Novel 2-methoxyacylhydrazones as potent, selective PDE10A inhibitors with activity in animal models of schizophrenia
Cutshall, Neil S., Onrust, Rene, Rohde, Alex, Gragerov, Sasha, Hamilton, Lauren, Harbol, Kevin, Shen, Hui-Rong, McKee, Shawn, Zuta, Charles, Gragerova, Galina, Florio, Vince, Wheeler, Thomas N., Gage, Jennifer L.
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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6-Azasteroids: Structure-Activity Relationships for Inhibition of Type 1 and 2 Human 5.alpha.-Reductase and Human Adrenal 3.beta.-Hydroxy-.DELTA.5-steroid Dehydrogenase/3-Keto-.DELTA.5-steroid Isomerase
Frye, Stephen V, Haffner, Curt D, Maloney, Patrick R, Mook, Robert A, Dorsey, George F, Hiner, Roger N, Cribbs, Cindy M, Wheeler, Thomas N, Ray, John A
Published in Journal of medicinal chemistry (01.07.1994)
Published in Journal of medicinal chemistry (01.07.1994)
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Synthesis and biological activity of pyrethroids derived from halo-4-alkenoic acids
Ayad, Hafez M, Wheeler, Thomas N
Published in Journal of agricultural and food chemistry (01.01.1984)
Published in Journal of agricultural and food chemistry (01.01.1984)
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Journal Article
D-Nor steroids. IV. Carbonium ion rearrangements of conformationally defined cyclobutanes
Meinwald, Jerrold, Wheeler, Thomas N
Published in Journal of the American Chemical Society (01.02.1970)
Published in Journal of the American Chemical Society (01.02.1970)
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Journal Article
Synthesis of spiro[4.6]undecane-1,6-dione
Wheeler, Thomas N, Jackson, Clifford A, Young, Kirk H
Published in Journal of organic chemistry (01.05.1974)
Published in Journal of organic chemistry (01.05.1974)
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Journal Article
Substrate Specificity in Short-Chain Phospholipid Analogs at the Active Site of Human Synovial Phospholipase A2
Wheeler, T. N, Blanchard, Steven G, Fang, Frank, Gray-Nunez, Yolanda, Harris, Cole O, Lambert, Millard H, Mehrotra, Mukund M, Parks, Derek J, Andrew, R. C
Published in Journal of medicinal chemistry (01.11.1994)
Published in Journal of medicinal chemistry (01.11.1994)
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