IN VITRO P-GLYCOPROTEIN INHIBITION ASSAYS FOR ASSESSMENT OF CLINICAL DRUG INTERACTION POTENTIAL OF NEW DRUG CANDIDATES: A RECOMMENDATION FOR PROBE SUBSTRATES
Rautio, Jarkko, Humphreys, Joan E, Webster, Lindsey O, Balakrishnan, Anand, Keogh, John P, Kunta, Jeevan R, Serabjit-Singh, Cosette J, Polli, Joseph W
Published in Drug metabolism and disposition (01.05.2006)
Published in Drug metabolism and disposition (01.05.2006)
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Passive Permeability and P-Glycoprotein-Mediated Efflux Differentiate Central Nervous System (CNS) and Non-CNS Marketed Drugs
Mahar Doan, Kelly M, Humphreys, Joan E, Webster, Lindsey O, Wring, Stephen A, Shampine, Larry J, Serabjit-Singh, Cosette J, Adkison, Kimberly K, Polli, Joseph W
Published in The Journal of pharmacology and experimental therapeutics (01.12.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2002)
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In vitro investigations into the roles of drug transporters and metabolizing enzymes in the disposition and drug interactions of dolutegravir, a HIV integrase inhibitor
Reese, Melinda J, Savina, Paul M, Generaux, Grant T, Tracey, Helen, Humphreys, Joan E, Kanaoka, Eri, Webster, Lindsey O, Harmon, Kelly A, Clarke, James D, Polli, Joseph W
Published in Drug metabolism and disposition (01.02.2013)
Published in Drug metabolism and disposition (01.02.2013)
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MULTIPLE MECHANISMS ARE INVOLVED IN THE BILIARY EXCRETION OF ACETAMINOPHEN SULFATE IN THE RAT: ROLE OF MRP2 AND BCRP1
Zamek-Gliszczynski, Maciej J, Hoffmaster, Keith A, Tian, Xianbin, Zhao, Rong, Polli, Joseph W, Humphreys, Joan E, Webster, Lindsey O, Bridges, Arlene S, Kalvass, J Cory, Brouwer, Kim L R
Published in Drug metabolism and disposition (01.08.2005)
Published in Drug metabolism and disposition (01.08.2005)
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Drug interaction profile of the HIV integrase inhibitor cabotegravir: assessment from in vitro studies and a clinical investigation with midazolam
Reese, Melinda J., Bowers, Gary D., Humphreys, Joan E., Gould, Elizabeth P., Ford, Susan L., Webster, Lindsey O., Polli, Joseph W.
Published in Xenobiotica (03.05.2016)
Published in Xenobiotica (03.05.2016)
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THE SYSTEMIC EXPOSURE OF AN N-METHYL-d-ASPARTATE RECEPTOR ANTAGONIST IS LIMITED IN MICE BY THE P-GLYCOPROTEIN AND BREAST CANCER RESISTANCE PROTEIN EFFLUX TRANSPORTERS
POLLI, Joseph W, BAUGHMAN, Todd M, SERABJIT-SINGH, Cosette J, HUMPHREYS, Joan E, JORDAN, Kelly H, MOTE, Angela L, WEBSTER, Lindsey O, BARNABY, Robert J, VITULLI, Giovanni, BERTOLOTTI, Luigina, READ, Kevin D
Published in Drug metabolism and disposition (01.07.2004)
Published in Drug metabolism and disposition (01.07.2004)
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Rational Use of in Vitro P-glycoprotein Assays in Drug Discovery
Joseph W. Polli, Stephen A. Wring, Joan E. Humphreys, Liyue Huang, Jonathon B. Morgan, Lindsey O. Webster, Cosette S. Serabjit-Singh
Published in The Journal of pharmacology and experimental therapeutics (01.11.2001)
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Published in The Journal of pharmacology and experimental therapeutics (01.11.2001)
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Hepatic Phospholipidosis Is Associated with Altered Hepatobiliary Function as Assessed by Gadoxetate Dynamic Contrast-enhanced Magnetic Resonance Imaging
Lenhard, Stephen C, Lev, Mally, Webster, Lindsey O, Peterson, Richard A, Goulbourne, Christopher N, Miller, Richard T, Jucker, Beat M
Published in Toxicologic pathology (01.01.2016)
Published in Toxicologic pathology (01.01.2016)
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Use of cassette dosing in sandwich-cultured rat and human hepatocytes to identify drugs that inhibit bile acid transport
Wolf, Kristina K., Vora, Sapana, Webster, Lindsey O., Generaux, Grant T., Polli, Joseph W., Brouwer, Kim L.R.
Published in Toxicology in vitro (01.02.2010)
Published in Toxicology in vitro (01.02.2010)
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Temporal kinetics and concentration-response relationships for induction of CYP1A, CYP2B, and CYP3A in primary cultures of beagle dog hepatocytes
Graham, Richard A., Tyler, Lindsey O., Krol, Wojciech L., Silver, Ivin S., Webster, Lindsey O., Clark, Philip, Chen, Liangfu, Banks, Troy, LeCluyse, Edward L.
Published in Journal of biochemical and molecular toxicology (01.01.2006)
Published in Journal of biochemical and molecular toxicology (01.01.2006)
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