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Hsieh, Gin C, Pai, Madhavi, Chandran, Prasant, Hooker, Bradley A, Zhu, Chang Z, Salyers, Anita K, Wensink, Erica J, Zhan, CenChen, Carroll, William A, Dart, Michael J, Yao, Betty B, Honore, Prisca, Meyer, Michael D
Published in British journal of pharmacology (01.01.2011)
Published in British journal of pharmacology (01.01.2011)
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[3H]A-804598 ([3H]2-cyano-1-[(1S)-1-phenylethyl]-3-quinolin-5-ylguanidine) is a novel, potent, and selective antagonist radioligand for P2X7 receptors
Donnelly-Roberts, Diana L., Namovic, Marian T., Surber, Bruce, Vaidyanathan, Srirajan X., Perez-Medrano, Arturo, Wang, Ying, Carroll, William A., Jarvis, Michael F.
Published in Neuropharmacology (01.01.2009)
Published in Neuropharmacology (01.01.2009)
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Selective P2X7 receptor antagonists for chronic inflammation and pain
Carroll, William A., Donnelly-Roberts, Diana, Jarvis, Michael F.
Published in Purinergic signalling (2009)
Published in Purinergic signalling (2009)
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Effects of Substitution on 9-(3-Bromo-4-fluorophenyl)-5,9-dihydro-3H,4H-2,6-dioxa-4- azacyclopenta[b]naphthalene-1,8-dione, a Dihydropyridine ATP-Sensitive Potassium Channel Opener
Altenbach, Robert J, Brune, Michael E, Buckner, Steven A, Coghlan, Michael J, Daza, Anthony V, Fabiyi, Adebola, Gopalakrishnan, Murali, Henry, Rodger F, Khilevich, Albert, Kort, Michael E, Milicic, Ivan, Scott, Victoria E, Smith, Jamie C, Whiteaker, Kristi L, Carroll, William A
Published in Journal of medicinal chemistry (16.11.2006)
Published in Journal of medicinal chemistry (16.11.2006)
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Central and peripheral sites of action for CB 2 receptor mediated analgesic activity in chronic inflammatory and neuropathic pain models in rats
Hsieh, Gin C, Pai, Madhavi, Chandran, Prasant, Hooker, Bradley A, Zhu, Chang Z, Salyers, Anita K, Wensink, Erica J, Zhan, CenChen, Carroll, William A, Dart, Michael J, Yao, Betty B, Honore, Prisca, Meyer, Michael D
Published in British journal of pharmacology (01.01.2011)
Published in British journal of pharmacology (01.01.2011)
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Selective P2X(7) receptor antagonists for chronic inflammation and pain
Carroll, William A, Donnelly-Roberts, Diana, Jarvis, Michael F
Published in Purinergic signalling (01.03.2009)
Published in Purinergic signalling (01.03.2009)
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Structure−Activity Relationship Studies on a Series of Novel, Substituted 1-Benzyl-5-phenyltetrazole P2X7 Antagonists
Nelson, Derek W, Gregg, Robert J, Kort, Michael E, Perez-Medrano, Arturo, Voight, Eric A, Wang, Ying, Grayson, George, Namovic, Marian T, Donnelly-Roberts, Diana L, Niforatos, Wende, Honore, Prisca, Jarvis, Michael F, Faltynek, Connie R, Carroll, William A
Published in Journal of medicinal chemistry (15.06.2006)
Published in Journal of medicinal chemistry (15.06.2006)
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(â)-(9S)-9-(3-Bromo-4-fluorophenyl)-2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-Dioxide (A-278637): A Novel ATP-Sensitive Potassium Channel Opener Efficacious in Suppressing Urinary Bladder Contractions. II. In Vivo Characterization
Brune, Michael E, Fey, Thomas A, Brioni, Jorge D, Sullivan, James P, Williams, Michael, Carroll, William A, Coghlan, Michael J, Gopalakrishnan, Murali
Published in The Journal of pharmacology and experimental therapeutics (01.10.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2002)
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(â)-(9S)-9-(3-Bromo-4-fluorophenyl)-2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-Dioxide (A-278637): A Novel ATP-Sensitive Potassium Channel Opener Efficacious in Suppressing Urinary Bladder Contractions. I. In Vitro Characterization
Gopalakrishnan, Murali, Buckner, Steven A, Whiteaker, Kristi L, Shieh, Char-Chang, Molinari, Eduardo J, Milicic, Ivan, Daza, Anthony V, Davis-Taber, Rachel, Scott, Victoria E, Sellers, Donna, Chess-Williams, Russ, Chapple, Christopher R, Liu, Yi, Liu, Dong, Brioni, Jorge D, Sullivan, James P, Williams, Michael, Carroll, William A, Coghlan, Michael J
