Efficient method to prepare diethylphosphonacetamides
Scaravelli, Federico, Bacchi, Sergio, Massari, Luca, Curcuruto, Ornella, Westerduin, Pieter, Maton, William
Published in Tetrahedron letters (29.09.2010)
Published in Tetrahedron letters (29.09.2010)
Get full text
Journal Article
Cover Feature: Synthesis of 2‐Substituted 1,2,3‐Triazoles via an Intramolecular N–N Bond Formation (Eur. J. Org. Chem. 5/2020)
Chen, Cheng‐yi, Lu, Xiaowei, Holland, Mareike C., Lv, Shichang, Ji, Xuebao, Liu, Wei, Liu, Jie, Depre, Dominique, Westerduin, Pieter
Published in European journal of organic chemistry (07.02.2020)
Published in European journal of organic chemistry (07.02.2020)
Get full text
Journal Article
Synthesis of 2‐Substituted 1,2,3‐Triazoles via an Intramolecular N–N Bond Formation
Chen, Cheng‐yi, Lu, Xiaowei, Holland, Mareike C., Lv, Shichang, Ji, Xuebao, Liu, Wei, Liu, Jie, Depre, Dominique, Westerduin, Pieter
Published in European journal of organic chemistry (07.02.2020)
Published in European journal of organic chemistry (07.02.2020)
Get full text
Journal Article
Correction to “Development of a Control Strategy for a Defluorinated Analogue in the Manufacturing Process of Casopitant Mesylate”
Bravo, Fernando, Cimarosti, Zadeo, Tinazzi, Francesco, Castoldi, Damiano, Stonestreet, Paul, Galgano, Annalisa, Westerduin, Pieter
Published in Organic process research & development (15.09.2017)
Published in Organic process research & development (15.09.2017)
Get full text
Journal Article
오렉신 수용체 조절제로서의 (2H-1,2,3-트라이아졸-2-일)페닐 화합물을 제조하는 개선된 합성 방법
MATCHA KIRAN, MEDINA FLORIAN DAMIEN, WESTERDUIN PIETER, CHEN CHENG YI, DEPRE DOMINIQUE PAUL M
Year of Publication 07.04.2022
Get full text
Year of Publication 07.04.2022
Patent
Application of the QbD Principles in the Development of the Casopitant Mesylate Manufacturing Process. Process Research Studies for the Definition of the Control Strategy of some Drug Substance-CQAs for Stages 2a, 2b, and 2c
Cimarosti, Zadeo, Bravo, Fernando, Castoldi, Damiano, Tinazzi, Francesco, Provera, Stefano, Perboni, Alcide, Papini, Damiano, Westerduin, Pieter
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
Get full text
Journal Article
Efficient Methods for the Synthesis of Arylacetonitriles
Stazi, Federica, Maton, William, Castoldi, Damiano, Westerduin, Pieter, Curcuruto, Ornella, Bacchi, Sergio
Published in Synthesis (Stuttgart) (01.10.2010)
Published in Synthesis (Stuttgart) (01.10.2010)
Get more information
Journal Article
A Mechanistic Insight into a Simple C−N Bond Formation via SN2 Displacement: A Synergistic Kinetics and Design of Experiment Approach
Massari, Luca, Panelli, Laura, Hughes, Mark, Stazi, Federica, Maton, William, Westerduin, Pieter, Scaravelli, Federico, Bacchi, Sergio
Published in Organic process research & development (19.11.2010)
Published in Organic process research & development (19.11.2010)
Get full text
Journal Article
Development of Drug Substances as Mixture of Polymorphs: Studies to Control Form 3 in Casopitant Mesylate
Cimarosti, Zadeo, Castagnoli, Carlo, Rossetti, Marco, Scarati, Mirka, Day, Caroline, Johnson, Brendan, Westerduin, Pieter
Published in Organic process research & development (19.11.2010)
Published in Organic process research & development (19.11.2010)
Get full text
Journal Article
Development of an Efficient Large-Scale Synthesis for a 4 H -imidazo[5,1- c ][1,4]benzoxazine-3-carboxamide Derivative for Depression and Anxiety
Giubellina, Nicola, Stabile, Paolo, Laval, Gilles, Perboni, Alcide D., Cimarosti, Zadeo, Westerduin, Pieter, Cooke, Jason W. B.
