Dual A1/A2B Receptor Blockade Improves Cardiac and Renal Outcomes in a Rat Model of Heart Failure with Preserved Ejection Fraction
Tofovic, Stevan P, Salah, Eman M, Smits, Glenn J, Whalley, Eric T, Ticho, Barry, Deykin, Aaron, Jackson, Edwin K
Published in The Journal of pharmacology and experimental therapeutics (01.02.2016)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2016)
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Discovery and therapeutic potential of kinin receptor antagonists
Whalley, Eric T, Figueroa, Carlos D, Gera, Lajos, Bhoola, Kanti D
Published in Expert opinion on drug discovery (01.12.2012)
Published in Expert opinion on drug discovery (01.12.2012)
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Synthesis of alkyne derivatives of a novel triazolopyrazine as A2A adenosine receptor antagonists
YAO, Gang, HAQUE, Serajul, PETTER, Russell C, LI SHA, KUMARAVEL, Gnanasambandam, WANG, Joy, ENGBER, Thomas M, WHALLEY, Eric T, CONLON, Patrick R, HEXI CHANG, KIESMAN, William F
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
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Novel Bicyclic Piperazine Derivatives of Triazolotriazine and Triazolopyrimidines as Highly Potent and Selective Adenosine A2A Receptor Antagonists
PENG, Hairuo, KUMARAVEL, Gnanasambandam, YAO, Gang, SHA, Li, WANG, Joy, VAN VLIJMEN, Herman, BOHNERT, Tonika, HUANG, Carol, VU, Chi B., ENSINGER, Carol L., CHANG, Hexi, ENGBER, Thomas M., WHALLEY, Eric T., PETTER, Russell C.
Published in Journal of medicinal chemistry (02.12.2004)
Published in Journal of medicinal chemistry (02.12.2004)
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Journal Article
A new class of bradykinin antagonists: synthesis and in vitro activity of bissuccinimidoalkane peptide dimers
Cheronis, John C, Whalley, Eric T, Nguyen, Khe T, Eubanks, Shad R, Allen, Lisa G, Duggan, Matthew J, Loy, Sharon D, Bonham, Kathryn A, Blodgett, James K
Published in Journal of medicinal chemistry (01.05.1992)
Published in Journal of medicinal chemistry (01.05.1992)
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Bradykinin Receptor Antagonists Containing N-Substituted Amino Acids: In Vitro and in Vivo B2 and B1 Receptor Antagonist Activity
Goodfellow, Val S, Marathe, Manoj V, Kuhlman, Karen G, Fitzpatrick, Timothy D, Cuadrado, David, Hanson, Wendy, Zuzack, John S, Ross, Sherman E, Wieczorek, Maciej, Burkard, Michael, Whalley, Eric T
Published in Journal of medicinal chemistry (29.03.1996)
Published in Journal of medicinal chemistry (29.03.1996)
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Differential effects of treatment with a small-molecule VLA-4 antagonist before and after onset of relapsing EAE
Theien, Bradley E., Vanderlugt, Carol L., Nickerson-Nutter, Cheryl, Cornebise, Mark, Scott, Daniel M., Perper, Stuart J., Whalley, Eric T., Miller, Stephen D.
Published in Blood (15.12.2003)
Published in Blood (15.12.2003)
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Potent, long-acting, orally-active bradykinin antagonists for a wide range of applications
Stewart, John M, Gera, Lajos, Chan, Daniel C, Whalley, Eric T, Hanson, Wendy L, Zuzack, John S
Published in Immunopharmacology (01.06.1997)
Published in Immunopharmacology (01.06.1997)
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Potent, long-acting bradykinin antagonists for a wide range of applications
Stewart, J M, Gera, L, Chan, D C, Whalley, E T, Hanson, W L, Zuzack, J S
Published in Canadian journal of physiology and pharmacology (01.06.1997)
Published in Canadian journal of physiology and pharmacology (01.06.1997)
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Design, synthesis, and in vitro activity of bis(succinimido)hexane peptide heterodimers with combined B1 and B2 antagonist activity
Cheronis, John C, Whalley, Eric T, Allen, Lisa G, Loy, Sharon D, Elder, Megan W, Duggan, Matthew J, Gross, Kelly L, Blodgett, James K
Published in Journal of medicinal chemistry (01.02.1994)
Published in Journal of medicinal chemistry (01.02.1994)
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Journal Article
Synthesis of alkyne derivatives of a novel triazolopyrazine as A 2A adenosine receptor antagonists
Yao, Gang, Haque, Serajul, Sha, Li, Kumaravel, Gnanasambandam, Wang, Joy, Engber, Thomas M., Whalley, Eric T., Conlon, Patrick R., Chang, Hexi, Kiesman, William F., Petter, Russell C.
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
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Journal Article
Effect of combined B1 and B2 kinin receptor blockade in porcine endotoxin shock
Siebeck, Matthias, Spannagl, Erwin, Schorr, Markus, Stumpf, Bernhard, Fritz, Hans, Whalley, Eric T., Cheronis, John C.
Published in Immunopharmacology (01.06.1996)
Published in Immunopharmacology (01.06.1996)
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Tachyphylaxis of the B1 kinin receptor in porcine endotoxin shock
Eich-Rathfelder, Sabine, Whalley, Eric T, Fautz, Michael, Hohenbleicher, Felix, Fritz, Hans, Siebeck, Matthias
Published in Immunopharmacology (01.06.1997)
Published in Immunopharmacology (01.06.1997)
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Journal Article
Synthesis of alkyne derivatives of a novel triazolopyrazine as A(2A) adenosine receptor antagonists
Yao, Gang, Haque, Serajul, Sha, Li, Kumaravel, Gnanasambandam, Wang, Joy, Engber, Thomas M, Whalley, Eric T, Conlon, Patrick R, Chang, Hexi, Kiesman, William F, Petter, Russell C
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
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Dopamine receptors in human basilar arteries
Forster, C, Drew, G M, Hilditch, A, Whalley, E T
Published in European journal of pharmacology (18.02.1983)
Published in European journal of pharmacology (18.02.1983)
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Journal Article
Novel Bicyclic Piperazine Derivatives of Triazolotriazine and Triazolopyrimidines as Highly Potent and Selective Adenosine A 2 A Receptor Antagonists
Peng, Hairuo, Kumaravel, Gnanasambandam, Yao, Gang, Sha, Li, Wang, Joy, Van Vlijmen, Herman, Bohnert, Tonika, Huang, Carol, Vu, Chi B., Ensinger, Carol L., Chang, Hexi, Engber, Thomas M., Whalley, Eric T., Petter, Russell C.
Published in Journal of medicinal chemistry (01.12.2004)
Published in Journal of medicinal chemistry (01.12.2004)
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