Discovery of SARS-CoV‑2 Papain-like Protease Inhibitors through a Combination of High-Throughput Screening and a FlipGFP-Based Reporter Assay
Ma, Chunlong, Sacco, Michael Dominic, Xia, Zilei, Lambrinidis, George, Townsend, Julia Alma, Hu, Yanmei, Meng, Xiangzhi, Szeto, Tommy, Ba, Mandy, Zhang, Xiujun, Gongora, Maura, Zhang, Fushun, Marty, Michael Thomas, Xiang, Yan, Kolocouris, Antonios, Chen, Yu, Wang, Jun
Published in ACS central science (28.07.2021)
Published in ACS central science (28.07.2021)
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Journal Article
Enantioselective Bromo-oxycyclization of Silanol
Xia, Zilei, Hu, Jiadong, Shen, Zhigao, Wan, Xiaolong, Yao, Qizheng, Lai, Yisheng, Gao, Jin-Ming, Xie, Weiqing
Published in Organic letters (04.01.2016)
Published in Organic letters (04.01.2016)
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Journal Article
Potent HIV‐1 Protease Inhibitors Containing Carboxylic and Boronic Acids: Effect on Enzyme Inhibition and Antiviral Activity and Protein‐Ligand X‐ray Structural Studies
Ghosh, Arun K., Xia, Zilei, Kovela, Satish, Robinson, William L., Johnson, Megan E., Kneller, Daniel W., Wang, Yuan‐Fang, Aoki, Manabu, Takamatsu, Yuki, Weber, Irene T., Mitsuya, Hiroaki
Published in ChemMedChem (06.11.2019)
Published in ChemMedChem (06.11.2019)
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Discovery of Di- and Trihaloacetamides as Covalent SARS-CoV‑2 Main Protease Inhibitors with High Target Specificity
Ma, Chunlong, Xia, Zilei, Sacco, Michael Dominic, Hu, Yanmei, Townsend, Julia Alma, Meng, Xiangzhi, Choza, Juliana, Tan, Haozhou, Jang, Janice, Gongora, Maura V, Zhang, Xiujun, Zhang, Fushun, Xiang, Yan, Marty, Michael Thomas, Chen, Yu, Wang, Jun
Published in Journal of the American Chemical Society (15.12.2021)
Published in Journal of the American Chemical Society (15.12.2021)
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Rational Design of Hybrid SARS-CoV‑2 Main Protease Inhibitors Guided by the Superimposed Cocrystal Structures with the Peptidomimetic Inhibitors GC-376, Telaprevir, and Boceprevir
Xia, Zilei, Sacco, Michael, Hu, Yanmei, Ma, Chunlong, Meng, Xiangzhi, Zhang, Fushun, Szeto, Tommy, Xiang, Yan, Chen, Yu, Wang, Jun
Published in ACS pharmacology & translational science (13.08.2021)
Published in ACS pharmacology & translational science (13.08.2021)
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Journal Article
Total Synthesis of (−)-Conolutinine
Feng, Xiangyang, Jiang, Guangde, Xia, Zilei, Hu, Jiadong, Wan, Xiaolong, Gao, Jin-Ming, Lai, Yisheng, Xie, Weiqing
Published in Organic letters (18.09.2015)
Published in Organic letters (18.09.2015)
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Journal Article
Synthesis of naked amino-pyrroloindoline via direct aminocyclization of tryptamine
Shen, Zhigao, Xia, Zilei, Zhao, Huijun, Hu, Jiadong, Wan, Xiaolong, Lai, Yisheng, Zhu, Chen, Xie, Weiqing
Published in Organic & biomolecular chemistry (21.05.2015)
Published in Organic & biomolecular chemistry (21.05.2015)
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Abstract 7277: Discovery of INV-9956, an orally available and highly selective Cyp11A1 inhibitor for the treatment of castration-resistant prostate cancer with drug resistant AR mutations
Bai, Chang, Chen, Danqi, Xia, Zilei, Huang, Shujuan, Lin, LIshan, Zeng, Zhaopie, Su, Jing, Sun, Yongkui
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Facile access to 2,2-disubstituted indolin-3-ones via a cascade Fischer indolization/Claisen rearrangement reactionElectronic supplementary information (ESI) available: General experimental procedures and spectroscopic data for all new compounds. CCDC 1036012 (5). For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c7cc03754f
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Synthesis of naked amino-pyrroloindoline via direct aminocyclization of tryptamineElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob00546a
Shen, Zhigao, Xia, Zilei, Zhao, Huijun, Hu, Jiadong, Wan, Xiaolong, Lai, Yisheng, Zhu, Chen, Xie, Weiqing
Year of Publication 07.05.2015
Year of Publication 07.05.2015
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Journal Article
Oxidative rearrangement of malondialdehyde: substrate scope and mechanistic insights
Yu, Xin, Liu, Zheng, Xia, Zilei, Shen, Zhigao, Pan, Xixian, Zhang, Hui, Xie, Weiqing
Published in RSC advances (01.01.2014)
Published in RSC advances (01.01.2014)
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Journal Article
Re sub(2)O sub(7) catalyzed dienone-phenol rearrangement
Xia, Zilei, Hu, Jiadong, Shen, Zhigao, Yao, Qizheng, Xie, Weiqing
Published in RSC advances (01.04.2015)
Published in RSC advances (01.04.2015)
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Journal Article
Discovery of SARS-CoV-2 papain-like protease inhibitors through a combination of high-throughput screening and FlipGFP-based reporter assay
Xia, Zilei, Sacco, Michael Dominic, Ma, Chunlong, Townsend, Julia Alma, Kitamura, Naoya, Hu, Yanmei, Ba, Mandy, Szeto, Tommy, Zhang, Xiujun, Meng, Xiangzhi, Zhang, Fushun, Xiang, Yan, Marty, Michael Thomas, Chen, Yu, Wang, Jun
Published in bioRxiv (16.03.2021)
Published in bioRxiv (16.03.2021)
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Paper
ChemInform Abstract: Re2O7 Catalyzed Dienone-Phenol Rearrangement
Xia, Zilei, Hu, Jiadong, Shen, Zhigao, Yao, Qizheng, Xie, Weiqing
Published in ChemInform (01.09.2015)
Published in ChemInform (01.09.2015)
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Journal Article
ChemInform Abstract: Re 2 O 7 Catalyzed Dienone‐Phenol Rearrangement
Xia, Zilei, Hu, Jiadong, Shen, Zhigao, Yao, Qizheng, Xie, Weiqing
Published in ChemInform (01.09.2015)
Published in ChemInform (01.09.2015)
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