Discovery of 6‑(Fluoro-18 F)‑3-(1H‑pyrrolo[2,3‑c]pyridin-1-yl)isoquinolin-5-amine ([18F]-MK-6240): A Positron Emission Tomography (PET) Imaging Agent for Quantification of Neurofibrillary Tangles (NFTs)
Walji, Abbas M, Hostetler, Eric D, Selnick, Harold, Zeng, Zhizhen, Miller, Patricia, Bennacef, Idriss, Salinas, Cristian, Connolly, Brett, Gantert, Liza, Holahan, Marie, O’Malley, Stacey, Purcell, Mona, Riffel, Kerry, Li, Jing, Balsells, Jaume, OBrien, Julie A, Melquist, Stacey, Soriano, Aileen, Zhang, Xiaoping, Ogawa, Aimie, Xu, Serena, Joshi, Elizabeth, Della Rocca, Joseph, Hess, Fred J, Schachter, Joel, Hesk, David, Schenk, David, Struyk, Arie, Babaoglu, Kerim, Lohith, Talakad G, Wang, Yaode, Yang, Kun, Fu, Jianmin, Evelhoch, Jeffrey L, Coleman, Paul J
Published in Journal of medicinal chemistry (26.05.2016)
Published in Journal of medicinal chemistry (26.05.2016)
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Discovery of a Novel cGAMP Competitive Ligand of the Inactive Form of STING
Siu, Tony, Altman, Michael D, Baltus, Gretchen A, Childers, Matthew, Ellis, J. Michael, Gunaydin, Hakan, Hatch, Harold, Ho, Thu, Jewell, James, Lacey, Brian M, Lesburg, Charles A, Pan, Bo-Sheng, Sauvagnat, Berengere, Schroeder, Gottfried K, Xu, Serena
Published in ACS medicinal chemistry letters (10.01.2019)
Published in ACS medicinal chemistry letters (10.01.2019)
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Combinatorial macrophage induced innate immunotherapy against Ewing sarcoma: Turning "Two Keys" simultaneously
Luo, Wen, Hoang, Hai, Miller, Katherine E, Zhu, Hongwen, Xu, Serena, Mo, Xiaokui, Garfinkle, Elizabeth A R, Costello, Heather, Wijeratne, Saranga, Chemnitz, Wiebke, Gandhi, Ronan, Liao, Yanling, Ayello, Janet, Gardenswartz, Aliza, Rosenblum, Jeremy M, Cassady, Kevin A, Mardis, Elaine R, Lee, Dean A, Cripe, Timothy P, Cairo, Mitchell S
Published in Journal of experimental & clinical cancer research (11.07.2024)
Published in Journal of experimental & clinical cancer research (11.07.2024)
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Discovery and Characterization of Vicriviroc (SCH 417690), a CCR5 Antagonist with Potent Activity against Human Immunodeficiency Virus Type 1
STRIZKI, Julie M, TREMBLAY, Cecile, TAGAT, Jayaram R, COX, Kathleen, PRIESTLEY, Tony, SOROTA, Steve, WEI HUANG, HIRSCH, Martin, REYES, Gregory R, BAROUDY, Bahige M, XU, Serena, WOJCIK, Lisa, WAGNER, Nicole, GONSIOREK, Waldemar, HIPKIN, R. William, CHOU, Chuan-Chu, PUGLIESE-SIVO, Catherine, YUSHI XIAO
Published in Antimicrobial Agents and Chemotherapy (01.12.2005)
Published in Antimicrobial Agents and Chemotherapy (01.12.2005)
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Generation and properties of a human immunodeficiency virus type 1 isolate resistant to the small molecule CCR5 inhibitor, SCH-417690 (SCH-D)
Marozsan, Andre J., Kuhmann, Shawn E., Morgan, Thomas, Herrera, Carolina, Rivera-Troche, Enid, Xu, Serena, Baroudy, Bahige M., Strizki, Julie, Moore, John P.
