Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase
Nocentini, Alessio, Angeli, Andrea, Carta, Fabrizio, Winum, Jean-Yves, Zalubovskis, Raivis, Carradori, Simone, Capasso, Clemente, Donald, William A., Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
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Journal Article
Multivalent Carbonic Anhydrases Inhibitors
Carta, Fabrizio, Dumy, Pascal, Supuran, Claudiu T, Winum, Jean-Yves
Published in International journal of molecular sciences (01.11.2019)
Published in International journal of molecular sciences (01.11.2019)
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Journal Article
Targeting Tumor Hypoxia: Suppression of Breast Tumor Growth and Metastasis by Novel Carbonic Anhydrase IX Inhibitors
YUANMEI LOU, MCDONALD, Paul C, CLARKE, Blaise, SUTHERLAND, Brent W, WATERHOUSE, Dawn, BALLY, Marcel, ROSKELLEY, Calvin, OVERALL, Christopher M, MINCHINTON, Andrew, PACCHIANO, Fabio, CARTA, Fabrizio, SCOZZAFAVA, Andrea, OLOUMI, Arusha, TOUISNI, Nadia, WINUM, Jean-Yves, SUPURAN, Claudiu T, DEDHAR, Shoukat, CHIA, Stephen, OSTLUND, Christina, AHMADI, Ardalan, KYLE, Alastair, AUF DEM KELLER, Ulrich, LEUNG, Samuel, HUNTSMAN, David
Published in Cancer research (Chicago, Ill.) (01.05.2011)
Published in Cancer research (Chicago, Ill.) (01.05.2011)
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Journal Article
Carbonic Anhydrase Inhibitors Featuring a Porphyrin Scaffold: Synthesis, Optical and Biological Properties
Merabti, Amina, Roger, Maxime, Nguyen, Christophe, Nocentini, Alessio, Gerbier, Philippe, Richeter, Sébastien, Gary‐Bobo, Magali, Supuran, Claudiu T., Clément, Sébastien, Winum, Jean‐Yves
Published in European journal of organic chemistry (07.06.2022)
Published in European journal of organic chemistry (07.06.2022)
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Journal Article
1,5‐Benzodiazepines as a platform for the design of carbonic anhydrase inhibitors
Ismail, Chiraz, Nocentini, Alessio, Supuran, Claudiu T., Winum, Jean‐Yves, Gharbi, Rafik
Published in Archiv der Pharmazie (Weinheim) (01.03.2022)
Published in Archiv der Pharmazie (Weinheim) (01.03.2022)
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Journal Article
Emerging trends in enzyme inhibition by multivalent nanoconstructs
Kanfar, Nasreddine, Bartolami, Eline, Zelli, Renaud, Marra, Alberto, Winum, Jean-Yves, Ulrich, Sébastien, Dumy, Pascal
Published in Organic & biomolecular chemistry (01.01.2015)
Published in Organic & biomolecular chemistry (01.01.2015)
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Journal Article
Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
Angeli, Andrea, Carta, Fabrizio, Nocentini, Alessio, Winum, Jean-Yves, Zalubovskis, Raivis, Akdemir, Atilla, Onnis, Valentina, Eldehna, Wagdy M., Capasso, Clemente, Simone, Giuseppina De, Monti, Simona Maria, Carradori, Simone, Donald, William A., Dedhar, Shoukat, Supuran, Claudiu T.
Published in Metabolites (14.10.2020)
Published in Metabolites (14.10.2020)
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Journal Article
Carbonic anhydrase IX: A new druggable target for the design of antitumor agents
Winum, Jean-Yves, Rami, Marouan, Scozzafava, Andrea, Montero, Jean-Louis, Supuran, Claudiu
Published in Medicinal research reviews (01.05.2008)
Published in Medicinal research reviews (01.05.2008)
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Journal Article
Carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani chagasi are inhibited by benzoxaboroles
Nocentini, Alessio, Cadoni, Roberta, Dumy, Pascal, Supuran, Claudiu T., Winum, Jean-Yves
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2018)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2018)
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Journal Article
Antimetastatic Effect of Sulfamate Carbonic Anhydrase IX Inhibitors in Breast Carcinoma Xenografts
Gieling, Roben G, Babur, Muhammad, Mamnani, Lupti, Burrows, Natalie, Telfer, Brian A, Carta, Fabrizio, Winum, Jean-Yves, Scozzafava, Andrea, Supuran, Claudiu T, Williams, Kaye J
Published in Journal of medicinal chemistry (14.06.2012)
Published in Journal of medicinal chemistry (14.06.2012)
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Journal Article
Carbonic Anhydrase Inhibitors as Novel Drugs against Mycobacterial β-Carbonic Anhydrases: An Update on In Vitro and In Vivo Studies
Aspatwar, Ashok, Winum, Jean-Yves, Carta, Fabrizio, Supuran, Claudiu T, Hammaren, Milka, Parikka, Mataleena, Parkkila, Seppo
Published in Molecules (Basel, Switzerland) (08.11.2018)
Published in Molecules (Basel, Switzerland) (08.11.2018)
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Journal Article
Inhibition of carbonic anhydrases by a substrate analog: benzyl carbamate directly coordinates the catalytic zinc ion mimicking bicarbonate binding
De Simone, Giuseppina, Angeli, Andrea, Bozdag, Murat, Supuran, Claudiu T, Winum, Jean-Yves, Monti, Simona Maria, Alterio, Vincenzo
Published in Chemical communications (Cambridge, England) (2018)
Published in Chemical communications (Cambridge, England) (2018)
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Journal Article
Therapeutic applications of glycosidic carbonic anhydrase inhibitors
Winum, Jean-Yves, Poulsen, Sally-Ann, Supuran, Claudiu T.
Published in Medicinal research reviews (01.05.2009)
Published in Medicinal research reviews (01.05.2009)
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Journal Article
Fluorescent Silica Nanoparticles with Multivalent Inhibitory Effects towards Carbonic Anhydrases
Touisni, Nadia, Kanfar, Nasreddine, Ulrich, Sébastien, Dumy, Pascal, Supuran, Claudiu T., Mehdi, Ahmad, Winum, Jean-Yves
Published in Chemistry : a European journal (13.07.2015)
Published in Chemistry : a European journal (13.07.2015)
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Journal Article
A Novel Inhibitor of Carbonic Anhydrases Prevents Hypoxia-Induced TNBC Cell Plasticity
Sarnella, Annachiara, D'Avino, Giuliana, Hill, Billy Samuel, Alterio, Vincenzo, Winum, Jean-Yves, Supuran, Claudiu T, De Simone, Giuseppina, Zannetti, Antonella
Published in International journal of molecular sciences (09.11.2020)
Published in International journal of molecular sciences (09.11.2020)
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Journal Article