Inhibition of the spindle assembly checkpoint kinase TTK enhances the efficacy of docetaxel in a triple-negative breast cancer model
Maia, A.R.R., de Man, J., Boon, U., Janssen, A., Song, J.-Y., Omerzu, M., Sterrenburg, J.G., Prinsen, M.B.W., Willemsen-Seegers, N., de Roos, J.A.D.M., van Doornmalen, A.M., Uitdehaag, J.C.M., Kops, G.J.P.L., Jonkers, J., Buijsman, R.C., Zaman, G.J.R., Medema, R.H.
Published in Annals of oncology (01.10.2015)
Published in Annals of oncology (01.10.2015)
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Compound selectivity and target residence time of kinase inhibitors studied with surface plasmon resonance
Willemsen-Seegers, N, Uitdehaag, J, Prinsen, M, De Vetter, J, De Man, J, Sawa, M, Kawase, Y, Buijsman, R, Zaman, G
Published in European journal of cancer (1990) (01.12.2016)
Published in European journal of cancer (1990) (01.12.2016)
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Journal Article
The unique binding mode of NTRC 0066-0, a novel inhibitor of the spindle assembly checkpoint kinase TTK (Mps1), leads to long target residence time and potent anti-tumor activity
Zaman, G, Uitdehaag, J, De Man, J, Willemsen-Seegers, N, Sterrenburg, J.G, De Wit, J, De Roos, J, Prinsen, M, Buijsman, R
Published in European journal of cancer (1990) (01.07.2016)
Published in European journal of cancer (1990) (01.07.2016)
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Cell panel profiling of pre-clinical and clinical anti-cancer agents reveals conserved therapeutic clusters and differentiates the mechanism of action of different PI3K/mTOR, Aurora kinase and EZH2 inhibitors
Uitdehaag, J.C.M, De Roos, J.A.D.M, Prinsen, M.B.W, Willemsen-Seegers, N, De Vetter, J.R.F, Dylus, J, Van Doornmalen, A.M, Kooijman, J, Sawa, M, Van Gerwen, S.J.C, De Man, J, Buijsman, R.C, Zaman, G.J.R
Published in European journal of cancer (1990) (01.12.2016)
Published in European journal of cancer (1990) (01.12.2016)
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30P Comparative biochemical and cellular profiling of kinase inhibitors approved for clinical use from 2018 to 2020
Kooijman, J., Van Riel, W., Prinsen, M., Dylus, J., Grobben, Y., De Roos, J., Melis, J., De Bitter, T., Narumi, Y., Kawase, Y., Willemsen-Seegers, N., Zaman, G.
Published in Annals of oncology (01.03.2022)
Published in Annals of oncology (01.03.2022)
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235 - Compound selectivity and target residence time of kinase inhibitors studied with surface plasmon resonance
Willemsen-Seegers, N., Uitdehaag, J., Prinsen, M., De Vetter, J., De Man, J., Sawa, M., Kawase, Y., Buijsman, R., Zaman, G.
Published in European journal of cancer (1990) (01.12.2016)
Published in European journal of cancer (1990) (01.12.2016)
Get full text
Journal Article
586 - The unique binding mode of NTRC 0066-0, a novel inhibitor of the spindle assembly checkpoint kinase TTK (Mps1), leads to long target residence time and potent anti-tumor activity
Zaman, G., Uitdehaag, J., De Man, J., Willemsen-Seegers, N., Sterrenburg, J.G., De Wit, J., De Roos, J., Prinsen, M., Buijsman, R.
Published in European journal of cancer (1990) (01.07.2016)
Published in European journal of cancer (1990) (01.07.2016)
Get full text
Journal Article
52 - Cell panel profiling of pre-clinical and clinical anti-cancer agents reveals conserved therapeutic clusters and differentiates the mechanism of action of different PI3K/mTOR, Aurora kinase and EZH2 inhibitors
Uitdehaag, J.C.M., De Roos, J.A.D.M., Prinsen, M.B.W., Willemsen-Seegers, N., De Vetter, J.R.F., Dylus, J., Van Doornmalen, A.M., Kooijman, J., Sawa, M., Van Gerwen, S.J.C., De Man, J., Buijsman, R.C., Zaman, G.J.R.
Published in European journal of cancer (1990) (01.12.2016)
Published in European journal of cancer (1990) (01.12.2016)
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Journal Article
Identification of selective inhibitors of the spindle assembly checkpoint kinase TTK (Mps1) for treatment of triple negative breast cancer
Zaman, G., de Man, J., Uitdehaag, J., Maia, A., Boon, U., Sterrenburg, J.-G., Prinsen, M., Willemsen-Seegers, N., Jonkers, J., Kops, G., Medema, R., Buijsman, R.
Published in Annals of oncology (01.03.2015)
Published in Annals of oncology (01.03.2015)
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