Species Specificity of Amidine-Based Urokinase Inhibitors
Klinghofer, Vered, Stewart, Kent, McGonigal, Tom, Smith, Richard, Sarthy, Aparna, Nienaber, Vicki, Butler, Chris, Dorwin, Sarah, Richardson, Paul, Weitzberg, Moshe, Wendt, Mike, Rockway, Todd, Zhao, Xumiao, Hulkower, Keren I, Giranda, Vincent L
Published in Biochemistry (Easton) (07.08.2001)
Published in Biochemistry (Easton) (07.08.2001)
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Journal Article
Probing Inhibitors Binding to Human Urokinase Crystals by Raman Microscopy: Implications for Compound Screening
Dong, Jian, Swift, Kerry, Matayoshi, Edmund, Nienaber, Vicki L, Weitzberg, Moshe, Rockway, Todd, Carey, Paul R
Published in Biochemistry (Easton) (21.08.2001)
Published in Biochemistry (Easton) (21.08.2001)
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Journal Article
N-(Fluorenyl-9-Methoxycarbonyl) Amino Acids, a Class of Antiinflammatory Agents With a different Mechanism of Action
Burch, Ronald M., Weitzberg, Moshe, Blok, Natalie, Muhlhauser, Richard, Martin, David, Farmer, Stephen G., Bator, Jenny M., Connor, Jane R., Ko, Chiew, Kuhn, Wendy, McMillan, Barbara A., Raynor, Maureen, Shearer, Barry G., Tiffany, Carol, Wilkins, Deidre E.
Published in Proceedings of the National Academy of Sciences - PNAS (15.01.1991)
Published in Proceedings of the National Academy of Sciences - PNAS (15.01.1991)
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Journal Article
NPC 15669 inhibits the reversed passive Arthus reaction in rats by blocking neutrophil recruitment
BURCH, R. M, CONNOR, J. R, BATOR, J. M, WEITZBERG, M, LAEMONT, K, NORONHA-BLOB, L, SULLIVAN, J. P, STERANKA, L. R
Published in The Journal of pharmacology and experimental therapeutics (01.12.1992)
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Published in The Journal of pharmacology and experimental therapeutics (01.12.1992)
Journal Article
Identification of Novel Binding Interactions in the Development of Potent, Selective 2-Naphthamidine Inhibitors of Urokinase. Synthesis, Structural Analysis, and SAR of N-Phenyl Amide 6-Substitution
Wendt, Michael D, Rockway, Todd W, Geyer, Andrew, McClellan, William, Weitzberg, Moshe, Zhao, Xumiao, Mantei, Robert, Nienaber, Vicki L, Stewart, Kent, Klinghofer, Vered, Giranda, Vincent L
Published in Journal of medicinal chemistry (15.01.2004)
Published in Journal of medicinal chemistry (15.01.2004)
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Journal Article
Syntheses and chemistry of some dibenz[c,e]azepines
Weitzberg, Moshe, Abu-Shakra, Elias, Azeb, Abdullatif, Aizenshtat, Zeev, Blum, Jochanan
Published in Journal of organic chemistry (01.02.1987)
Published in Journal of organic chemistry (01.02.1987)
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Journal Article
N-{3-[2-(4-Alkoxyphenoxy)thiazol-5-yl]-1-methylprop-2-ynyl}carboxy Derivatives as Acetyl-CoA Carboxylase InhibitorsImprovement of Cardiovascular and Neurological Liabilities via Structural Modifications
Gu, Yu Gui, Weitzberg, Moshe, Clark, Richard F, Xu, Xiangdong, Li, Qun, Lubbers, Nathan L, Yang, Yi, Beno, David W. A, Widomski, Deborah L, Zhang, Tianyuan, Hansen, T. Matthew, Keyes, Robert F, Waring, Jeffrey F, Carroll, Sherry L, Wang, Xiaojun, Wang, Rongqi, Healan-Greenberg, Christine H, Blomme, Eric A, Beutel, Bruce A, Sham, Hing L, Camp, Heidi S
Published in Journal of medicinal chemistry (08.03.2007)
Published in Journal of medicinal chemistry (08.03.2007)
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Journal Article
Structure-directed discovery of potent non-peptidic inhibitors of human urokinase that access a novel binding subsite
Nienaber, Vicki L, Davidson, Donald, Edalji, Rohinton, Giranda, Vincent L, Klinghofer, Vered, Henkin, Jack, Magdalinos, Peter, Mantei, Robert, Merrick, Sean, Severin, Jean M, Smith, Richard A, Stewart, Kent, Walter, Karl, Wang, Jieyi, Wendt, Michael, Weitzberg, Moshe, Zhao, Xumiao, Rockway, Todd
Published in Structure (London) (15.05.2000)