Published in Virology (New York, N.Y.) (20.07.2005)
Published in Virology (New York, N.Y.) (20.07.2005)
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HIV-1 Escape from a Small Molecule, CCR5-Specific Entry Inhibitor Does Not Involve CXCR4 Use
Trkola, Alexandra, Kuhmann, Shawn E., Strizki, Julie M., Maxwell, Elizabeth, Ketas, Tom, Morgan, Tom, Pugach, Pavel, Xu, Serena, Wojcik, Lisa, Tagat, Jayaram, Palani, Anandan, Shapiro, Sherry, Clader, John W., McCombie, Stuart, Reyes, Gregory R., Baroudy, Bahige M., Moore, John P.
Published in Proceedings of the National Academy of Sciences - PNAS (08.01.2002)
Published in Proceedings of the National Academy of Sciences - PNAS (08.01.2002)
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SCH-C (SCH 351125), An Orally Bioavailable, Small Molecule Antagonist of the Chemokine Receptor CCR5, is a Potent Inhibitor of HIV-1 Infection in vitro and in vivo
Strizki, Julie M., Xu, Serena, Wagner, Nicole E., Wojcik, Lisa, Liu, Jia, Hou, Yan, Endres, Michael, Palani, Anandan, Shapiro, Sherry, Clader, John W., Greenlee, William J., Tagat, Jayaram R., McCombie, Stuart, Cox, Kathleen, Fawzi, Ahmad B., Chou, Chuan-Chu, Pugliese-Sivo, Catherine, Davies, Liza, Moreno, Mary E., Ho, David D., Trkola, Alexandra, Stoddart, Cheryl A., Moore, John P., Reyes, Gregory R., Baroudy, Bahige M.
Published in Proceedings of the National Academy of Sciences - PNAS (23.10.2001)
Published in Proceedings of the National Academy of Sciences - PNAS (23.10.2001)
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Neutralization Profiles of Primary Human Immunodeficiency Virus Type 1 Isolates in the Context of Coreceptor Usage
Cecilia, D, KewalRamani, V N, O'Leary, J, Volsky, B, Nyambi, P, Burda, S, Xu, S, Littman, D R, Zolla-Pazner, S
Published in Journal of Virology (01.09.1998)
Published in Journal of Virology (01.09.1998)
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Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. II. Discovery of 1-[(2,4-Dimethyl-3-pyridinyl)carbonyl]-4- methyl-4-[3(S)-methyl-4-[1(S)-[4-(trifluoro- methyl)phenyl]ethyl]-1-piperazinyl]- piperidine N1-Oxide (Sch-350634), an Orally Bioavailable, Potent CCR5 Antagonist
Tagat, Jayaram R, Steensma, Ruo W, McCombie, Stuart W, Nazareno, Dennis V, Lin, Sue-Ing, Neustadt, Bernard R, Cox, Kathleen, Xu, Serena, Wojcik, Lisa, Murray, Michael G, Vantuno, Nicole, Baroudy, Bahige M, Strizki, Julie M
Published in Journal of medicinal chemistry (11.10.2001)
Published in Journal of medicinal chemistry (11.10.2001)
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An orally available non-nucleotide STING agonist with antitumor activity
Pan, Bo-Sheng, Perera, Samanthi A, Piesvaux, Jennifer A, Presland, Jeremy P, Schroeder, Gottfried K, Cumming, Jared N, Trotter, B Wesley, Altman, Michael D, Buevich, Alexei V, Cash, Brandon, Cemerski, Saso, Chang, Wonsuk, Chen, Yiping, Dandliker, Peter J, Feng, Guo, Haidle, Andrew, Henderson, Timothy, Jewell, James, Kariv, Ilona, Knemeyer, Ian, Kopinja, Johnny, Lacey, Brian M, Laskey, Jason, Lesburg, Charles A, Liang, Rui, Long, Brian J, Lu, Min, Ma, Yanhong, Minnihan, Ellen C, O'Donnell, Greg, Otte, Ryan, Price, Laura, Rakhilina, Larissa, Sauvagnat, Berengere, Sharma, Sharad, Tyagarajan, Sriram, Woo, Hyun, Wyss, Daniel F, Xu, Serena, Bennett, David Jonathan, Addona, George H
