Targeting Pharmacokinetic Drug Resistance in Acute Myeloid Leukemia Cells with CDK4/6 Inhibitors
Sorf, Ales, Sucha, Simona, Morell, Anselm, Novotna, Eva, Staud, Frantisek, Zavrelova, Alzbeta, Visek, Benjamin, Wsol, Vladimir, Ceckova, Martina
Published in Cancers (16.06.2020)
Published in Cancers (16.06.2020)
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Journal Article
Inactivation of the anticancer drugs doxorubicin and oracin by aldo–keto reductase (AKR) 1C3
Novotna, Romana, Wsol, Vladimir, Xiong, Guangming, Maser, Edmund
Published in Toxicology letters (10.09.2008)
Published in Toxicology letters (10.09.2008)
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Journal Article
Acetylcholinesterase Inhibitors and Drugs Acting on Muscarinic Receptors- Potential Crosstalk of Cholinergic Mechanisms During Pharmacological Treatment
Soukup, Ondrej, Winder, Michael, Killi, Uday Kumar, Wsol, Vladimir, Jun, Daniel, Kuca, Kamil, Tobin, Gunnar
Published in Current neuropharmacology (01.01.2017)
Published in Current neuropharmacology (01.01.2017)
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Journal Article
Structural basis for substrate specificity in human monomeric carbonyl reductases
Pilka, Ewa S, Niesen, Frank H, Lee, Wen Hwa, El-Hawari, Yasser, Dunford, James E, Kochan, Grazyna, Wsol, Vladimir, Martin, Hans-Joerg, Maser, Edmund, Oppermann, Udo
Published in PloS one (20.10.2009)
Published in PloS one (20.10.2009)
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Journal Article
Inhibition of Nitric Oxide Synthase Prevents Muscarinic and Purinergic Functional Changes and Development of Cyclophosphamide-Induced Cystitis in the Rat
Aronsson, Patrik, Vesela, Renata, Johnsson, Martin, Tayem, Yasin I., Wsol, Vladimir, Winder, Michael, Tobin, Gunnar
Published in BioMed research international (01.01.2014)
Published in BioMed research international (01.01.2014)
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Journal Article
In vitro functional interactions of acetylcholine esterase inhibitors and muscarinic receptor antagonists in the urinary bladder of the rat
Killi, Uday K, Wsol, Vladimir, Soukup, Ondrej, Kuca, Kamil, Winder, Michael, Tobin, Gunnar
Published in Clinical and experimental pharmacology & physiology (01.02.2014)
Published in Clinical and experimental pharmacology & physiology (01.02.2014)
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Journal Article
Enzyme stereospecificity as a powerful tool in searching for new enzymes
Skarydová, Lucie, Skarka, Adam, Solich, Petr, Wsól, Vladimír
Published in Current drug metabolism (01.07.2010)
Published in Current drug metabolism (01.07.2010)
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Journal Article
Flavones Inhibit the Activity of AKR1B10, a Promising Therapeutic Target for Cancer Treatment
Zemanova, Lucie, Hofman, Jakub, Novotna, Eva, Musilek, Kamil, Lundova, Tereza, Havrankova, Jana, Hostalkova, Anna, Chlebek, Jakub, Cahlikova, Lucie, Wsol, Vladimír
Published in Journal of natural products (Washington, D.C.) (25.11.2015)
Published in Journal of natural products (Washington, D.C.) (25.11.2015)
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Journal Article
Hydantoins and thiohydantoins derived from 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Jansa, Petr, Wsol, Vladimir, Bertolasi, Valerio, Machacek, Vladimir
Published in Heterocycles (01.12.2006)
Published in Heterocycles (01.12.2006)
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Journal Article
Deeper Insight into the Reducing Biotransformation of Bupropion in the Human Liver
Lucie SKARYDOVA, Radana TOMANOVA, Lucie HAVLIKOVA, Hana STAMBERGOVA, Petr SOLICH, Vladimir WSOL
Published in DRUG METABOLISM AND PHARMACOKINETICS (25.04.2014)
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Published in DRUG METABOLISM AND PHARMACOKINETICS (25.04.2014)
Journal Article
Buparlisib is a novel inhibitor of daunorubicin reduction mediated by aldo-keto reductase 1C3
Bukum, Neslihan, Novotna, Eva, Morell, Anselm, Hofman, Jakub, Wsol, Vladimir
Published in Chemico-biological interactions (01.04.2019)
Published in Chemico-biological interactions (01.04.2019)
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Journal Article
Synthesis and Biological Activity of Quaternary Ammonium Salt-Type Agents Containing Cholesterol and Terpenes
Novotná, Eva, Waisser, Karel, Kuneš, Jiří, Palát, Karel, Buchta, Vladimír, Stolaříková, Jiřina, Beckert, Rainer, Wsól, Vladimír
Published in Archiv der Pharmazie (Weinheim) (01.06.2014)
Published in Archiv der Pharmazie (Weinheim) (01.06.2014)
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Journal Article
Pharmacokinetic interactions of breast cancer chemotherapeutics with human doxorubicin reductases
Hofman, Jakub, Skarka, Adam, Havrankova, Jana, Wsol, Vladimir
Published in Biochemical pharmacology (01.08.2015)
Published in Biochemical pharmacology (01.08.2015)
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