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Published in Journal of medicinal chemistry (24.03.2005)
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Design, Synthesis, and Biological Characterization of a Peptide-Mimetic Antagonist for a Tethered-Ligand Receptor
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Published in Proceedings of the National Academy of Sciences - PNAS (26.10.1999)
Published in Proceedings of the National Academy of Sciences - PNAS (26.10.1999)
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Macrocyclic bisindolylmaleimides as inhibitors of protein kinase C and glycogen synthase kinase-3
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Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Efficient synthesis of 3-substituted 2-arylindoles via Suzuki coupling reactions on the solid phase
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Published in Tetrahedron letters (16.07.2001)
Published in Tetrahedron letters (16.07.2001)
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Discovery and Optimization of a Novel Series of Thrombin Receptor (PAR-1) Antagonists: Potent, Selective Peptide Mimetics Based on Indole and Indazole Templates
Zhang, Han-Cheng, Derian, Claudia K, Andrade-Gordon, Patricia, Hoekstra, William J, McComsey, David F, White, Kimberly B, Poulter, Brenda L, Addo, Michael F, Cheung, Wai-Man, Damiano, Bruce P, Oksenberg, Donna, Reynolds, Elwood E, Pandey, Anjali, Scarborough, Robert M, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (29.03.2001)
Published in Journal of medicinal chemistry (29.03.2001)
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High-affinity thrombin receptor (PAR-1) ligands: a new generation of indole-based peptide mimetic antagonists with a basic amine at the C-terminus
Zhang, Han-Cheng, White, Kimberly B., McComsey, David F., Addo, Michael F., Andrade-Gordon, Patricia, Derian, Claudia K., Oksenberg, Donna, Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
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Thrombin receptor (PAR-1) antagonists. Solid-Phase synthesis of indole-Based peptide mimetics by anchoring to a secondary amide
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Published in Bioorganic & medicinal chemistry letters (20.08.2001)
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Novel indolylindazolylmaleimides as inhibitors of protein kinase C- : Synthesis, biological activity, and cardiovascular safety
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Published in Journal of medicinal chemistry (2005)
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Published in Journal of medicinal chemistry (2005)
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Macrocyclic bisindolylmaleimides as inhibitors of protein kinase C and glycogen synthase kinase-3: Recent advances in the design of kinase inhibitors as novel therapeutic agents
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Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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Substituted benzothiazole and benzoxazole derivatives useful as inhibitors of dpp-1
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Year of Publication 29.04.2015
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Benzimidazolone peptidomimetics as thrombin receptor antagonists
Zhang, Han-Cheng, Maryanoff, Bruce E, McComsey, David F, White, Kimberly B
Year of Publication 13.09.2005
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Year of Publication 13.09.2005
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Benzimidazolone peptidometics as thrombin receptor antagonist
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Year of Publication 07.10.2003
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Year of Publication 07.10.2003
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