Published in Science (American Association for the Advancement of Science) (21.08.2020)
Published in Science (American Association for the Advancement of Science) (21.08.2020)
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Induction of Neutralizing Antibodies to T-Cell Line-Adapted and Primary Human Immunodeficiency Virus Type 1 Isolates with a Prime-Boost Vaccine Regimen in Chimpanzees
Zolla-Pazner, S, Lubeck, M, Xu, S, Burda, S, Natuk, R J, Sinangil, F, Steimer, K, Gallo, R C, Eichberg, J W, Matthews, T, Robert-Guroff, M
Published in Journal of Virology (01.02.1998)
Published in Journal of Virology (01.02.1998)
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Preclinical Characterization of 18 F-MK-6240, a Promising PET Tracer for In Vivo Quantification of Human Neurofibrillary Tangles
Hostetler, Eric D., Walji, Abbas M., Zeng, Zhizhen, Miller, Patricia, Bennacef, Idriss, Salinas, Cristian, Connolly, Brett, Gantert, Liza, Haley, Hyking, Holahan, Marie, Purcell, Mona, Riffel, Kerry, Lohith, Talakad G., Coleman, Paul, Soriano, Aileen, Ogawa, Aimie, Xu, Serena, Zhang, Xiaoping, Joshi, Elizabeth, Della Rocca, Joseph, Hesk, David, Schenk, David J., Evelhoch, Jeffrey L.
Published in Journal of Nuclear Medicine (01.10.2016)
Published in Journal of Nuclear Medicine (01.10.2016)
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Preclinical Characterization of ^sup 18^F-MK-6240, a Promising PET Tracer for In Vivo Quantification of Human Neurofibrillary Tangles
Hostetler, Eric D, Walji, Abbas M, Zeng, Zhizhen, Miller, Patricia, Bennacef, Idriss, Salinas, Cristian, Connolly, Brett, Gantert, Liza, Haley, Hyking, Holahan, Marie, Purcell, Mona, Riffel, Kerry, Lohith, Talakad G, Coleman, Paul, Soriano, Aileen, Ogawa, Aimie, Xu, Serena, Zhang, Xiaoping, Joshi, Elizabeth, Della Rocca, Joseph, Hesk, David, Schenk, David J, Evelhoch, Jeffrey L
Published in The Journal of nuclear medicine (1978) (01.10.2016)
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Published in The Journal of nuclear medicine (1978) (01.10.2016)
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Preclinical Characterization of super( 18)F-MK-6240, a Promising PET Tracer for In Vivo Quantification of Human Neurofibrillary Tangles
Hostetler, Eric D, Walji, Abbas M, Zeng, Zhizhen, Miller, Patricia, Bennacef, Idriss, Salinas, Cristian, Connolly, Brett, Gantert, Liza, Haley, Hyking, Holahan, Marie, Purcell, Mona, Riffel, Kerry, Lohith, Talakad G, Coleman, Paul, Soriano, Aileen, Ogawa, Aimie, Xu, Serena, Zhang, Xiaoping, Joshi, Elizabeth, Della Rocca, Joseph, Hesk, David, Schenk, David J, Evelhoch, Jeffrey L
Published in The Journal of nuclear medicine (1978) (01.10.2016)
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Published in The Journal of nuclear medicine (1978) (01.10.2016)
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Live Cell Membranome cDNA Screen: A Novel Homogenous Live Cell Binding Assay to Study Membrane Protein-Ligand Interaction
Shen, Xun, Smith, Elizabeth, Ai, Xi, McElroy, William T., Liaw, Andy, Kreamer, Tony, Chang, Meiping, Devito, Kristine, Hudak, Edward, Xu, Serena, Pei, Yi, Sur, Sylvie, Peier, Andrea, Li, Jing
