Novel isoindoline compounds for potent and selective inhibition of prolyl dipeptidase DPP8
Jiaang, Weir-Torn, Chen, Yuan-Shou, Hsu, Tsu, Wu, Ssu-Hui, Chien, Chia-Hui, Chang, Chung-Nien, Chang, Sheng-Ping, Lee, Shiow-Ju, Chen, Xin
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
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Journal Article
A three-dimensional pharmacophore model for dipeptidyl peptidase IV inhibitors
Lu, I.-Lin, Tsai, Keng-Chang, Chiang, Yi-Kun, Jiaang, Weir-Torn, Wu, Ssu-Hui, Mahindroo, Neeraj, Chien, Chia-Hui, Lee, Shiow-Ju, Chen, Xin, Chao, Yu-Sheng, Wu, Su-Ying
Published in European journal of medicinal chemistry (01.08.2008)
Published in European journal of medicinal chemistry (01.08.2008)
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Journal Article
Rational design and synthesis of potent and long-lasting glutamic acid-based dipeptidyl peptidase IV inhibitors
Tsai, Ting-Yueh, Hsu, Tsu, Chen, Chiung-Tong, Cheng, Jai-Hong, Chiou, Mei-Chun, Huang, Chih-Hsiang, Tseng, Ya-Ju, Yeh, Teng-Kuang, Huang, Chung-Yu, Yeh, Kai-Chia, Huang, Yu-Wen, Wu, Ssu-Hui, Wang, Min-Hsien, Chen, Xin, Chao, Yu-Sheng, Jiaang, Weir-Torn
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
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Journal Article
Novel trans-2-aryl-cyclopropylamine analogues as potent and selective dipeptidyl peptidase IV inhibitors
Tsai, Ting-Yueh, Hsu, Tsu, Chen, Chiung-Tong, Cheng, Jai-Hong, Yeh, Teng-Kuang, Chen, Xin, Huang, Chung-Yu, Chang, Chung-Nien, Yeh, Kai-Chia, Hsieh, Su-Huei, Chien, Chia-Hui, Chang, Yi-Wei, Huang, Chih-Hsiang, Huang, Yu-Wen, Huang, Chen-Lung, Wu, Ssu-Hui, Wang, Min-Hsien, Lu, Cheng-Tai, Chao, Yu-Sheng, Jiaang, Weir-Torn
Published in Bioorganic & medicinal chemistry (15.03.2009)
Published in Bioorganic & medicinal chemistry (15.03.2009)
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Journal Article
Analogues of 2-phenyl-ethenesulfonic acid phenyl ester have dual functions of inhibiting expression of inducible nitric oxide synthase and activating peroxisome proliferator-activated receptor γ
Lee, Yue-Zhi, Yang, Cheng-Wei, Kang, Iou-Jiun, Wu, Ssu-Hui, Chao, Yu-Sheng, Chern, Jyh-Haur, Lee, Shiow-Ju
Published in Bioorganic & medicinal chemistry (15.10.2008)
Published in Bioorganic & medicinal chemistry (15.10.2008)
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Journal Article
Corrigendum to “A three-dimensional pharmacophore model for dipeptidyl peptidase IV inhibitiors” [Eur. J. Med. Chem. 43 (2008) 1603–1611]
Lu, I.-Lin, Tsai, Keng-Chang, Chiang, Yi-Kun, Jiaang, Weir-Torn, Wu, Ssu-Hui, Mahindroo, Neeraj, Chien, Chia-Hui, Lee, Shiow-Ju, Chen, Xin, Chao, Yu-Sheng, Wu, Su-Ying
Published in European journal of medicinal chemistry (01.06.2009)
Published in European journal of medicinal chemistry (01.06.2009)
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Journal Article
Substituted pyrrolidine-2,4-dicarboxylic acid amides as potent dipeptidyl peptidase IV inhibitors
Tsai, Ting-Yueh, Coumar, Mohane Selvaraj, Hsu, Tsu, Hsieh, Hsing-Pang, Chien, Chia-Hui, Chen, Chiung-Tong, Chang, Chung-Nien, Lo, Yu-Kang, Wu, Ssu-Hui, Huang, Chung-Yu, Huang, Yu-Wen, Wang, Min-Hsien, Wu, Hsin-Yi, Lee, Hong-Jen, Chen, Xin, Chao, Yu-Sheng, Jiaang, Weir-Torn
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
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Journal Article
Benzothiazolium compounds: novel classes of inhibitors that suppress the nitric oxide production in RAW264.7 cells stimulated by LPS/IFNγ
