Design of potent thiophene inhibitors of polo-like kinase 1 with improved solubility and reduced protein binding
EMMITTE, Kyle A, ADJEBANG, George M, JACKSON, Jeffrey R, KUNTZ, Kevin W, LANSING, Timothy J, MOOK, Robert A, NAILOR, Kristen E, POBANZ, Mark A, SMITH, Stephon C, SUNG, Chiu-Mei, CHEUNG, Mui, WEBB ANDREWS, C, BADIANG ALBERTI, Jennifer G, BAMBAL, Ramesh, CHAMBERLAIN, Stanley D, DAVIS-WARD, Ronda G, DICKSON, Hamilton D, HASSLER, Daniel F, HORNBERGER, Keith R
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
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Discovery of thiophene inhibitors of polo-like kinase
Emmitte, Kyle A., Andrews, C. Webb, Badiang, Jennifer G., Davis-Ward, Ronda G., Dickson, Hamilton D., Drewry, David H., Emerson, Holly K., Epperly, Andrea H., Hassler, Daniel F., Knick, Victoria B., Kuntz, Kevin W., Lansing, Timothy J., Linn, James A., Mook, Robert A., Nailor, Kristen E., Salovich, James M., Spehar, Glenn M., Cheung, Mui
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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Heteroaryl-linked 5-(1H-benzimidazol-1-yl)-2-thiophenecarboxamides: Potent inhibitors of polo-like kinase 1 (PLK1) with improved drug-like properties
Rheault, Tara R., Donaldson, Kelly H., Badiang-Alberti, Jennifer G., Davis-Ward, Ronda G., Andrews, C. Webb, Bambal, Ramesh, Jackson, Jeffrey R., Cheung, Mui
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Corrigendum to “Design of potent thiophene inhibitors of polo-like kinase 1 with improved solubility and reduced protein binding” [Bioorg. Med. Chem. Lett. 19 (2009) 1694]
Emmitte, Kyle A., Adjabeng, George M., Webb Andrews, C., Badiang Alberti, Jennifer G., Bambal, Ramesh, Chamberlain, Stanley D., Davis-Ward, Ronda G., Dickson, Hamilton D., Hassler, Daniel F., Hornberger, Keith R., Jackson, Jeffrey R., Kuntz, Kevin W., Lansing, Timothy J., Mook, Robert A., Nailor, Kristen E., Pobanz, Mark A., Smith, Stephon C., Sung, Chiu-Mei, Cheung, Mui
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Degenerate Racemization of Chiral Saddle Conformations in a Cyclic Dioxadithia Aryl Polyether
Boros, Eric E, Andrews, C. Webb, Davis, Ann O
Published in Journal of organic chemistry (05.04.1996)
Published in Journal of organic chemistry (05.04.1996)
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Novel carbohydrate transformations discovered en route to natural products
Fraser-Reid, B., Mootoo, D. R., Konradsson, P., Udodong, U. E., Andrews, C. Webster, Ratcliffe, A. J., Wu, Z., Yu, K. L.
Published in Pure and applied chemistry (01.01.1989)
Published in Pure and applied chemistry (01.01.1989)
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