Renal transporters in drug development
Morrissey, Kari M, Stocker, Sophie L, Wittwer, Matthias B, Xu, Lu, Giacomini, Kathleen M
Published in Annual review of pharmacology and toxicology (01.01.2013)
Published in Annual review of pharmacology and toxicology (01.01.2013)
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Transporters in Drug Development: 2018 ITC Recommendations for Transporters of Emerging Clinical Importance
Zamek-Gliszczynski, Maciej J, Taub, Mitchell E, Chothe, Paresh P, Chu, Xiaoyan, Giacomini, Kathleen M, Kim, Richard B, Ray, Adrian S, Stocker, Sophie L, Unadkat, Jashvant D, Wittwer, Matthias B, Xia, Cindy, Yee, Sook-Wah, Zhang, Lei, Zhang, Yan
Published in Clinical pharmacology and therapeutics (01.11.2018)
Published in Clinical pharmacology and therapeutics (01.11.2018)
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Transporters in drug development: International transporter consortium update on emerging transporters of clinical importance
Zamek-Gliszczynski, Maciej J, Sangha, Vishal, Shen, Hong, Feng, Bo, Wittwer, Matthias B, Varma, Manthena V S, Liang, Xiaomin, Sugiyama, Yuichi, Zhang, Lei, Bendayan, Reina
Published in Clinical pharmacology and therapeutics (01.09.2022)
Published in Clinical pharmacology and therapeutics (01.09.2022)
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Considerations and recommendations for assessment of plasma protein binding and drug-drug interactions for siRNA therapeutics
Humphreys, Sara C, Davis, John A, Iqbal, Sajida, Kamel, Amin, Kulmatycki, Kenneth, Lao, Yanbin, Liu, Xiumin, Rodgers, John, Snoeys, Jan, Vigil, Adam, Weng, Yan, Wiethoff, Christopher M, Wittwer, Matthias B
Published in Nucleic acids research (24.06.2022)
Published in Nucleic acids research (24.06.2022)
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Discovery of Potent, Selective Multidrug and Toxin Extrusion Transporter 1 (MATE1, SLC47A1) Inhibitors Through Prescription Drug Profiling and Computational Modeling
Wittwer, Matthias B, Zur, Arik A, Khuri, Natalia, Kido, Yasuto, Kosaka, Alan, Zhang, Xuexiang, Morrissey, Kari M, Sali, Andrej, Huang, Yong, Giacomini, Kathleen M
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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Involvement of CB1 and CB2 receptors in neuroprotective effects of cannabinoids in experimental TDP-43 related frontotemporal dementia using male mice
Gonzalo-Consuegra, Claudia, Santos-García, Irene, García-Toscano, Laura, Martín-Baquero, Raquel, Rodríguez-Cueto, Carmen, Wittwer, Matthias B., Dzygiel, Pawel, Grether, Uwe, de Lago, Eva, Fernández-Ruiz, Javier
Published in Biomedicine & pharmacotherapy (01.05.2024)
Published in Biomedicine & pharmacotherapy (01.05.2024)
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The Effect of Famotidine, a MATE1-Selective Inhibitor, on the Pharmacokinetics and Pharmacodynamics of Metformin
Hibma, Jennifer E., Zur, Arik A., Castro, Richard A., Wittwer, Matthias B., Keizer, Ron J., Yee, Sook Wah, Goswami, Srijib, Stocker, Sophie L., Zhang, Xuexiang, Huang, Yong, Brett, Claire M., Savic, Radojka M., Giacomini, Kathleen M.
Published in Clinical pharmacokinetics (01.06.2016)
Published in Clinical pharmacokinetics (01.06.2016)
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Fundamental aspects of DMPK optimization of targeted protein degraders
Cantrill, Carina, Chaturvedi, Prasoon, Rynn, Caroline, Petrig Schaffland, Jeannine, Walter, Isabelle, Wittwer, Matthias B.
Published in Drug discovery today (01.06.2020)
Published in Drug discovery today (01.06.2020)
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P17.08 RENAL THROMBOTIC MICROANGIOPATHY INDUCED BY BEVACIZUMAB IN HIGH GRADE GLIOMA PATIENTS - ABOUT SIX CASES
Blonski, M., Simon, L., Houillier, C., Idbaih, A., Wittwer, B., Beauchesne, P., Hoang-Xuan, K., Taillandier, L.
Published in Neuro-oncology (Charlottesville, Va.) (01.09.2014)
Published in Neuro-oncology (Charlottesville, Va.) (01.09.2014)
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Cerebral diffusion tensor imaging, awakening, consciousness recovery prognosis in comatose patients and physical and rehabilitation medicine: A case report
Wittwer, B, Fraser, A., Dr, Le Chapelain, L., Dr, Khalil, N., Dr, Planel, S., Dr, Beis, J.M., Dr, Paysant, J., Prof
Published in Annals of physical and rehabilitation medicine (01.09.2015)
Published in Annals of physical and rehabilitation medicine (01.09.2015)
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Genotypic and Phenotypic Spectrum in Tricho-Rhino-Phalangeal Syndrome Types I and III
Lüdecke, H.-J., Schaper, J., Meinecke, P., Momeni, P., Groß, S., von Holtum, D., Hirche, H., Abramowicz, M.J., Albrecht, B., Apacik, C., Christen, H.-J., Claussen, U., Devriendt, K., Fastnacht, E., Forderer, A., Friedrich, U., Goodship, T.H.J., Greiwe, M., Hamm, H., Hennekam, R.C.M., Hinkel, G.K., Hoeltzenbein, M., Kayserili, H., Majewski, F., Mathieu, M., McLeod, R., Midro, A.T., Moog, U., Nagai, T., Niikawa, N., Ørstavik, K.H., Plöchl, E., Seitz, C., Schmidtke, J., Tranebjærg, L., Tsukahara, M., Wittwer, B., Zabel, B., Gillessen-Kaesbach, G., Horsthemke, B.
