Inhibition of prenylated KRAS in a lipid environment
Jansen, Johanna M, Wartchow, Charles, Jahnke, Wolfgang, Fong, Susan, Tsang, Tiffany, Pfister, Keith, Zavorotinskaya, Tatiana, Bussiere, Dirksen, Cheng, Jan Marie, Crawford, Kenneth, Dai, Yumin, Dove, Jeffrey, Fang, Eric, Feng, Yun, Florent, Jean-Michel, Fuller, John, Gossert, Alvar D, Hekmat-Nejad, Mohammad, Henry, Chrystèle, Klopp, Julia, Lenahan, William P, Lingel, Andreas, Ma, Sylvia, Meyer, Arndt, Mishina, Yuji, Narberes, Jamie, Pardee, Gwynn, Ramurthy, Savithri, Rieffel, Sebastien, Stuart, Darrin, Subramanian, Sharadha, Tandeske, Laura, Widger, Stephania, Widmer, Armin, Winterhalter, Aurelie, Zaror, Isabel, Hardy, Stephen
Published in PloS one (06.04.2017)
Published in PloS one (06.04.2017)
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Terminal Adenosyl Transferase Activity of Posttranscriptional Regulator HuR Revealed by Confocal On-Bead Screening
Meisner, Nicole-Claudia, Hintersteiner, Martin, Seifert, Jan-Marcus, Bauer, Roman, Benoit, Roger Marc, Widmer, Armin, Schindler, Torsten, Uhl, Volker, Lang, Michaela, Gstach, Hubert, Auer, Manfred
Published in Journal of molecular biology (20.02.2009)
Published in Journal of molecular biology (20.02.2009)
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Discovery of Novel Allosteric Non-Bisphosphonate Inhibitors of Farnesyl Pyrophosphate Synthase by Integrated Lead Finding
Marzinzik, Andreas L., Amstutz, René, Bold, Guido, Bourgier, Emmanuelle, Cotesta, Simona, Glickman, J. Fraser, Götte, Marjo, Henry, Christelle, Lehmann, Sylvie, Hartwieg, J. Constanze D., Ofner, Silvio, Pellé, Xavier, Roddy, Thomas P., Rondeau, Jean-Michel, Stauffer, Frédéric, Stout, Steven J., Widmer, Armin, Zimmermann, Johann, Zoller, Thomas, Jahnke, Wolfgang
Published in ChemMedChem (01.11.2015)
Published in ChemMedChem (01.11.2015)
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Abstract B38: Inhibiting mutated KRAS, a broken switch of effector pathways
Jansen, Johanna, Jahnke, Wolfgang, Fong, Susan, Tandeske, Laura, Wartchow, Charles, Pfister, Keith, Zavorotinskaya, Tatiana, Blechschmidt, Anke, Bussiere, Dirksen, Dai, Yumin, Dove, Jeff, Fang, Eric, Farley, David, Florent, Jean-Michel, Fuller, John, Gokhin, Simona, Gossert, Alvar, Hekmat-Nejad, Mohammad, Henry, Chrystèle, Klopp, Julia, Lenahan, Bill, Lingel, Andreas, Meyer, Arndt, Narberes, Jamie, Pardee, Gwynn, Paris, C Gregory, Ramurthy, Savithri, Renhowe, Paul, Rieffel, Sebastien, Shoemaker, Kevin, Subramanian, Sharadha, Tsang, Tiffany, Widger, Stephania, Widmer, Armin, Zaror, Isabel, Hardy, Stephen
Published in Molecular cancer research (01.12.2014)
Published in Molecular cancer research (01.12.2014)
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Use of organic solvents and small molecules for locating binding sites on proteins in solution
Dalvit, Claudio, Floersheim, Philipp, Zurini, Mauro, Widmer, Armin
Published in Journal of biomolecular NMR (01.05.1999)
Published in Journal of biomolecular NMR (01.05.1999)
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Non-peptide itam mimics as ZAP-70 antagonists
Revesz, Laszlo, Blum, Ernst, Manning, Ute, Demange, B.Jachez, Widmer, Armin, Zuber, Jean-François
Published in Bioorganic & medicinal chemistry letters (18.11.1997)
Published in Bioorganic & medicinal chemistry letters (18.11.1997)
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Structure-activity relationships in the trans-hexahydroindolo[4,3-ab]phenanthridine ("benzergoline") series. 2. Resolution, absolute configuration, and dopaminergic activity of the selective D1 agonist CY 208-243 and its implication for an "extended rotamer-based dopamine receptor model"
Seiler, Max P, Floersheim, Philipp, Markstein, Rudolf, Widmer, Armin
Published in Journal of medicinal chemistry (01.04.1993)
Published in Journal of medicinal chemistry (01.04.1993)
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Journal Article
GEOM: a new tool for molecular modelling based on distance geometry calculations with NMR data
Sanner, M, Widmer, A, Senn, H, Braun, W
Published in Journal of computer-aided molecular design (01.09.1989)
Published in Journal of computer-aided molecular design (01.09.1989)
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