Discovery of Novel PI3Kδ Inhibitors Based on the p110δ Crystal Structure
Jia, Wenqing, Luo, Shuyu, Zhao, Wennan, Xu, Weiren, Zhong, Yuxu, Kong, Dexin
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Conjugated bile acids activate the sphingosine-1-phosphate receptor 2 in primary rodent hepatocytes
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Study on the Effect of Three CYP2C9 Variants on Drug–Drug Interaction Related to Six Drugs In Vitro by LC–MS/MS Method
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Systematic Structure-Activity Relationship (SAR) Exploration of Diarylmethane Backbone and Discovery of A Highly Potent Novel Uric Acid Transporter 1 (URAT1) Inhibitor
Cai, Wenqing, Wu, Jingwei, Liu, Wei, Xie, Yafei, Liu, Yuqiang, Zhang, Shuo, Xu, Weiren, Tang, Lida, Wang, Jianwu, Zhao, Guilong
Published in Molecules (Basel, Switzerland) (27.01.2018)
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Discovery of a Flexible Triazolylbutanoic Acid as a Highly Potent Uric Acid Transporter 1 (URAT1) Inhibitor
Tian, He, Liu, Wei, Zhou, Zhixing, Shang, Qian, Liu, Yuqiang, Xie, Yafei, Liu, Changying, Xu, Weiren, Tang, Lida, Wang, Jianwu, Zhao, Guilong
Published in Molecules (Basel, Switzerland) (16.11.2016)
Published in Molecules (Basel, Switzerland) (16.11.2016)
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Novel Anthranilamide-Based FXa Inhibitors: Drug Design, Synthesis and Biological Evaluation
Wang, Wenzhi, Yuan, Jing, Fu, Xiaoli, Meng, Fancui, Zhang, Shijun, Xu, Weiren, Xu, Yongnan, Huang, Changjiang
Published in Molecules (Basel, Switzerland) (14.04.2016)
Published in Molecules (Basel, Switzerland) (14.04.2016)
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GLP-1 analogs containing disulfide bond exhibited prolonged half-life in vivo than GLP-1
Li, Ying, Zheng, Xuemin, Tang, Lida, Xu, Weiren, Gong, Min
Published in Peptides (New York, N.Y. : 1980) (01.06.2011)
Published in Peptides (New York, N.Y. : 1980) (01.06.2011)
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The influence of genetic polymorphisms in drug metabolism enzymes and transporters on the pharmacokinetics of different fluvastatin formulations
Xiang, Qian, Wu, Weidang, Zhao, Nan, Li, Chuan, Xu, Junyu, Ma, Lingyue, Zhang, Xiaodan, Xie, Qiufen, Zhang, Zhuo, Wang, Jiancheng, Xu, Weiren, Zhao, Xia, Cui, Yimin
Published in Asian journal of pharmceutical sciences (01.03.2020)
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Inhibition of P-glycoprotein by HIV protease inhibitors increases intracellular accumulation of berberine in murine and human macrophages
Zha, Weibin, Wang, Guangji, Xu, Weiren, Liu, Xuyuan, Wang, Yun, Zha, Beth S, Shi, Jian, Zhao, Qijin, Gerk, Phillip M, Studer, Elaine, Hylemon, Phillip B, Pandak, Jr, William M, Zhou, Huiping
Published in PloS one (23.01.2013)
Published in PloS one (23.01.2013)
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Discovery of Flexible Naphthyltriazolylmethane-based Thioacetic Acids as Highly Active Uric Acid Transporter 1 (URAT1) Inhibitors for the Treatment of Hyperuricemia of Gout
Zhang, Xiansheng, Wu, Jingwei, Liu, Wei, Liu, Yuqiang, Xie, Yafei, Shang, Qian, Zhou, Zhixing, Xu, Weiren, Tang, Lida, Wang, Jianwu, Zhao, Guilong
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.05.2017)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.05.2017)
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Design, Synthesis and Biological Activity of Tetrazole-bearing Uric Acid Transporter 1 Inhibitors
Cai, Wenqing, Liu, Wei, Xie, Yafei, Wu, Jingwei, Liu, Yuqiang, Liu, Changying, Xu, Weiren, Tang, Lida, Wang, Jianwu, Zhao, Guilong
Published in Chemical research in Chinese universities (01.02.2017)
Published in Chemical research in Chinese universities (01.02.2017)
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Effects of Astragaloside IV on heart failure in rats
Zhao, Zhuanyou, Wang, Weiting, Wang, Fang, Zhao, Kerui, Han, Yingmei, Xu, Weiren, Tang, Lida
Published in Chinese medicine (02.04.2009)
Published in Chinese medicine (02.04.2009)
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Discovery of 6-deoxydapagliflozin as a highly potent sodium-dependent glucose cotransporter 2 (SGLT2) inhibitor for the treatment of type 2 diabetes
Zhang, Lingyu, Wang, Yuli, Xu, Huaqiang, Shi, Yongheng, Liu, Bingni, Wei, Qunchao, Xu, Weiren, Tang, Lida, Wang, Jianwu, Zhao, Guilong
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.05.2014)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.05.2014)
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Disulfide bond prolongs the half-life of therapeutic peptide-GLP-1
Li, Ying, Li, Xin, Zheng, Xuemin, Tang, Lida, Xu, Weiren, Gong, Min
Published in Peptides (New York, N.Y. : 1980) (01.07.2011)
Published in Peptides (New York, N.Y. : 1980) (01.07.2011)
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Synthesis and biological evaluation of 3-(1H-indol-3-yl)pyrazole-5-carboxylic acid derivatives
Zhang, Datong, Wang, Guangtian, Tan, Chubing, Xu, Weiren, Pei, Yuan, Huo, Lingyan
Published in Archives of pharmacal research (01.03.2011)
Published in Archives of pharmacal research (01.03.2011)
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1-(5-Bromo-2-chlorophenyl)-2,2-dichloro-1-(4-ethoxyphenyl)cyclopropane
Han, Shuwen, Shi, Yongheng, Yuli, Wang, Zhao, Guilong, Xu, Weiren
Published in Acta crystallographica. Section E, Structure reports online (01.03.2013)
Published in Acta crystallographica. Section E, Structure reports online (01.03.2013)
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