Proteolysis Targeting Chimera (PROTAC) for Macrophage Migration Inhibitory Factor (MIF) Has Anti‐Proliferative Activity in Lung Cancer Cells
Xiao, Zhangping, Song, Shanshan, Chen, Deng, Merkerk, Ronald, Wouden, Petra E., Cool, Robbert H., Quax, Wim J., Poelarends, Gerrit J., Melgert, Barbro N., Dekker, Frank J.
Published in Angewandte Chemie International Edition (02.08.2021)
Published in Angewandte Chemie International Edition (02.08.2021)
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Identification of a Bromodomain‐like Region in 15‐Lipoxygenase‐1 Explains Its Nuclear Localization
Chen, Deng, Xiao, Zhangping, Guo, Hao, Gogishvili, Dea, Setroikromo, Rita, Wouden, Petra E., Dekker, Frank J.
Published in Angewandte Chemie International Edition (27.09.2021)
Published in Angewandte Chemie International Edition (27.09.2021)
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A next-generation sequencing method for gene doping detection that distinguishes low levels of plasmid DNA against a background of genomic DNA
de Boer, Eddy N., van der Wouden, Petra E., Johansson, Lennart F., van Diemen, Cleo C., Haisma, Hidde J.
Published in Gene therapy (01.08.2019)
Published in Gene therapy (01.08.2019)
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4‐Iodopyrimidine Labeling Reveals Nuclear Translocation and Nuclease Activity for Both MIF and MIF2
Xiao, Zhangping, Chen, Deng, Mulder, Fabian, Song, Shanshan, Wouden, Petra E., Cool, Robbert H., Melgert, Barbro N., Poelarends, Gerrit J., Dekker, Frank J.
Published in Chemistry : a European journal (03.01.2022)
Published in Chemistry : a European journal (03.01.2022)
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Induced protein degradation of histone deacetylases 3 (HDAC3) by proteolysis targeting chimera (PROTAC)
Cao, Fangyuan, de Weerd, Sander, Chen, Deng, Zwinderman, Martijn R.H., van der Wouden, Petra E., Dekker, Frank J.
Published in European journal of medicinal chemistry (15.12.2020)
Published in European journal of medicinal chemistry (15.12.2020)
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Small Molecule MIF Modulation Enhances Ferroptosis by Impairing DNA Repair Mechanisms
Chen, Deng, Zhao, Chunlong, Zhang, Jianqiu, Knol, Catharina W. J., Osipyan, Angelina, Majerníková, Nad'a, Chen, Tingting, Xiao, Zhangping, Adriana, Jeaunice, Griffith, Andrew J., Gamez, Abel Soto, Wouden, Petra E., Coppes, Robert P., Dolga, Amalia M., Haisma, Hidde J., Dekker, Frank J.
Published in Advanced science (01.08.2024)
Published in Advanced science (01.08.2024)
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Protocol of the Double‐Click Seq Method to Evaluate the Deposition Bias of Chromatin Proteins
Wouden, Petra E., Zwinderman, Martijn R. H., Chen, Deng, Borghesan, Michela, Dekker, Frank J.
Published in Current protocols (01.06.2023)
Published in Current protocols (01.06.2023)
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Histone Deacetylase 3-Directed PROTACs Have Anti-inflammatory Potential by Blocking Polarization of M0-like into M1-like Macrophages
Zhao, Chunlong, Chen, Shipeng, Chen, Deng, Rio-Berge, Claudia, Zhang, Jianqiu, Van Der Wouden, Petra E., Daemen, Toos, Dekker, Frank J.
Published in Angewandte Chemie International Edition (16.10.2023)
Published in Angewandte Chemie International Edition (16.10.2023)
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Light-controlled inhibition of BRAFV600E kinase
Hoorens, Mark W.H., Ourailidou, Maria E., Rodat, Theo, van der Wouden, Petra E., Kobauri, Piermichele, Kriegs, Malte, Peifer, Christian, Feringa, Ben L., Dekker, Frank J., Szymanski, Wiktor
Published in European journal of medicinal chemistry (01.10.2019)
Published in European journal of medicinal chemistry (01.10.2019)
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HDAC1-3 inhibitor MS-275 enhances IL10 expression in RAW264.7 macrophages and reduces cigarette smoke-induced airway inflammation in mice
Leus, Niek G. J., van den Bosch, Thea, van der Wouden, Petra E., Krist, Kim, Ourailidou, Maria E., Eleftheriadis, Nikolaos, Kistemaker, Loes E. M., Bos, Sophie, Gjaltema, Rutger A. F., Mekonnen, Solomon A., Bischoff, Rainer, Gosens, Reinoud, Haisma, Hidde J., Dekker, Frank J.
