Discovery of CMX990: A Potent SARS-CoV‑2 3CL Protease Inhibitor Bearing a Novel Warhead
Dayan Elshan, N. G. R., Wolff, Karen C., Riva, Laura, Woods, Ashley K., Grabovyi, Gennadii, Wilson, Katy, Pedroarena, James, Ghorai, Sourav, Nazarian, Armen, Weiss, Frank, Liu, Yuyin, Mazumdar, Wrickban, Song, Lirui, Okwor, Neechi, Malvin, Jacqueline, Bakowski, Malina A., Beutler, Nathan, Kirkpatrick, Melanie G., Gebara-Lamb, Amal, Huang, Edward, Nguyen-Tran, Vân T. B., Chi, Victor, Li, Shuangwei, Rogers, Thomas F., McNamara, Case W., Gupta, Anil Kumar, Rahimi, Alireza, Chen, Jian Jeffrey, Joseph, Sean B., Schultz, Peter G., Chatterjee, Arnab K.
Published in Journal of medicinal chemistry (22.02.2024)
Published in Journal of medicinal chemistry (22.02.2024)
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Correction to “Discovery of CMX990: A Potent SARS-CoV‑2 3CL Protease Inhibitor Bearing a Novel Warhead”
Elshan, N. G. R. Dayan, Wolff, Karen C., Riva, Laura, Woods, Ashley K., Grabovyi, Gennadii, Wilson, Katy, Pedroarena, James, Ghorai, Sourav, Nazarian, Armen, Weiss, Frank, Liu, Yuyin, Mazumdar, Wrickban, Song, Lirui, Okwor, Neechi, Malvin, Jacqueline, Liu, Dongdong, Bakowski, Malina A., Beutler, Nathan, Kirkpatrick, Melanie G., Gebara-Lamb, Amal, Huang, Edward, Nguyen-Tran, Vân T. B., Chi, Victor, Li, Shuangwei, Rogers, Thomas F., McNamara, Case W., Gupta, Anil Kumar, Rahimi, Alireza, Chen, Jian Jeffrey, Joseph, Sean B., Schultz, Peter G., Chatterjee, Arnab K.
Published in Journal of medicinal chemistry (27.06.2024)
Published in Journal of medicinal chemistry (27.06.2024)
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Dexamethasone inhibits respiratory syncytial virus-driven mucus production while increasing viral replication without altering antiviral interferon signaling
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Published in Virology (New York, N.Y.) (15.01.2020)
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Design, synthesis and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part I
Jiang, Tao, Kuhen, Kelli L., Wolff, Karen, Yin, Hong, Bieza, Kimberly, Caldwell, Jeremy, Bursulaya, Badry, Wu, Tom Yao-Hsing, He, Yun
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
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Drug repurposing screens identify chemical entities for the development of COVID-19 interventions
Bakowski, Malina A, Beutler, Nathan, Wolff, Karen C, Kirkpatrick, Melanie G, Chen, Emily, Nguyen, Tu-Trinh H, Riva, Laura, Shaabani, Namir, Parren, Mara, Ricketts, James, Gupta, Anil K, Pan, Kastin, Kuo, Peiting, Fuller, MacKenzie, Garcia, Elijah, Teijaro, John R, Yang, Linlin, Sahoo, Debashis, Chi, Victor, Huang, Edward, Vargas, Natalia, Roberts, Amanda J, Das, Soumita, Ghosh, Pradipta, Woods, Ashley K, Joseph, Sean B, Hull, Mitchell V, Schultz, Peter G, Burton, Dennis R, Chatterjee, Arnab K, McNamara, Case W, Rogers, Thomas F
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Published in Nature communications (03.06.2021)
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Design, synthesis, and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part 2
Jiang, Tao, Kuhen, Kelli L., Wolff, Karen, Yin, Hong, Bieza, Kimberly, Caldwell, Jeremy, Bursulaya, Badry, Tuntland, Tove, Zhang, Kanyin, Karanewsky, Donald, He, Yun
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
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Identification of broad-spectrum antiviral compounds and assessment of the druggability of their target for efficacy against respiratory syncytial virus (RSV)
Bonavia, Aurelio, Franti, Michael, Pusateri Keaney, Erin, Kuhen, Kelli, Seepersaud, Mohindra, Radetich, Branko, Shao, Jian, Honda, Ayako, Dewhurst, Janetta, Balabanis, Kara, Monroe, James, Wolff, Karen, Osborne, Colin, Lanieri, Leanne, Hoffmaster, Keith, Amin, Jakal, Markovits, Judit, Broome, Michelle, Skuba, Elizabeth, Cornella-Taracido, Ivan, Joberty, Gerard, Bouwmeester, Tewis, Hamann, Lawrence, Tallarico, John A, Tommasi, Ruben, Compton, Teresa, Bushell, Simon M
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Published in Proceedings of the National Academy of Sciences - PNAS (26.04.2011)