Published in American journal of human genetics (01.01.2001)
Published in American journal of human genetics (01.01.2001)
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Conference Proceeding
Targeted protein degraders: a call for collective action to advance safety assessment
Jones, Lyn H., Mitchell, Constance A., Loberg, Lise, Pavkovic, Mira, Rao, Mohan, Roberts, Ruth, Stamp, Katie, Volak, Laurie, Wittwer, Matthias B., Pettit, Syril
Published in Nature reviews. Drug discovery (01.06.2022)
Published in Nature reviews. Drug discovery (01.06.2022)
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A gene (RPGR) with homology to the RCC1 guanine nucleotide exchange factor is mutated in X-linked retinitis pigmentosa (RP3)
Meindl, A, Dry, K, Herrmann, K, Manson, E, Ciccodicola, A, Edgar, A, Carvalho, M.R.S, Achatz, H, Hellebrand, H, Lennon, A, Migliaccio, C, Porter, K, Zrenner, E, Bird, A, Jay, M, Lorenz, B, Wittwer, B, D'Urso, M, Meitinger, T, Wright, A
Published in Nature genetics (01.05.1996)
Published in Nature genetics (01.05.1996)
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Identification of ( R )-[ 18 F]YH134 for Monoacylglycerol Lipase Neuroimaging and Exploration of Its Use for Central Nervous System and Peripheral Drug Development
He, Yingfang, Krämer, Stefanie D, Grether, Uwe, Wittwer, Matthias B, Collin, Ludovic, Kuhn, Bernd, Topp, Andreas, Heer, Dominik, O'Hara, Fionn, Honer, Michael, Pavlovic, Anto, Richter, Hans, Ritter, Martin, Rombach, Didier, Keller, Claudia, Gobbi, Luca, Mu, Linjing
Published in Journal of Nuclear Medicine (01.02.2024)
Published in Journal of Nuclear Medicine (01.02.2024)
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ITC Commentary on Metformin Clinical Drug-Drug Interaction Study Design That Enables an Efficacy- and Safety-Based Dose Adjustment Decision
Zamek-Gliszczynski, Maciej J, Chu, Xiaoyan, Cook, Jack A, Custodio, Joseph M, Galetin, Aleksandra, Giacomini, Kathleen M, Lee, Caroline A, Paine, Mary F, Ray, Adrian S, Ware, Joseph A, Wittwer, Matthias B, Zhang, Lei
Published in Clinical pharmacology and therapeutics (01.11.2018)
Published in Clinical pharmacology and therapeutics (01.11.2018)
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Involvement of CB 1 and CB 2 receptors in neuroprotective effects of cannabinoids in experimental TDP-43 related frontotemporal dementia using male mice
Gonzalo-Consuegra, Claudia, Santos-García, Irene, García-Toscano, Laura, Martín-Baquero, Raquel, Rodríguez-Cueto, Carmen, Wittwer, Matthias B, Dzygiel, Pawel, Grether, Uwe, de Lago, Eva, Fernández-Ruiz, Javier
Published in Biomedicine & pharmacotherapy (01.05.2024)
Published in Biomedicine & pharmacotherapy (01.05.2024)
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Multi-parameter optimization: Development of a morpholin-3-one derivative with an improved kinetic profile for imaging monoacylglycerol lipase in the brain
He, Yingfang, Grether, Uwe, Taddio, Marco F., Meier, Carla, Keller, Claudia, Edelmann, Martin R., Honer, Michael, Huber, Sylwia, Wittwer, Matthias B., Heer, Dominik, Richter, Hans, Collin, Ludovic, Hug, Melanie N., Hilbert, Manuel, Postmus, Annemarieke G.J., Stevens, Anna Floor, van der Stelt, Mario, Krämer, Stefanie D., Schibli, Roger, Mu, Linjing, Gobbi, Luca C.
Published in European journal of medicinal chemistry (05.12.2022)
Published in European journal of medicinal chemistry (05.12.2022)
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Discovery, synthesis and evaluation of novel reversible monoacylglycerol lipase radioligands bearing a morpholine-3-one scaffold
He, Yingfang, Gobbi, Luca C., Herde, Adrienne Müller, Rombach, Didier, Ritter, Martin, Kuhn, Bernd, Wittwer, Matthias B., Heer, Dominik, Hornsperger, Benoit, Bell, Charles, O'Hara, Fionn, Benz, Jörg, Honer, Michael, Keller, Claudia, Collin, Ludovic, Richter, Hans, Schibli, Roger, Grether, Uwe, Mu, Linjing
Published in Nuclear medicine and biology (01.05.2022)
Published in Nuclear medicine and biology (01.05.2022)
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