Warfarin-fluconazole. II. A metabolically based drug interaction: in vivo studies
Black, D J, Kunze, K L, Wienkers, L C, Gidal, B E, Seaton, T L, McDonnell, N D, Evans, J S, Bauwens, J E, Trager, W F
Published in Drug metabolism and disposition (01.04.1996)
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Published in Drug metabolism and disposition (01.04.1996)
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Bioactivation of the anticancer agent CPT-11 to SN-38 by human hepatic microsomal carboxylesterases and the in vitro assessment of potential drug interactions
SLATTER, J. G, SU, P, SAMS, J. P, SCHAAF, L. J, WIENKERS, L. C
Published in Drug metabolism and disposition (01.10.1997)
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Published in Drug metabolism and disposition (01.10.1997)
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Oxidation of the Novel Oxazolidinone Antibiotic Linezolid in Human Liver Microsomes
WYNALDA, M. A, HAUER, M. J, WIENKERS, L. C
Published in Drug metabolism and disposition (01.09.2000)
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Published in Drug metabolism and disposition (01.09.2000)
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Formation of (R)-8-hydroxywarfarin in human liver microsomes. A new metabolic marker for the (S)-mephenytoin hydroxylase, P4502C19
Wienkers, L C, Wurden, C J, Storch, E, Kunze, K L, Rettie, A E, Trager, W F
Published in Drug metabolism and disposition (01.05.1996)
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Published in Drug metabolism and disposition (01.05.1996)
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Characterization of bropirimine O-glucuronidation in human liver microsomes
Wynalda, M. A., Wynalda, K. M., Amore, B. M., Fagerness, P. E., Wienkers, L. C.
Published in Xenobiotica (01.10.2003)
Published in Xenobiotica (01.10.2003)
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Pharmacology of AMG 181, a human anti‐α4β7 antibody that specifically alters trafficking of gut‐homing T cells
Pan, WJ, Hsu, H, Rees, WA, Lear, SP, Lee, F, Foltz, IN, Rathanaswami, P, Manchulenko, K, Chan, BM, Zhang, M, Xia, XZ, Patel, SK, Prince, PJ, Doherty, DR, Sheckler, CM, Reynhardt, KO, Krill, CD, Harder, BJ, Wisler, JA, Brandvig, JL, Lynch, JL, Anderson, AA, Wienkers, LC, Borie, DC
Published in British journal of pharmacology (01.05.2013)
Published in British journal of pharmacology (01.05.2013)
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Biotransformation of tirilazad in human: 1. Cytochrome P450 3A-mediated hydroxylation of tirilazad mesylate in human liver microsomes
Wienkers, L C, Steenwyk, R C, Sanders, P E, Pearson, P G
Published in The Journal of pharmacology and experimental therapeutics (01.05.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.05.1996)
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Relationships between the levels of cytochrome P4502C9 and its prototypic catalytic activities in human liver microsomes
Hall, S D, Hamman, M A, Rettie, A E, Wienkers, L C, Trager, W F, Vandenbranden, M, Wrighton, S A
Published in Drug metabolism and disposition (01.11.1994)
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Published in Drug metabolism and disposition (01.11.1994)
Journal Article
Biotransformation of tirilazad in human: 2. Effect of ketoconazole on tirilazad clearance and oral bioavailability
Fleishaker, J C, Pearson, P G, Wienkers, L C, Pearson, L K, Peters, G R
Published in The Journal of pharmacology and experimental therapeutics (01.05.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.05.1996)
Journal Article
Hormonal effects on tirilazad clearance in women: assessment of the role of CYP3A
Fleishaker, J C, Pearson, L K, Pearson, P G, Wienkers, L C, Hopkins, N K, Peters, G R
Published in Journal of clinical pharmacology (01.03.1999)
Published in Journal of clinical pharmacology (01.03.1999)
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Covalent Alteration of the CYP3A4 Active Site: Evidence for Multiple Substrate Binding Domains
Schrag, Michael L., Wienkers, Larry C.
Published in Archives of biochemistry and biophysics (01.07.2001)
Published in Archives of biochemistry and biophysics (01.07.2001)
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Mechanism-Based Inactivation of Cytochrome P450 2D6 by 1-[(2-Ethyl-4-methyl-1H-imidazol-5-yl)methyl]- 4-[4-(trifluoromethyl)-2-pyridinyl]piperazine: Kinetic Characterization and Evidence for Apoprotein Adduction
Hutzler, J. Matthew, Steenwyk, Rick C, Smith, Evan B, Walker, Gregory S, Wienkers, Larry C
Published in Chemical research in toxicology (01.02.2004)
Published in Chemical research in toxicology (01.02.2004)
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