Published in The Journal of pharmacology and experimental therapeutics (01.10.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2002)
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[125I]A-312110, a Novel High-Affinity 1,4-Dihydropyridine ATP-sensitive K+ Channel Opener: Characterization and Pharmacology of Binding
Davis-Taber, Rachel, Molinari, Eduardo J, Altenbach, Robert J, Whiteaker, Kristi L, Shieh, Char-Chang, Rotert, Gary, Buckner, Steven A, Malysz, John, Milicic, Ivan, McDermott, Jeffrey S, Gintant, Gary A, Coghlan, Michael J, Carroll, William A, Scott, Victoria E, Gopalakrishnan, Murali
Published in Molecular pharmacology (01.07.2003)
Published in Molecular pharmacology (01.07.2003)
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The discovery of a new class of large-conductance Ca2+-activated K+ channel opener targeted for overactive bladder: Synthesis and structure-activity relationships of 2-amino-4-azaindoles
TURNER, Sean C, CARROLL, William A, SULLIVAN, James P, WHITE, Tammie K, GOPALAKRISHNAN, Murali, COGHLAN, Michael J, SHIEH, Char-Chang, ZHANG, Xu-Feng, PARIHAR, Ashutosh S, BUCKNER, Steven A, MILICIC, Ivan
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
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Discovery and Biological Evaluation of Novel Cyanoguanidine P2X(7) Antagonists with Analgesic Activity in a Rat Model of Neuropathic Pain
Perez-Medrano, Arturo, Donnelly-Roberts, Diana L., Honore, Prisca, Hsieh, Gin C., Namovic, Marian T., Peddi, Sridhar, Shuai, Qi, Wang, Ying, Faltynek, Connie R., Jarvis, Michael F., Carroll, William A.
Published in Journal of medicinal chemistry (28.05.2009)
Published in Journal of medicinal chemistry (28.05.2009)
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World Brain Day 2020: Move together to end Parkinson's disease
Wijeratne, Tissa, Grisold, Wolfgang, Trenkwalder, Claudia, Carroll, A.M. William
Published in Journal of the neurological sciences (15.09.2020)
Published in Journal of the neurological sciences (15.09.2020)
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Two novel and potent 3-[(o-methoxyphenyl)piperazinylethyl]-5-phenylthieno[2,3-d]pyrimidine-2,4-diones selective for the α1D receptor
CARROLL, William A, SIPPY, Kevin B, ESBENSHADE, Timothy A, BUCKNER, Steven A, HANCOCK, Arthur A, MEYER, Michael D
Published in Bioorganic & medicinal chemistry letters (01.05.2001)
Published in Bioorganic & medicinal chemistry letters (01.05.2001)
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Discovery and Biological Evaluation of Novel Cyanoguanidine P2X7 Antagonists with Analgesic Activity in a Rat Model of Neuropathic Pain
Perez-Medrano, Arturo, Donnelly-Roberts, Diana L, Honore, Prisca, Hsieh, Gin C, Namovic, Marian T, Peddi, Sridhar, Shuai, Qi, Wang, Ying, Faltynek, Connie R, Jarvis, Michael F, Carroll, William A
Published in Journal of medicinal chemistry (28.05.2009)
Published in Journal of medicinal chemistry (28.05.2009)
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Structure−Activity Relationship Studies on N′-Aryl Carbohydrazide P2X7 Antagonists
Nelson, Derek W, Sarris, Kathy, Kalvin, Douglas M, Namovic, Marian T, Grayson, George, Donnelly-Roberts, Diana L, Harris, Richard, Honore, Prisca, Jarvis, Michael F, Faltynek, Connie R, Carroll, William A
Published in Journal of medicinal chemistry (22.05.2008)
Published in Journal of medicinal chemistry (22.05.2008)
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Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1H-tetrazol-5-amine P2X(7) antagonists
Perez-Medrano, Arturo, Donnelly-Roberts, Diana L, Florjancic, Alan S, Nelson, Derek W, Li, Tongmei, Namovic, Marian T, Peddi, Sridhar, Faltynek, Connie R, Jarvis, Michael F, Carroll, William A
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
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Synthesis and evaluation of 2-amido-3-carboxamide thiophene CB2 receptor agonists for pain management
Nelson, Derek W., Frost, Jennifer M., Tietje, Karin R., Florjancic, Alan S., Ryther, Keith, Carroll, William A., Dart, Michael J., Daza, Anthony V., Hooker, Bradley A., Grayson, George K., Fan, Yihong, Garrison, Tiffany R., El-Kouhen, Odile F., Yao, Betty, Pai, Madhavi, Chandran, Prasant, Zhu, Chang, Hsieh, Gin C., Meyer, Michael D.
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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