Abstract 1729: Discovery of a synthetic small molecule inhibitor of HSP90 for cancer therapy
Bao, Rudi, Pan, Zhongzong, Zhao, Zhiming, Yu, Hongping, Xu, Yaochang
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Journal Article
Abstract LB-288: A highly selective small molecule CSF-1R inhibitor demonstrates strong immunomodulatory activity in syngeneic models
Yang, Shuqun, Zhao, Baowei, Zhang, Mingming, Zhao, Yuan, Chen, Xin, Zhang, Lei, Yu, Hongping, Chen, Zhui, Xu, Yaochang
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 3063: Discovery of a third-generation EGFR inhibitor, which is highly selective and potent against both resistant and activating EGFR mutations for NSCLC therapy
Bao, Rudi, Gao, Peng, Zhang, Fujun, Tong, Zhaolong, Yu, Hongping, Xu, Yaochang
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
Abstract LB525: Discovery and characterization of ABSK111, a selective, CNS-penetrable, and broad-spectrum EGFR inhibitor targeting exon20 insertion, atypical and extracellular mutations
Dai, Cheng, Peng, Juan, Yang, Fei, Deng, Haibing, Zhao, Yuan, Yu, Hongping, Xu, Yaochang, Chen, Zhui, Yang, Shuqun
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
2,3-DIHYDRO-1H-PYRROLO[3,2-B]PYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Zhang, Mingming, Zhao, Baowei
Year of Publication 04.04.2024
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Year of Publication 04.04.2024
Patent
Azaaryl derivative, preparation method therefor, and application thereof for use in pharmacy
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Zhang, Mingming, Zhao, Baowei
Year of Publication 28.09.2021
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Year of Publication 28.09.2021
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FGFR4 inhibitor, preparation method therefor and pharmaceutical use thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Deng, Haibing, Ying, Haiyan, Yang, Fei
Year of Publication 17.01.2023
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Year of Publication 17.01.2023
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Biaryl derivative, preparation method thereof and pharmaceutical application thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Zhang, Yongxian, Ying, Haiyan, Yang, Fei
Year of Publication 04.10.2022
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Year of Publication 04.10.2022
Patent
N-(azaaryl)cyclolactam-1-carboxamide derivative, preparation method therefor, and use thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Zhang, Mingming, Yang, Shuqun, Zhao, Baowei
Year of Publication 19.10.2021
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Year of Publication 19.10.2021
Patent
N-(azaaryl)cyclolactam-1-carboxamide derivative, preparation method therefor, and use thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Zhang, Mingming, Yang, Shuqun, Zhao, Baowei
Year of Publication 19.08.2021
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Year of Publication 19.08.2021
Patent
FGFR4 inhibitor, preparation method therefor and pharmaceutical use thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Deng, Haibing, Ying, Haiyan, Yang, Fei
Year of Publication 06.04.2021
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Year of Publication 06.04.2021
Patent
N-(azaaryl)cyclolactam-1-carboxamide derivative, preparation method therefor, and use thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Zhang, Mingming, Yang, Shuqun, Zhao, Baowei
Year of Publication 08.10.2020
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Year of Publication 08.10.2020
Patent
FGFR4 inhibitor, preparation method therefor and pharmaceutical use thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Deng, Haibing, Ying, Haiyan, Yang, Fei
Year of Publication 18.06.2020
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Year of Publication 18.06.2020
Patent
N-(azaaryl)cyclolactam-1-carboxamide derivative, preparation method therefor, and use thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Zhang, Mingming, Yang, Shuqun, Zhao, Baowei
Year of Publication 12.12.2019
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Year of Publication 12.12.2019
Patent
FGFR4 inhibitor, preparation method therefor and pharmaceutical use thereof
Xu, Yaochang, Yu, Hongping, Chen, Zhui, Deng, Haibing, Ying, Haiyan, Yang, Fei
Year of Publication 16.05.2019
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Year of Publication 16.05.2019
Patent