Editorial: Incorporating Phase 0 microdosing as a powerful tool into a new vision of drug development
Weiss, H. Markus, Sugiyama, Yuichi, van Duijn, Esther
Published in Frontiers in pharmacology (16.07.2024)
Published in Frontiers in pharmacology (16.07.2024)
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Journal Article
A Study of the Effect of Cyclosporine on Fevipiprant Pharmacokinetics and its Absolute Bioavailability Using an Intravenous Microdose Approach
Weiss, H Markus, Umehara, Ken-Ichi, Erpenbeck, Veit J, Cain, Meredith, Vemula, Janardhana, Elbast, Walid, Zollinger, Markus
Published in Drug metabolism and disposition (01.10.2020)
Published in Drug metabolism and disposition (01.10.2020)
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Journal Article
Biodistribution and Plasma Protein Binding of Zoledronic Acid
MARKUS WEISS, H, PFAAR, Ulrike, SCHWEITZER, Alain, WIEGAND, Hansjörg, SKERJANEC, Andrej, SCHRAN, Horst
Published in Drug metabolism and disposition (01.10.2008)
Published in Drug metabolism and disposition (01.10.2008)
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Journal Article
LTA4H inhibitor LYS006: Clinical PK/PD and safety in a randomized phase I clinical trial
Loesche, Christian, Picard, Damien, Van Hoorick, Benjamin, Schuhmann, Imelda, Jäger, Petra, Klein, Kai, Schuhler, Carole, Thoma, Gebhard, Markert, Christian, Poller, Birk, Zamurovic, Natasa, Weiss, H. Markus, Otto, Heike, Fink, Martin, Röhn, Till A.
Published in Clinical and translational science (01.02.2024)
Published in Clinical and translational science (01.02.2024)
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Journal Article
Binding of Pimecrolimus and Tacrolimus to Skin and Plasma Proteins: Implications for Systemic Exposure after Topical Application
WEISS, H. Markus, FRESNEAU, Marcel, MOENIUS, Thomas, STUETZ, Anton, BILLICH, Andreas
Published in Drug metabolism and disposition (01.09.2008)
Published in Drug metabolism and disposition (01.09.2008)
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Journal Article
Clinical Investigation of Metabolic and Renal Clearance Pathways Contributing to the Elimination of Fevipiprant Using Probenecid as Perpetrator
Weiss, H Markus, Langenickel, Thomas, Cain, Meredith, Kulkarni, Swarupa, Shah, Bharti, Vemula, Janardhana, Rahmanzadeh, Gholamreza, Poller, Birk
Published in Drug metabolism and disposition (01.05.2021)
Published in Drug metabolism and disposition (01.05.2021)
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Journal Article
Metabolism and disposition of the oral absorption enhancer 14C-radiolabeled 8-(N-2-hydroxy-5-chlorobenzoyl)-amino-caprylic acid (5-CNAC) in healthy postmenopausal women and supplementary investigations in vitro
Gschwind, Hans-Peter, Glaenzel, Ulrike, Waldmeier, Felix, Wirz, Bernard, Sabia, Helene D., Picard, Franck, Markus Weiss, H., Choi, Leslie, Swart, Pieter Jacob, Vasudevan, Ajithkumar, Azria, Moïse
Published in European journal of pharmaceutical sciences (30.08.2012)
Published in European journal of pharmaceutical sciences (30.08.2012)
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Journal Article
Human Pharmacokinetics of LYS006, an Oral Leukotriene A4 Hydrolase Inhibitor Displaying Target-Mediated Drug Disposition
Poller, Birk, Pearson, David, Leuthold, Luc Alexis, Fink, Martin, Jullion, Astrid, Schweigler, Patrick, Tor Carreras, Ester, Marvalin, Cyrille, Loesche, Christian, Weiss, H. Markus
Published in Drug metabolism and disposition (01.12.2022)
Published in Drug metabolism and disposition (01.12.2022)
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Journal Article
HEPATIC TRANSPORT OF PKI166, AN EPIDERMAL GROWTH FACTOR RECEPTOR KINASE INHIBITOR OF THE PYRROLO-PYRIMIDINE CLASS, AND ITS MAIN METABOLITE, ACU154
TAKADA, Tappei, WEISS, H. Markus, KRETZ, Olivier, GROSS, Gerhard, SUGIYAMA, Yuichi
Published in Drug metabolism and disposition (01.11.2004)
Published in Drug metabolism and disposition (01.11.2004)
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Journal Article
Fevipiprant (QAW039) does not affect the pharmacokinetics of zidovudine, its glucuronide, and penicillin G via inhibition of UGT2B7 and/or OAT3
Kulkarni, Swarupa, Poller, Birk, Drollmann, Anton, Shah, Bharti, Gray, Cathy, Greco, Erin, Rahmanzadeh, Gholamreza, Hanna, Imad, Weiss, H Markus
Published in Pulmonary pharmacology & therapeutics (01.02.2022)
Published in Pulmonary pharmacology & therapeutics (01.02.2022)
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Journal Article
Absorption, Distribution, Metabolism, and Excretion of the Oral Prostaglandin D2 Receptor 2 Antagonist Fevipiprant (QAW039) in Healthy Volunteers and In Vitro
Pearson, David, Weiss, H Markus, Jin, Yi, Jaap van Lier, Jan, Erpenbeck, Veit J, Glaenzel, Ulrike, End, Peter, Woessner, Ralph, Eggimann, Fabian, Camenisch, Gian
Published in Drug metabolism and disposition (01.07.2017)
Published in Drug metabolism and disposition (01.07.2017)
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Journal Article
IN VITRO BLOOD DISTRIBUTION AND PLASMA PROTEIN BINDING OF THE IRON CHELATOR DEFERASIROX (ICL670) AND ITS IRON COMPLEX FE-[ICL670]2 FOR RAT, MARMOSET, RABBIT, MOUSE, DOG, AND HUMAN
MARKUS WEISS, H, FRESNEAU, Marcel, CAMENISCH, Gian P, KRETZ, Olivier, GROSS, Gerhard
Published in Drug metabolism and disposition (01.06.2006)
Published in Drug metabolism and disposition (01.06.2006)
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Journal Article
In vitro blood distribution and plasma protein binding of the tyrosine kinase inhibitor imatinib and its active metabolite, CGP74588, in rat, mouse, dog, monkey, healthy humans and patients with acute lymphatic leukaemia
Kretz, Olivier, Weiss, H Markus, Schumacher, Martin M, Gross, Gerhard
Published in British journal of clinical pharmacology (01.08.2004)
Published in British journal of clinical pharmacology (01.08.2004)
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Journal Article
Comparative biochemical and pharmacological characterization of the mouse 5HT5A 5-hydroxytryptamine receptor and the human β2-adrenergic receptor produced in the methylotrophic yeast Pichia pastoris
WEISS, H. Markus, HAASE, Winfried, MICHEL, Hartmut, REILÄNDER, Helmut
Published in Biochemical journal (15.03.1998)
Published in Biochemical journal (15.03.1998)
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Journal Article
ADME Investigations of Unnatural Peptides: Distribution of a 14C-Labeled β 3-Octaarginine in Rats
Weiss, H. Markus, Wirz, Bernard, Schweitzer, Alain, Amstutz, René, Perez, Maria I. Rodriguez, Andres, Hendrik, Metz, Yves, Gardiner, James, Seebach, Dieter
Published in Chemistry & biodiversity (01.07.2007)
Published in Chemistry & biodiversity (01.07.2007)
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