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“UnPAKing” Human Immunodeficiency Virus (HIV) Replication: Using Small Interfering RNA Screening To Identify Novel Cofactors and Elucidate the Role of Group I PAKs in HIV Infection
NGUYEN, Deborah G, WOLFF, Karen C, HONG YIN, CALDWELL, Jeremy S, KUHEN, Kelli L
Published in Journal of Virology (01.01.2006)
Published in Journal of Virology (01.01.2006)
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Mutations in an Auxin Receptor Homolog AFB5 and in SGT1b Confer Resistance to Synthetic Picolinate Auxins and Not to 2,4-Dichlorophenoxyacetic Acid or Indole-3-Acetic Acid in Arabidopsis
Walsh, Terence A, Neal, Roben, Merlo, Ann Owens, Honma, Mary, Hicks, Glenn R, Wolff, Karen, Matsumura, Wendy, Davies, John P
Published in Plant physiology (Bethesda) (01.10.2006)
Published in Plant physiology (Bethesda) (01.10.2006)
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NAZARIAN ARMEN, MAZUMDAR WRICKBAN, GRABOVYI GENNADII, OKWOR NEECHI, ROGERS THOMAS F, JOSEPH SEAN, RIVA LAURA, GHORAI SOURAV, LIU YUYIN, GUPTA ANIL KUMAR, MALVIN JACQUELINE, CHATTERJEE ARNAB K, BAKOWSKI MALINA A, WILSON KATY, WEISS FRANK, WOLFF KAREN, WOODS ASHLEY, CHEN JIAN JEFFREY, RAHIMI ALIREZA, LI SHUANGWEI, SONG LIRUI, NAKATH ELSHAN, PEDROARENA JAMES, MCNAMARA CASE W
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Year of Publication 15.03.2024
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Design, synthesis, and biological evaluations of novel quinolones as HIV-1 non-nucleoside reverse transcriptase inhibitors
Ellis, David, Kuhen, Kelli L., Anaclerio, Beth, Wu, Baogen, Wolff, Karen, Yin, Hong, Bursulaya, Badry, Caldwell, Jeremy, Karanewsky, Donald, He, Yun
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
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Chemical Genetic Identification of Glutamine Phosphoribosylpyrophosphate Amidotransferase as the Target for a Novel Bleaching Herbicide in Arabidopsis
Walsh, Terence A, Bauer, Teresa, Neal, Roben, Merlo, Ann Owens, Schmitzer, Paul R, Hicks, Glenn R, Honma, Mary, Matsumura, Wendy, Wolff, Karen, Davies, John P
Published in Plant physiology (Bethesda) (01.07.2007)
Published in Plant physiology (Bethesda) (01.07.2007)
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Synthesis and evaluation of N-aryl pyrrolidinones as novel anti-HIV-1 agents. Part 1
Wu, Baogen, Kuhen, Kelli, Ngoc Nguyen, Truc, Ellis, David, Anaclerio, Beth, He, Xiaohui, Yang, Kunyong, Karanewsky, Donald, Yin, Hong, Wolff, Karen, Bieza, Kimberly, Caldwell, Jeremy, He, Yun
Published in Bioorganic & medicinal chemistry letters (01.07.2006)
Published in Bioorganic & medicinal chemistry letters (01.07.2006)
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Corrosion monitoring with speckle correlation
Fricke-Begemann, T, Gülker, G, Hinsch, K D, Wolff, K
Published in Applied optics (2004) (01.10.1999)
Published in Applied optics (2004) (01.10.1999)
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Homogeneous High-Throughput Screening Assays for HIV-1 Integrase 3'-Processing and Strand Transfer Activities
Wang, Yu, Klock, Heath, Yin, Hong, Wolff, Karen, Bieza, Kimberly, Niswonger, Kirk, Matzen, Jason, Gunderson, Drew, Hale, Joanna, Lesley, Scott, Kuhen, Kelli, Caldwell, Jeremy, Brinker, Achim
Published in SLAS discovery (01.08.2005)
Published in SLAS discovery (01.08.2005)
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Just-in-time purification: an effective solution for cherry-picking and purifying active compounds from large legacy libraries
Guintu, Christina, Kwok, Michael, Hanlon, James J, Spalding, Tracy A, Wolff, Karen, Yin, Hong, Kuhen, Kelli, Sasher, Kimberly, Calvin, Paul, Jiang, Shumei, Zhou, Yingyao, Isbell, John J
Published in Journal of biomolecular screening (01.12.2006)
Published in Journal of biomolecular screening (01.12.2006)
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METHODS AND COMPOSITIONS FOR THE TREATMENT OF SARS-COV-2
ROGERS, Thomas F, BEUTLER, Nathan, CHATTERJEE, Arnab K, MCNAMARA, Case W, RIVA, Laura, BAKOWSKI, Malina A, SCHULTZ, Peter G, WOLFF, Karen, BURTON, Dennis R
Year of Publication 02.11.2023
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Year of Publication 02.11.2023
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