RS-102221: A Novel High Affinity and Selective, 5-HT 2C Receptor Antagonist
BONHAUS, D.W, WEINHARDT, K.K, TAYLOR, M, DESOUZA, A, MCNEELEY, P.M, SZCZEPANSKI, K, FONTANA, D.J, TRINH, J, ROCHA, C.L, DAWSON, M.W, FLIPPIN, L.A, EGLEN, R.M
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Published in Neuropharmacology (01.04.1997)
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Synthesis and preliminary pharmacological evaluation of 2-benzyloxy substituted aryl ketones as 5-HT4 receptor antagonists
Clark, R.D., Jahangir, A., Langston, J.A., Weinhardt, K.K., Miller, A.B., Leung, E., Bonhaus, D.W., Wong, E.H.F., Eglen, R.M.
Published in Bioorganic & medicinal chemistry letters (01.10.1994)
Published in Bioorganic & medicinal chemistry letters (01.10.1994)
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N-(Quinuclidin-3-yl)-2-(1-methyl-1H-indol-3-yl)-2-oxo-acetamide: a high affinity 5-HT3 receptor partial agonist
Clark, R.D., Muchowski, J.M., Weinhardt, K.K., Dillon, M.P., Lee, C-H., Bley, K.R., Bonhaus, D.W., Wong, E.H.F., Eglen, R.M.
Published in Bioorganic & medicinal chemistry letters (17.08.1995)
Published in Bioorganic & medicinal chemistry letters (17.08.1995)
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Journal Article
N-(Quinuclidin-3-yl)-2-(1-methyl-1H-indol-3-yl)-2-oxo-acetamide: a high affinity 5-HT 3 receptor partial agonist
Clark, R.D., Muchowski, J.M., Weinhardt, K.K., Dillon, M.P., Lee, C-H., Bley, K.R., Bonhaus, D.W., Wong, E.H.F., Eglen, R.M.
Published in Bioorganic & medicinal chemistry letters (1995)
Published in Bioorganic & medicinal chemistry letters (1995)
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Journal Article
N-(quinuclidin-3-YL)-1,8,-naphthalimides with 5-HT3 receptor antagonist and 5-HT4 receptor agonist properties
Clark, R.D., Weinhardt, K.K., Berger, J., Lee, C.-H., Leung, E., Wong, E.H.F., Smith, W.L., Eglen, R.M.
Published in Bioorganic & medicinal chemistry letters (01.06.1993)
Published in Bioorganic & medicinal chemistry letters (01.06.1993)
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Journal Article
Synthesis and preliminary pharmacological evaluation of 2-benzyloxy substituted aryl ketones as 5-HT 4 receptor antagonists
Clark, R.D., Jahangir, A., Langston, J.A., Weinhardt, K.K., Miller, A.B., Leung, E., Bonhaus, D.W., Wong, E.H.F., Eglen, R.M.
Published in Bioorganic & medicinal chemistry letters (1994)
Published in Bioorganic & medicinal chemistry letters (1994)
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Journal Article
N-(quinuclidin-3-YL)-1,8,-naphthalimides with 5-HT 3 receptor antagonist and 5-HT 4 receptor agonist properties
Clark, R.D., Weinhardt, K.K., Berger, J., Lee, C.-H., Leung, E., Wong, E.H.F., Smith, W.L., Eglen, R.M.
Published in Bioorganic & medicinal chemistry letters (1993)
Published in Bioorganic & medicinal chemistry letters (1993)
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A new class of antimalarial drugs: derivatives of benzothiopyrans
Razdan, Raj K, Bruni, Robert J, Mehta, Avinash C, Weinhardt, Klaus K, Papanastassiou, Zinon B
Published in Journal of medicinal chemistry (01.07.1978)
Published in Journal of medicinal chemistry (01.07.1978)
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