In Vitro Activities of MMV Malaria Box Compounds against the Apicomplexan Parasite Neospora caninum , the Causative Agent of Neosporosis in Animals
Müller, Joachim, Winzer, Pablo A, Samby, Kirandeep, Hemphill, Andrew
Published in Molecules (Basel, Switzerland) (24.03.2020)
Published in Molecules (Basel, Switzerland) (24.03.2020)
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Journal Article
Comparative assessment of the effects of bumped kinase inhibitors on early zebrafish embryo development and pregnancy in mice
Anghel, Nicoleta, Winzer, Pablo A., Imhof, Dennis, Müller, Joachim, Langa, Xavier, Rieder, Jessica, Barrett, Lynn K., Vidadala, Rama Subba Rao, Huang, Wenlin, Choi, Ryan, Hulverson, Mathew A., Whitman, Grant R., Arnold, Samuel L., Van Voorhis, Wesley C., Ojo, Kayode K., Maly, Dustin J., Fan, Erkang, Hemphill, Andrew
Published in International journal of antimicrobial agents (01.09.2020)
Published in International journal of antimicrobial agents (01.09.2020)
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Journal Article
In vitro activity, safety and in vivo efficacy of the novel bumped kinase inhibitor BKI-1748 in non-pregnant and pregnant mice experimentally infected with Neospora caninum tachyzoites and Toxoplasma gondii oocysts
Imhof, Dennis, Anghel, Nicoleta, Winzer, Pablo, Balmer, Vreni, Ramseier, Jessica, Hänggeli, Kai, Choi, Ryan, Hulverson, Matthew A., Whitman, Grant R., Arnold, Samuel L.M., Ojo, Kayode K., Van Voorhis, Wesley C., Doggett, J. Stone, Ortega-Mora, Luis M., Hemphill, Andrew
Published in International journal for parasitology -- drugs and drug resistance (01.08.2021)
Published in International journal for parasitology -- drugs and drug resistance (01.08.2021)
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Journal Article
Neospora caninum : Structure and Fate of Multinucleated Complexes Induced by the Bumped Kinase Inhibitor BKI-1294
Winzer, Pablo, Anghel, Nicoleta, Imhof, Dennis, Balmer, Vreni, Ortega-Mora, Luis-Miguel, Ojo, Kayode K, Van Voorhis, Wesley C, Müller, Joachim, Hemphill, Andrew
Published in Pathogens (Basel) (16.05.2020)
Published in Pathogens (Basel) (16.05.2020)
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Journal Article
Endochin-like quinolones (ELQs) and bumped kinase inhibitors (BKIs): Synergistic and additive effects of combined treatments against Neospora caninum infection in vitro and in vivo
Anghel, Nicoleta, Imhof, Dennis, Winzer, Pablo, Balmer, Vreni, Ramseier, Jessica, Haenggeli, Kai, Choi, Ryan, Hulverson, Matthew A., Whitman, Grant R., Arnold, Samuel L.M., Ojo, Kayode K., Van Voorhis, Wesley C., Doggett, J. Stone, Ortega-Mora, Luis M., Hemphill, Andrew
Published in International journal for parasitology -- drugs and drug resistance (01.12.2021)
Published in International journal for parasitology -- drugs and drug resistance (01.12.2021)
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Journal Article
Neospora caninum : Differential Proteome of Multinucleated Complexes Induced by the Bumped Kinase Inhibitor BKI-1294
Winzer, Pablo, Müller, Joachim, Imhof, Dennis, Ritler, Dominic, Uldry, Anne-Christine, Braga-Lagache, Sophie, Heller, Manfred, Ojo, Kayode K, Van Voorhis, Wesley C, Ortega-Mora, Luis-Miguel, Hemphill, Andrew
Published in Microorganisms (Basel) (26.05.2020)
Published in Microorganisms (Basel) (26.05.2020)
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Journal Article
The Impact of BKI-1294 Therapy in Mice Infected With the Apicomplexan Parasite Neospora caninum and Re-infected During Pregnancy
Winzer, Pablo, Imhof, Dennis, Anghel, Nicoleta, Ritler, Dominic, Müller, Joachim, Boubaker, Ghalia, Aguado-Martinez, Adriana, Ortega-Mora, Luis-Miguel, Ojo, Kayode K., VanVoorhis, Wesley C., Hemphill, Andrew
Published in Frontiers in veterinary science (15.10.2020)