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
Get full text
Journal Article
Development of a Control Strategy for a Defluorinated Analogue in the Manufacturing Process of Casopitant Mesylate
Bravo, Fernando, Cimarosti, Zadeo, Tinazzi, Francesco, Castoldi, Damiano, Stonestreet, Paul, Galgano, Annalisa, Westerduin, Pieter
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
Get full text
Journal Article
Application of the Quality by Design Principles for the Development of the Crystallization Process for a Piperazinyl-Quinoline and Definition of the Control Strategy for Form 1
Cimarosti, Zadeo, Rossi, Sara, Tramarin, Davide, Laval, Gilles, Stabile, Paolo, Giubellina, Nicola, Maton, William, Allieri, Brigida, Campi, Francesca, Cooke, Jason, Westerduin, Pieter
Published in Organic process research & development (19.10.2012)
Published in Organic process research & development (19.10.2012)
Get full text
Journal Article
Development of a Dynamic Kinetic Resolution for the Isolation of an Intermediate in the Synthesis of Casopitant Mesylate: Application of QbD Principles in the Definition of the Parameter Ranges, Issues in the Scale-Up and Mitigation Strategies
Bravo, Fernando, Cimarosti, Zadeo, Tinazzi, Francesco, Smith, Gillian E, Castoldi, Damiano, Provera, Stefano, Westerduin, Pieter
Published in Organic process research & development (17.09.2010)
Published in Organic process research & development (17.09.2010)
Get full text
Journal Article
Identification of a Manufacturing Route of Novel CRF-1 Antagonists Containing a 2,3-Dihydro-1 H -pyrrolo[2,3- b ]pyridine Moiety
Ribecai, Arianna, Bacchi, Sergio, Delpogetto, Monica, Guelfi, Simone, Manzo, Angelo Maria, Perboni, Alcide, Stabile, Paolo, Westerduin, Pieter, Hourdin, Marie, Rossi, Sara, Provera, Stefano, Turco, Lucilla
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
Get full text
Journal Article
Identification of a Manufacturing Route of Novel CRF-1 Antagonists Containing a 2,3-Dihydro-1H-pyrrolo[2,3-b]pyridine Moiety
Ribecai, Arianna, Bacchi, Sergio, Delpogetto, Monica, Guelfi, Simone, Manzo, Angelo Maria, Perboni, Alcide, Stabile, Paolo, Westerduin, Pieter, Hourdin, Marie, Rossi, Sara, Provera, Stefano, Turco, Lucilla
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
Get full text
Journal Article
Development of an Efficient Large-Scale Synthesis for a 4H-imidazo[5,1-c][1,4]benzoxazine-3-carboxamide Derivative for Depression and Anxiety
Giubellina, Nicola, Stabile, Paolo, Laval, Gilles, Perboni, Alcide D, Cimarosti, Zadeo, Westerduin, Pieter, Cooke, Jason W. B
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
Get full text
Journal Article
A Mechanistic Insight into a Simple C−N Bond Formation via S N 2 Displacement: A Synergistic Kinetics and Design of Experiment Approach
Massari, Luca, Panelli, Laura, Hughes, Mark, Stazi, Federica, Maton, William, Westerduin, Pieter, Scaravelli, Federico, Bacchi, Sergio
Published in Organic process research & development (19.11.2010)
Published in Organic process research & development (19.11.2010)
Get full text
Journal Article
Overall Synthesis of GSK356278: Quick Delivery of a PDE4 Inhibitor Using a Fit-for-Purpose Approach
Guercio, Giuseppe, Castoldi, Damiano, Giubellina, Nicola, Lamonica, Alessandro, Ribecai, Arianna, Stabile, Paolo, Westerduin, Pieter, Dams, Riet, Nicoletti, Anna, Rossi, Sara, Bismara, Claudio, Provera, Stefano, Turco, Lucilla
Published in Organic process research & development (17.09.2010)
Published in Organic process research & development (17.09.2010)
Get full text
Journal Article