
Wei, Jing, Wang, Songqing, Gao, Shaofen, Dai, Xuedong, Gao, Qingzhi
Published in Journal of chemical information and modeling (26.03.2007)
Published in Journal of chemical information and modeling (26.03.2007)
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Discovery of a novel 2,3,11,11a-tetrahydro-1H-pyrazino[1,2-b]isoquinoline-1,4(6H)-dione series promoting neurogenesis of human neural progenitor cells
Lin, Hong, Fang, Haiyan, Wang, Jamie, Meng, Qinghua, Dai, Xuedong, Wu, Sharon, Luo, Jie, Pu, Dan, Chen, Libo, Minick, Douglas, Arai, Ken, Mandeville, Emiri T., Lo, Eng, Holder, Julie C., Chuang, Tsu Tshen, Zhao, Jing
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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The discovery of a facile access to the synthesis of NSAID dendritic prodrugs
Du, Zuyin, Lu, Yanhui, Dai, Xuedong, Zhang-Negrerie, Daisy, Gao, Qingzhi
Published in Journal of chemical research (01.03.2013)
Published in Journal of chemical research (01.03.2013)
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3D-Pharmacophore Models for Selective A 2A and A 2B Adenosine Receptor Antagonists
Wei, Jing, Wang, Songqing, Gao, Shaofen, Dai, Xuedong, Gao, Qingzhi
Published in Journal of chemical information and modeling (01.03.2007)
Published in Journal of chemical information and modeling (01.03.2007)
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3D-Pharmacophore Models for Selective A^sub 2A^ and A^sub 2B^ Adenosine Receptor Antagonists
Wei, Jing, Wang, Songqing, Gao, Shaofen, Dai, Xuedong, Gao, Qingzhi
Published in Journal of chemical information and modeling (01.03.2007)
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Published in Journal of chemical information and modeling (01.03.2007)
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