Published in Frontiers in veterinary science (15.10.2020)
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Journal Article
Buparvaquone is active against Neospora caninum in vitro and in experimentally infected mice
Müller, Joachim, Aguado-Martinez, Adriana, Manser, Vera, Balmer, Vreni, Winzer, Pablo, Ritler, Dominic, Hostettler, Isabel, Arranz-Solís, David, Ortega-Mora, Luis, Hemphill, Andrew
Published in International journal for parasitology -- drugs and drug resistance (01.04.2015)
Published in International journal for parasitology -- drugs and drug resistance (01.04.2015)
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Journal Article
Endochin-Like Quinolones Exhibit Promising Efficacy Against Neospora Caninum in vitro and in Experimentally Infected Pregnant Mice
Anghel, Nicoleta, Balmer, Vreni, Müller, Joachim, Winzer, Pablo, Aguado-Martinez, Adriana, Roozbehani, Mona, Pou, Sovitj, Nilsen, Aaron, Riscoe, Michael, Doggett, J Stone, Hemphill, Andrew
Published in Frontiers in veterinary science (19.11.2018)
Published in Frontiers in veterinary science (19.11.2018)
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Journal Article
Neospora caninum calcium-dependent protein kinase 1 is an effective drug target for neosporosis therapy
Ojo, Kayode K, Reid, Molly C, Kallur Siddaramaiah, Latha, Müller, Joachim, Winzer, Pablo, Zhang, Zhongsheng, Keyloun, Katelyn R, Vidadala, Rama Subba Rao, Merritt, Ethan A, Hol, Wim G J, Maly, Dustin J, Fan, Erkang, Van Voorhis, Wesley C, Hemphill, Andrew
Published in PloS one (28.03.2014)
Published in PloS one (28.03.2014)
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Journal Article
In Vitro and In Vivo Effects of the Bumped Kinase Inhibitor 1294 in the Related Cyst-Forming Apicomplexans Toxoplasma gondii and Neospora caninum
Winzer, Pablo, Müller, Joachim, Aguado-Martínez, Adriana, Rahman, Mahbubur, Balmer, Vreni, Manser, Vera, Ortega-Mora, Luis Miguel, Ojo, Kayode K, Fan, Erkang, Maly, Dustin J, Van Voorhis, Wesley C, Hemphill, Andrew
Published in Antimicrobial agents and chemotherapy (01.10.2015)
Published in Antimicrobial agents and chemotherapy (01.10.2015)
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Journal Article
In vitro effects of new artemisinin derivatives in Neospora caninum -infected human fibroblasts
Müller, Joachim, Balmer, Vreni, Winzer, Pablo, Rahman, Mahbubur, Manser, Vera, Haynes, Richard K, Hemphill, Andrew
Published in International journal of antimicrobial agents (01.07.2015)
Published in International journal of antimicrobial agents (01.07.2015)
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Journal Article
One health therapeutics: Target-Based drug development for cryptosporidiosis and other apicomplexa diseases
Van Voorhis, Wesley C., Hulverson, Matthew A., Choi, Ryan, Huang, Wenlin, Arnold, Samuel L.M., Schaefer, Deborah A., Betzer, Dana P., Vidadala, Rama S.R., Lee, Sangun, Whitman, Grant R., Barrett, Lynn K., Maly, Dustin J., Riggs, Michael W., Fan, Erkang, Kennedy, Thomas J., Tzipori, Saul, Doggett, J. Stone, Winzer, Pablo, Anghel, Nicoleta, Imhof, Dennis, Müller, Joachim, Hemphill, Andrew, Ferre, Ignacio, Sanchez-Sanchez, Roberto, Ortega-Mora, Luis Miguel, Ojo, Kayode K.
Published in Veterinary parasitology (01.01.2021)
Published in Veterinary parasitology (01.01.2021)
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Journal Article
Neospora caninum Calcium-Dependent Protein Kinase 1 Is an Effective Drug Target for Neosporosis Therapy: e92929
Ojo, Kayode K, Reid, Molly C, Siddaramaiah, Latha Kallur, Mueller, Joachim, Winzer, Pablo, Zhang, Zhongsheng, Keyloun, Katelyn R, Vidadala, Rama SubbaRao, Merritt, Ethan A, Hol, Wim GJ
Published in PloS one (01.03.2014)
Published in PloS one (01.03.2014)
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Journal Article