Tseng, Huan-Yi, Wu, Ssu-Hui, Huang, Wen-Hsin, Wang, Shao-Fang, Yang, Yung-Ning, Mahindroo, Neeraj, Hsu, Tsu, Jiaang, Weir-Torn, Lee, Shiow-Ju
Published in Bioorganic & medicinal chemistry letters (15.04.2005)
Published in Bioorganic & medicinal chemistry letters (15.04.2005)
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Journal Article
2-[3-[2-[(2S)-2-Cyano-1-pyrrolidinyl]-2-oxoethylamino]-3-methyl-1-oxobutyl]- 1,2,3,4-tetrahydroisoquinoline: A Potent, Selective, and Orally Bioavailable Dipeptide-Derived Inhibitor of Dipeptidyl Peptidase IV
Tsu, Hsu, Chen, Xin, Chen, Chiung-Tong, Lee, Shiow-Ju, Chang, Chung-Nien, Kao, Kuo-His, Coumar, Mohane Selvaraj, Yeh, Yen-Ting, Chien, Chia-Hui, Wang, Hsin-Sheng, Lin, Ke-Ta, Chang, Ying-Ying, Wu, Ssu-Hui, Chen, Yuan-Shou, Lu, I-Lin, Wu, Su-Ying, Tsai, Ting-Yueh, Chen, Wei-Cheng, Hsieh, Hsing-Pang, Chao, Yu-Sheng, Jiaang, Weir-Torn
Published in Journal of medicinal chemistry (12.01.2006)
Published in Journal of medicinal chemistry (12.01.2006)
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Journal Article
Novel Isoindoline Compounds for Potent and Selective Inhibition of Prolyl Dipeptidase DPP8
Jiaang, Weir-Torn, Chen, Yuan-Shou, Hsu, Tsu, Wu, Ssu-Hui, Chien, Chia-Hui, Chang, Chung-Nien, Chang, Sheng-Ping, Lee, Shiow-Ju, Chen, Xin
Published in ChemInform (21.06.2005)
Published in ChemInform (21.06.2005)
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Journal Article
3-[2-((2 S)-2-Cyano-pyrrolidin-1-yl)-2-oxo-ethylamino]-3-methyl-butyramide analogues as selective DPP-IV inhibitors for the treatment of type-II diabetes
Coumar, Mohane Selvaraj, Chang, Chung-Nien, Chen, Chiung-Tong, Chen, Xin, Chien, Chia-Hui, Tsai, Ting-Yueh, Cheng, Jai-Hong, Wu, Hsin-Yi, Han, Chia-Hung, Wu, Ssu-Hui, Huang, Yu-Wen, Hsu, Tsu, Hsu, Li-Jen, Chao, Yu-Sheng, Hsieh, Hsing-Pang, Jiaang, Weir-Torn
Published in Bioorganic & medicinal chemistry letters (01.03.2007)
Published in Bioorganic & medicinal chemistry letters (01.03.2007)
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Journal Article
Benzothiazolium compounds: novel classes of inhibitors that suppress the nitric oxide production in RAW264.7 cells stimulated by LPS/IFNgamma
Tseng, Huan-Yi, Wu, Ssu-Hui, Huang, Wen-Hsin, Wang, Shao-Fang, Yang, Yung-Ning, Mahindroo, Neeraj, Hsu, Tsu, Jiaang, Weir-Torn, Lee, Shiow-Ju
Published in Bioorganic & medicinal chemistry letters (15.04.2005)
Get full text
Published in Bioorganic & medicinal chemistry letters (15.04.2005)
Journal Article
Analogues of 2-phenyl-ethenesulfonic acid phenyl ester have dual functions of inhibiting expression of inducible nitric oxide synthase and activating peroxisome proliferator-activated receptor y
LEE, Yue-Zhi, YANG, Cheng-Wei, KANG, Iou-Jiun, WU, Ssu-Hui, CHAO, Yu-Sheng, CHERN, Jyh-Haur, LEE, Shiow-Ju
Published in Bioorganic & medicinal chemistry letters (2008)
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Published in Bioorganic & medicinal chemistry letters (2008)
Journal Article
Benzothiazolium compounds : novel classes of inhibitors that suppress the nitric oxide production in RAW264.7 cells stimulated by LPS/IFN
TSENG, Huan-Yi, WU, Ssu-Hui, HUANG, Wen-Hsin, WANG, Shao-Fang, YANG, Yung-Ning, MAHINDROO, Neeraj, HSU, Tsu, JIAANG, Weir-Torn, LEE, Shiow-Ju
Published in Bioorganic & medicinal chemistry letters (2005)
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Published in Bioorganic & medicinal chemistry letters (2005)
Journal Article