Synthesis of Urea-Based Inhibitors as Active Site Probes of Glutamate Carboxypeptidase II: Efficacy as Analgesic Agents
Kozikowski, Alan P, Zhang, Jiazhong, Nan, Fajun, Petukhov, Pavel A, Grajkowska, Ewa, Wroblewski, Jarda T, Yamamoto, Tatsuo, Bzdega, Tomasz, Wroblewska, Barbara, Neale, Joseph H
Published in Journal of medicinal chemistry (25.03.2004)
Published in Journal of medicinal chemistry (25.03.2004)
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Chloride is an Agonist of Group II and III Metabotropic Glutamate Receptors
DiRaddo, John O, Miller, Eric J, Bowman-Dalley, Carrie, Wroblewska, Barbara, Javidnia, Monica, Grajkowska, Ewa, Wolfe, Barry B, Liotta, Dennis C, Wroblewski, Jarda T
Published in Molecular pharmacology (01.09.2015)
Published in Molecular pharmacology (01.09.2015)
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Metabotropic glutamate receptor 1 acts as a dependence receptor creating a requirement for glutamate to sustain the viability and growth of human melanomas
Gelb, T, Pshenichkin, S, Rodriguez, O C, Hathaway, H A, Grajkowska, E, DiRaddo, J O, Wroblewska, B, Yasuda, R P, Albanese, C, Wolfe, B B, Wroblewski, J T
Published in Oncogene (21.05.2015)
Published in Oncogene (21.05.2015)
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l-Homocysteine Sulfinic Acid and Other Acidic Homocysteine Derivatives Are Potent and Selective Metabotropic Glutamate Receptor Agonists
Shi, Qi, Savage, Jason E, Hufeisen, Sandra J, Rauser, Laura, Grajkowska, Ewa, Ernsberger, Paul, Wroblewski, Jarda T, Nadeau, Joseph H, Roth, Bryan L
Published in The Journal of pharmacology and experimental therapeutics (01.04.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2003)
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Dual neurotoxic and neuroprotective role of metabotropic glutamate receptor 1 in conditions of trophic deprivation – Possible role as a dependence receptor
Pshenichkin, Sergey, Dolińska, Monika, Klauzińska, Małgorzata, Luchenko, Victoria, Grajkowska, Ewa, Wroblewski, Jarda T.
Published in Neuropharmacology (01.09.2008)
Published in Neuropharmacology (01.09.2008)
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Design of Remarkably Simple, Yet Potent Urea-Based Inhibitors of Glutamate Carboxypeptidase II (NAALADase)
Kozikowski, Alan P, Nan, Fajun, Conti, Paola, Zhang, Jiazhong, Ramadan, Epolia, Bzdega, Tomasz, Wroblewska, Barbara, Neale, Joseph H, Pshenichkin, Sergey, Wroblewski, Jarda T
Published in Journal of medicinal chemistry (01.02.2001)
Published in Journal of medicinal chemistry (01.02.2001)
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NAAG peptidase inhibition reduces locomotor activity and some stereotypes in the PCP model of schizophrenia via group II mGluR
Olszewski, Rafal T., Bukhari, Noreen, Zhou, Jia, Kozikowski, Alan P., Wroblewski, Jarda T., Shamimi‐Noori, Susan, Wroblewska, Barbara, Bzdega, Tomasz, Vicini, Stefano, Barton, Franca B., Neale, Joseph H.
Published in Journal of neurochemistry (01.05.2004)
Published in Journal of neurochemistry (01.05.2004)
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Metabotropic glutamate receptors: From the workbench to the bedside
Nicoletti, F., Bockaert, J., Collingridge, G.L., Conn, P.J., Ferraguti, F., Schoepp, D.D., Wroblewski, J.T., Pin, J.P.
Published in Neuropharmacology (01.06.2011)
Published in Neuropharmacology (01.06.2011)
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Synthesis and Structure−Activity Relationships of 3-[(2-Methyl-1,3-thiazol-4-yl)ethynyl]pyridine Analogues as Potent, Noncompetitive Metabotropic Glutamate Receptor Subtype 5 Antagonists; Search for Cocaine Medications
Iso, Yasuyoshi, Grajkowska, Ewa, Wroblewski, Jarda T, Davis, Jared, Goeders, Nicholas E, Johnson, Kenneth M, Sanker, Subramaniam, Roth, Bryan L, Tueckmantel, Werner, Kozikowski, Alan P
Published in Journal of medicinal chemistry (09.02.2006)
Published in Journal of medicinal chemistry (09.02.2006)
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Diffuse cavernous hemangioma of rectosigmoid colon treated with n-butyl-2-cyanoacrylate injections
Żurakowski, J., Świercz, P., Wróblewski, T., Paluszkiewicz, R., Patkowski, W., Smoter, P., Dudek, K., Leonowicz, D., Nawrot, I., Ziarkiewicz-Wróblewska, B., Szmidt, J.
Published in Endoscopy (01.09.2008)
Published in Endoscopy (01.09.2008)
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Biliary Complications in Relation to the Technique of Biliary Reconstruction in Adult Liver Transplant Recipients
Alsharabi, A, Zieniewicz, K, Michałowicz, B, Patkowski, W, Nyckowski, P, Wróblewski, T, Grzelak, I, Paluszkiewicz, R, Hevelke, P, Remiszewski, P, Cieślak, B, Kornasiewicz, O, Kotulski, M, Skwarek, A, Urban, M, Sańko-Resmer, J, Krawczyk, M
Published in Transplantation proceedings (01.11.2007)
Published in Transplantation proceedings (01.11.2007)
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Conference Proceeding
Surface and bulk residual stresses in Li2O· 2SiO2 glass-ceramics
PINTO, H, ITO, L, CROVACE, M, FERREIRA, E. B, FAUTH, F, WROBLEWSKI, T, ZANOTTO, E. D, PYZALLA, A. R
Published in Journal of non-crystalline solids (15.07.2007)
Published in Journal of non-crystalline solids (15.07.2007)
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Lattice misfit measurement in Inconel 706 containing coherent γ ′ and γ″ precipitates
Mukherji, D, Gilles, R, Barbier, B, Genovese, D.Del, Hasse, B, Strunz, P, Wroblewski, T, Fuess, H, Rösler, J
Published in Scripta materialia (01.02.2003)
Published in Scripta materialia (01.02.2003)
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