Published in SLAS discovery (01.12.2019)
Published in SLAS discovery (01.12.2019)
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Neutralization of HIV-1 primary isolates by polyclonal and monoclonal human antibodies
Hioe, C E, Xu, S, Chigurupati, P, Burda, S, Williams, C, Gorny, M K, Zolla-Pazner, S
Published in International immunology (01.09.1997)
Published in International immunology (01.09.1997)
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IC‐P‐187: Discovery and First‐in‐Human Evaluation of the TAU‐imaging PET Radiotracer [18F]MK‐6240
Bennacef, Idriss, Zeng, Zhizhen, Lohith, Talakad, Miller, Patricia J., Salinas, Cristian A., Connolly, Brett M., Gantert, Liza T., Hyking, Haley D., Holahan, Marie A., O’Malley, Stacey S., Purcell, Mona L., Riffel, Kerry, Coleman, Paul J., Li, Jing, Balsells-Padros, Jaume, Soriano, Aileen, Ogawa, Aimie M., Xu, Serena, Xiaoping, Zhang, Della Rocca, Joseph, Schachter, Joel B., Hesk, David, Telan-Choing, Florestina, Struyk, Arie, Sur, Cyrille, Celen, Sofie, Serdons, Kim, Bormans, Guy, Vandenbulcke, Mathieu, Vandenberghe, Rik, De Hoon, Jan, Koole, Michel, Van Laere, Koen, Declercq, Ruben, Reynders, Tom, Abbas, Walji, Hostetler, Eric D., Evelhoch, Jeffrey
Published in Alzheimer's & dementia (01.07.2016)
Published in Alzheimer's & dementia (01.07.2016)
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Journal Article
P1‐246: Discovery and First‐in‐Human Evaluation of the TAU‐Imaging PET Radiotracer [18F]MK‐6240
Bennacef, Idriss, Zeng, Zhizhen, Lohith, Talakad, Miller, Patricia J., Salinas, Cristian A., Connolly, Brett M., Gantert, Liza T., Haley, Hyking D., Marie, Holahan A., O’Malley, Stacey S., Purcell, Mona L., Riffel, Kerry, Coleman, Paul J., Li, Jing, Balsells-Padros, Jaume, Soriano, Aileen, Ogawa, Aimie M., Xu, Serena, Xiaoping, Zhang, Della Rocca, Joseph, Schachter, Joel B., Hesk, David, David, Schenk J., Telan-Choing, Florestina, Struyk, Arie, Sur, Cyrille, Celen, Sofie, Serdons, Kim, Bormans, Guy, Vandenbulcke, Mathieu, Vandenberghe, Rik, De Hoon, Jan, Koole, Michel, Van Laere, Koen, Declercq, Ruben, Tom, Reynders, Abbas, Walji, Eric, Hostetler D., Evelhoch, Jeffrey
Published in Alzheimer's & dementia (01.07.2016)
Published in Alzheimer's & dementia (01.07.2016)
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Journal Article
DISCOVERY AND FIRST-IN-HUMAN EVALUATION OF THE TAU-IMAGING PET RADIOTRACER [18 F]MK-6240
Bennacef, Idriss, Zeng, Zhizhen, Lohith, Talakad, Miller, Patricia J, Salinas, Cristian A, Connolly, Brett M, Gantert, Liza T, Haley, Hyking D, Marie, Holahan A, O’Malley, Stacey S, Purcell, Mona L, Riffel, Kerry, Coleman, Paul J, Li, Jing, Balsells-Padros, Jaume, Soriano, Aileen, Ogawa, Aimie M, Xu, Serena, Xiaoping, Zhang, Della Rocca, Joseph, Schachter, Joel B, Hesk, David, David, Schenk J, Telan-Choing, Florestina, Struyk, Arie, Sur, Cyrille, Celen, Sofie, Serdons, Kim, Bormans, Guy, Vandenbulcke, Mathieu, Vandenberghe, Rik, De Hoon, Jan, Koole, Michel, Van Laere, Koen, Declercq, Ruben, Tom, Reynders, Abbas, Walji, Eric, Hostetler D, Evelhoch, Jeffrey
Published in Alzheimer's & dementia (01.07.2016)
Published in Alzheimer's & dementia (01.07.2016)
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