Published in Scientific reports (27.03.2017)
Published in Scientific reports (27.03.2017)
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De novo CoA biosynthesis is required to maintain DNA integrity during development of the Drosophila nervous system
Bosveld, Floris, Rana, Anil, van der Wouden, Petra E., Lemstra, Willy, Ritsema, Martha, Kampinga, Harm H., Sibon, Ody C. M.
Published in Human molecular genetics (01.07.2008)
Published in Human molecular genetics (01.07.2008)
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Proteolysis Targeting Chimera (PROTAC) for Macrophage Migration Inhibitory Factor (MIF) Has Anti‐Proliferative Activity in Lung Cancer Cells
Xiao, Zhangping, Song, Shanshan, Chen, Deng, Merkerk, Ronald, Wouden, Petra E., Cool, Robbert H., Quax, Wim J., Poelarends, Gerrit J., Melgert, Barbro N., Dekker, Frank J.
Published in Angewandte Chemie (02.08.2021)
Published in Angewandte Chemie (02.08.2021)
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Thieno[2,3‑d]pyrimidine-2,4(1H,3H)‑dione Derivative Inhibits d‑Dopachrome Tautomerase Activity and Suppresses the Proliferation of Non-Small Cell Lung Cancer Cells
Xiao, Zhangping, Osipyan, Angelina, Song, Shanshan, Chen, Deng, Schut, Reinder A, van Merkerk, Ronald, van der Wouden, Petra E, Cool, Robbert H, Quax, Wim J, Melgert, Barbro N, Poelarends, Gerrit J, Dekker, Frank J
Published in Journal of medicinal chemistry (10.02.2022)
Published in Journal of medicinal chemistry (10.02.2022)
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Allosteric Inhibitors of Macrophage Migration Inhibitory Factor (MIF) Interfere with Apoptosis-Inducing Factor (AIF) Co-Localization to Prevent Parthanatos
Chen, Deng, Osipyan, Angelina, Adriana, Jeaunice, Kader, Mohammed, Gureev, Maxim, Knol, Catharina W. J., Sigmund, Marie-Cathérine, Xiao, Zhangping, van der Wouden, Petra E., Cool, Robbert H., Poelarends, Gerrit J., Dekker, Frank J.
Published in Journal of medicinal chemistry (13.07.2023)
Published in Journal of medicinal chemistry (13.07.2023)
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HDAC 3-selective inhibitor RGFP966 demonstrates anti-inflammatory properties in RAW 264.7 macrophages and mouse precision-cut lung slices by attenuating NF-κB p65 transcriptional activity
Leus, Niek G.J., van der Wouden, Petra E., van den Bosch, Thea, Hooghiemstra, Wouter T.R., Ourailidou, Maria E., Kistemaker, Loes E.M., Bischoff, Rainer, Gosens, Reinoud, Haisma, Hidde J., Dekker, Frank J.
Published in Biochemical pharmacology (15.05.2016)
Published in Biochemical pharmacology (15.05.2016)
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The synthesis of 1,2,3-triazoles as binders of D-dopachrome tautomerase (D-DT) for the development of dual-targeting inhibitors
Osipyan, Angelina, Bulai, Radu-George, Wu, Zhengyang, de Witte, Jarno, van der Velde, Jesse J.H., Kader, Mohammed, van der Wouden, Petra E., Poelarends, Gerrit J., Dekker, Frank J.
Published in European journal of medicinal chemistry (05.10.2024)
Published in European journal of medicinal chemistry (05.10.2024)
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7‑Hydroxycoumarins Are Affinity-Based Fluorescent Probes for Competitive Binding Studies of Macrophage Migration Inhibitory Factor
Xiao, Zhangping, Chen, Deng, Song, Shanshan, van der Vlag, Ramon, van der Wouden, Petra E, van Merkerk, Ronald, Cool, Robbert H, Hirsch, Anna K. H, Melgert, Barbro N, Quax, Wim J, Poelarends, Gerrit J, Dekker, Frank J
Published in Journal of medicinal chemistry (22.10.2020)
Published in Journal of medicinal chemistry (22.10.2020)
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Rational Development of a Potent 15-Lipoxygenase‑1 Inhibitor with in Vitro and ex Vivo Anti-inflammatory Properties
Eleftheriadis, Nikolaos, Neochoritis, Constantinos G., Leus, Niek G. J., van der Wouden, Petra E., Dömling, Alexander, Dekker, Frank J.
Published in Journal of medicinal chemistry (08.10.2015)
Published in Journal of medicinal chemistry (08.10.2015)
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