A multiple in silico program approach for the prediction of mutagenicity from chemical structure
White, Anita C, Mueller, Richard A, Gallavan, Robert H, Aaron, Sid, Wilson, Alan G.E
Published in Mutation research (05.08.2003)
Published in Mutation research (05.08.2003)
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In vivo toxicology of excipients commonly employed in drug discovery in rats
Gopinathan, Suma, O’Neill, Emily, Rodriguez, Lawrence A., Champ, Rose, Phillips, Megan, Nouraldeen, Amr, Wendt, Mary, Wilson, Alan G.E., Kramer, Jeffrey A.
Published in Journal of pharmacological and toxicological methods (01.09.2013)
Published in Journal of pharmacological and toxicological methods (01.09.2013)
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Evaluation of a basic physiologically based pharmacokinetic model for simulating the first-time-in-animal study
Germani, Massimiliano, Crivori, Patrizia, Rocchetti, Maurizio, Burton, Philip S., Wilson, Alan G.E., Smith, Mark E., Poggesi, Italo
Published in European journal of pharmaceutical sciences (01.07.2007)
Published in European journal of pharmaceutical sciences (01.07.2007)
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Mechanism of Thiazopyr-Induced Effects on Thyroid Hormone Homeostasis in Male Sprague–Dawley Rats
Hotz, Kathy J., Wilson, Alan G.E., Thake, Daryl C., Roloff, Marston V., Capen, Charles C., Kronenberg, Joel M., Brewster, David W.
Published in Toxicology and applied pharmacology (01.01.1997)
Published in Toxicology and applied pharmacology (01.01.1997)
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Discovery of LX2761, a Sodium-Dependent Glucose Cotransporter 1 (SGLT1) Inhibitor Restricted to the Intestinal Lumen, for the Treatment of Diabetes
Goodwin, Nicole C, Ding, Zhi-Ming, Harrison, Bryce A, Strobel, Eric D, Harris, Angela L, Smith, Melinda, Thompson, Andrea Y, Xiong, Wendy, Mseeh, Faika, Bruce, Debra J, Diaz, Damaris, Gopinathan, Suma, Li, Ling, O’Neill, Emily, Thiel, Mary, Wilson, Alan G. E, Carson, Kenneth G, Powell, David R, Rawlins, David B
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Stimulation of cortical bone formation with thienopyrimidine based inhibitors of Notum Pectinacetylesterase
Tarver, James E., Pabba, Praveen K., Barbosa, Joseph, Han, Qiang, Gardyan, Michael W., Brommage, Robert, Thompson, Andrea Y., Schmidt, James M., Wilson, Alan G.E., He, Wei, Lombardo, Victoria K., Carson, Kenneth G.
Published in Bioorganic & medicinal chemistry letters (15.03.2016)
Published in Bioorganic & medicinal chemistry letters (15.03.2016)
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Iris small break loca phenomena identification and ranking table (PIRT)
Larson, T.K., Moody, F.J., Wilson, G.E., Brown, W.L., Frepoli, C., Hartz, J., Woods, B.G., Oriani, L.
Published in Nuclear engineering and design (01.03.2007)
Published in Nuclear engineering and design (01.03.2007)
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4H-Thieno[3,2-c]chromene based inhibitors of Notum Pectinacetylesterase
Han, Qiang, Pabba, Praveen K., Barbosa, Joseph, Mabon, Ross, Healy, Jason P., Gardyan, Michael W., Terranova, Kristen M., Brommage, Robert, Thompson, Andrea Y., Schmidt, James M., Wilson, Alan G.E., Xu, Xiaolian, Tarver, James E., Carson, Kenneth G.
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
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Novel l-Xylose Derivatives as Selective Sodium-Dependent Glucose Cotransporter 2 (SGLT2) Inhibitors for the Treatment of Type 2 Diabetes
Goodwin, Nicole C, Mabon, Ross, Harrison, Bryce A, Shadoan, Melanie K, Almstead, Zheng Y, Xie, Yiling, Healy, Jason, Buhring, Lindsey M, DaCosta, Christopher M, Bardenhagen, Jennifer, Mseeh, Faika, Liu, Qingyun, Nouraldeen, Amr, Wilson, Alan G. E, Kimball, S. David, Powell, David R, Rawlins, David B
Published in Journal of medicinal chemistry (22.10.2009)
Published in Journal of medicinal chemistry (22.10.2009)
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Discovery and Development of LX7101, a Dual LIM-Kinase and ROCK Inhibitor for the Treatment of Glaucoma
Harrison, Bryce A, Almstead, Zheng Y, Burgoon, Hugh, Gardyan, Michael, Goodwin, Nicole C, Healy, Jason, Liu, Ying, Mabon, Ross, Marinelli, Brett, Samala, Lakshman, Zhang, Yulian, Stouch, Terry R, Whitlock, N. Andrew, Gopinathan, Suma, McKnight, Beth, Wang, Shuli, Patel, Nita, Wilson, Alan G. E, Hamman, Brian D, Rice, Dennis S, Rawlins, David B
Published in ACS medicinal chemistry letters (08.01.2015)
Published in ACS medicinal chemistry letters (08.01.2015)
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Influence of Molecular Flexibility and Polar Surface Area Metrics on Oral Bioavailability in the Rat
Lu, Jing J, Crimin, Kimberly, Goodwin, Jay T, Crivori, Patrizia, Orrenius, Christian, Xing, Li, Tandler, Peter J, Vidmar, Thomas J, Amore, Benny M, Wilson, Alan G. E, Stouten, Pieter F. W, Burton, Philip S
Published in Journal of medicinal chemistry (18.11.2004)
Published in Journal of medicinal chemistry (18.11.2004)
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Novel Class of LIM-Kinase 2 Inhibitors for the Treatment of Ocular Hypertension and Associated Glaucoma
Harrison, Bryce A, Whitlock, N. Andrew, Voronkov, Michael V, Almstead, Zheng Y, Gu, Kun-jian, Mabon, Ross, Gardyan, Michael, Hamman, Brian D, Allen, Jason, Gopinathan, Suma, McKnight, Beth, Crist, Mike, Zhang, Yulian, Liu, Ying, Courtney, Lawrence F, Key, Billie, Zhou, Julia, Patel, Nita, Yates, Phil W, Liu, Qingyun, Wilson, Alan G. E, Kimball, S. David, Crosson, Craig E, Rice, Dennis S, Rawlins, David B
Published in Journal of medicinal chemistry (12.11.2009)
Published in Journal of medicinal chemistry (12.11.2009)
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Pharmacokinetic/pharmacodynamic modelling of 2-acetyl-4(5)-tetrahydroxybutyl imidazole-induced peripheral lymphocyte sequestration through increasing lymphoid sphingosine 1-phosphate
Yu, X. Q., Kramer, J., Moran, L., O'Neill, E., Nouraldeen, A., Oravecz, T., Wilson, A. G. E.
Published in Xenobiotica (01.05.2010)
Published in Xenobiotica (01.05.2010)
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