Chemoselective Suzuki-Miyaura reactions of 4-bromo-3-O-triflylestrone. Synthesis and atropisomerism of arylated estrones
Jopp, Stefan, Wallaschkowski, Tina, Ehlers, Peter, Frank, Eva, Schneider, Gyula, Woelfling, Janos, Mernyak, Erzsebet, Villinger, Alexander, Langer, Peter
Published in Tetrahedron (07.06.2018)
Published in Tetrahedron (07.06.2018)
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Efficient Approach to Androstene-Fused Arylpyrazolines as Potent Antiproliferative Agents. Experimental and Theoretical Studies of Substituent Effects on BF3-Catalyzed Intramolecular [3+2] Cycloadditions of Olefinic Phenylhydrazonest
Frank, Eva, Mucsi, Zoltan, Zupko, Istvan, Rethy, Borbala, Falkay, George, Schneider, Gyula, Woelfling, Janos
Published in Journal of the American Chemical Society (25.03.2009)
Published in Journal of the American Chemical Society (25.03.2009)
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An efficient approach to novel 17-5 '-(1 ',2 ',4 ')-oxadiazolyl androstenes via the cyclodehydration of cytotoxic O-steroidacylamidoximes, and an evaluation of their inhibitory action on 17 alpha-hydroxylase/C-17,C-20-lyase
Kovacs, Dora, Woelfling, Janos, Szabo, Nikoletta, Szecsi, Mihaly, Kovacs, Ida, Zupko, Istvan, Frank, Eva
Published in European journal of medicinal chemistry (01.12.2013)
Published in European journal of medicinal chemistry (01.12.2013)
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Journal Article
Efficient access to novel androsteno-17-(1′,3′,4′)-oxadiazoles and 17β-(1′,3′,4′)-thiadiazoles via N-substituted hydrazone and N,N′-disubstituted hydrazine intermediates, and their pharmacological evaluation in vitro
Kovács, Dóra, Wölfling, János, Szabó, Nikoletta, Szécsi, Mihály, Minorics, Renáta, Zupkó, István, Frank, Éva
Published in European journal of medicinal chemistry (15.06.2015)
Published in European journal of medicinal chemistry (15.06.2015)
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Journal Article
Microwave-assisted one-pot synthesis of steroid–quinoline hybrids and an evaluation of their antiproliferative activities on gynecological cancer cell lines
Baji, Ádám, Gyovai, András, Wölfling, János, Minorics, Renáta, Ocsovszki, Imre, Zupkó, István, Frank, Éva
Published in RSC advances (01.01.2016)
Published in RSC advances (01.01.2016)
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Journal Article
A facile access to novel steroidal 17-2 '-(1 ',3 ',4 ')-oxadiazoles, and an evaluation of their cytotoxic activities in vitro
Kovacs, Dora, Motyan, Gergo, Woelfling, Janos, Kovacs, Ida, Zupko, Istvan, Frank, Eva
Published in Bioorganic & medicinal chemistry letters (01.03.2014)
Published in Bioorganic & medicinal chemistry letters (01.03.2014)
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A molecular understanding of d‐homoestrone‐induced G2/M cell cycle arrest in HeLa human cervical carcinoma cells
Minorics, Renáta, Bózsity, Noémi, Molnár, Judit, Wölfling, János, Mernyák, Erzsébet, Schneider, Gyula, Ocsovszki, Imre, Zupkó, István
Published in Journal of cellular and molecular medicine (01.10.2015)
Published in Journal of cellular and molecular medicine (01.10.2015)
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Journal Article
Synthesis and in vitro investigation of potential antiproliferative monosaccharide–d-secoestrone bioconjugates
Bodnár, Brigitta, Mernyák, Erzsébet, Szabó, Johanna, Wölfling, János, Schneider, Gyula, Zupkó, István, Kupihár, Zoltán, Kovács, Lajos
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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Journal Article
Synthesis of antiproliferative 13α-d-homoestrones via Lewis acid-promoted one-pot Prins–Ritter reactions of d-secosteroidal δ-alkenyl-aldehydes
Huber, Judit, Wölfling, János, Schneider, Gyula, Ocsovszki, Imre, Varga, Mónika, Zupkó, István, Mernyák, Erzsébet
Published in Steroids (01.10.2015)
Published in Steroids (01.10.2015)
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Synthesis and investigation of the anticancer effects of estrone-16-oxime ethers in vitro
Berényi, Ágnes, Minorics, Renáta, Iványi, Zoltán, Ocsovszki, Imre, Ducza, Eszter, Thole, Hubert, Messinger, Josef, Wölfling, János, Mótyán, Gergő, Mernyák, Erzsébet, Frank, Éva, Schneider, Gyula, Zupkó, István
Published in Steroids (01.01.2013)
Published in Steroids (01.01.2013)
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Journal Article
Synthesis and in vitro antiproliferative evaluation of d-secooxime derivatives of 13β- and 13α-estrone
Mernyák, Erzsébet, Fiser, Gabriella, Szabó, Johanna, Bodnár, Brigitta, Schneider, Gyula, Kovács, Ida, Ocsovszki, Imre, Zupkó, István, Wölfling, János
Published in Steroids (01.11.2014)
Published in Steroids (01.11.2014)
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Journal Article
Synthesis of A-ring halogenated 13α-estrone derivatives as potential 17β-HSD1 inhibitors
Bacsa, Ildikó, Jójárt, Rebeka, Schneider, Gyula, Wölfling, János, Maróti, Péter, Herman, Bianka Edina, Szécsi, Mihály, Mernyák, Erzsébet
Published in Steroids (01.12.2015)
Published in Steroids (01.12.2015)
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Journal Article
CYP24A1 inhibition facilitates the anti-tumor effect of vitamin D3 on colorectal cancer cells
Kósa, János P, Horváth, Péter, Wölfling, János, Kovács, Dóra, Balla, Bernadett, Mátyus, Péter, Horváth, Evelin, Speer, Gábor, Takács, István, Nagy, Zsolt, Horváth, Henrik, Lakatos, Péter
Published in World journal of gastroenterology : WJG (07.05.2013)
Published in World journal of gastroenterology : WJG (07.05.2013)
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Journal Article
A click approach to novel D-ring-substituted 16α-triazolylestrone derivatives and characterization of their antiproliferative properties
Molnár, Judit, Frank, Éva, Minorics, Renáta, Kádár, Zalán, Ocsovszki, Imre, Schönecker, Bruno, Wölfling, János, Zupkó, István
Published in PloS one (18.02.2015)
Published in PloS one (18.02.2015)
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Journal Article
Antiproliferative effect of normal and 13-epi-d-homoestrone and their 3-methyl ethers on human reproductive cancer cell lines
Minorics, Renáta, Bózsity, Noémi, Wölfling, János, Mernyák, Erzsébet, Schneider, Gyula, Márki, Árpád, Falkay, George, Ocsovszki, Imre, Zupkó, István
Published in The Journal of steroid biochemistry and molecular biology (01.10.2012)
Published in The Journal of steroid biochemistry and molecular biology (01.10.2012)
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