Published in Structure (London) (15.05.2000)
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Journal Article
Novel Antibacterial Class
DANDLIKER, Peter J, PRATT, Steve D, CHOVAN, Linda E, HICKMAN, Robert K, DALY, Melissa M, KAKAVAS, Stephan, PING ZHONG, ZHENSHENG CAO, DAVID, Caroline A, XIAOLING XUEI, LERNER, Claude G, SONI, Niru B, NILIUS, Angela M, MAI BUI, SHEN, Linus L, YINGNA CAI, MERTA, Philip J, SAIKI, Anne Y. C, BEUTEL, Bruce A, BLACK-SCHAEFER, Candace, XIAOAN RUAN, TOWNE, Danli L, CLARK, Richard F, ENGLUND, Erika E, WAGNER, Rolf, WEITZBERG, Moshe
Published in Antimicrobial Agents and Chemotherapy (01.12.2003)
Published in Antimicrobial Agents and Chemotherapy (01.12.2003)
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Journal Article
Naphthamidine urokinase plasminogen activator inhibitors with improved pharmacokinetic properties
Bruncko, Milan, McClellan, William J., Wendt, Michael D., Sauer, Daryl R., Geyer, Andrew, Dalton, Christopher R., Kaminski, Michele A., Weitzberg, Moshe, Gong, Jane, Dellaria, Joseph F., Mantei, Robert, Zhao, Xumiao, Nienaber, Vicki L., Stewart, Kent, Klinghofer, Vered, Bouska, Jennifer, Rockway, Todd W., Giranda, Vincent L.
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
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Journal Article
Novel inhibitors of bacterial protein synthesis: structure–activity relationships for 1,8-naphthyridine derivatives incorporating position 3 and 4 variants
Clark, Richard F., Wang, Sanyi, Ma, Zhenkun, Weitzberg, Moshe, Motter, Christopher, Tufano, Michael, Wagner, Rolf, Gu, Yu-Gui, Dandliker, Peter J., Lerner, Claude G., Chovan, Linda E., Cai, Yingna, Black-Schaefer, Candace L., Lynch, Linda, Kalvin, Douglas, Nilius, Angela M., Pratt, Steve D., Soni, Niru, Zhang, Tianyuan, Zhang, Xiaolin, Beutel, Bruce A.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Journal Article
NPC 15669 enhances survival and reverses leukopenia in endotoxin-treated mice
Noronha-Blob, L, Lowe, V C, Weitzberg, M, Burch, R M
Published in European journal of pharmacology (09.07.1991)
Published in European journal of pharmacology (09.07.1991)
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Journal Article
ASYMMETRIC MICHAEL ADDITIONS OF ESTER ENOLATES TO ENANTIOMERICALLY PURE VINYLIC SULFOXIDES - SYNTHESIS OF 3-SUBSTITUTED GLUTARATE ESTERS IN HIGH ENANTIOMERIC PURITY
POSNER, GH, WEITZBERG, M, HAMILL, TG, ASIRVATHAM, E, HE, CH, CLARDY, J
Published in Tetrahedron (01.01.1986)
Published in Tetrahedron (01.01.1986)
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Journal Article
An improved synthesis of carbocyclic and heterocyclic arene imines
Weitzberg, Moshe, Aizenshtat, Zeev, Jerushalmy, Parvin, Blum, Jochanan
Published in Journal of organic chemistry (01.10.1980)
Published in Journal of organic chemistry (01.10.1980)
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Journal Article
Synthesis of some 3-(1-azabicyclo[2.2.2]octyl) 3-amino-2-hydroxy-2-phenylpropionates: profile of antimuscarinic efficacy and selectivity
Audia, Vicki H, McPherson, Daniel W, Weitzberg, Moshe, Rzeszotarski, W. Janusz, Sturm, Bonnie, Kachur, James F, Abreu, Mary, Kaiser, Carl
Published in Journal of medicinal chemistry (01.01.1990)
Published in Journal of medicinal chemistry (01.01.1990)
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Journal Article
1,2-Dioxetanes from vinyl aromatics
Posner, Gary H, Weitzberg, Moshe, Nelson, William M, Murr, Brown L, Seliger, Howard H
Published in Journal of the American Chemical Society (01.01.1987)
Published in Journal of the American Chemical Society (01.01.1987)
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Journal Article
Oxidative addition of aryl halides to iridium(I) complexes. A new arylation reagent
Blum, Jochanan, Weitzberg, Moshe, Mureinik, Roland J.
Published in Journal of organometallic chemistry (01.01.1976)
Published in Journal of organometallic chemistry (01.01.1976)
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