An Allosteric Inhibitor of the Human Cdc34 Ubiquitin-Conjugating Enzyme
Ceccarelli, Derek F., Tang, Xiaojing, Pelletier, Benoit, Orlicky, Stephen, Xie, Weilin, Plantevin, Veronique, Neculai, Dante, Chou, Yang-Chieh, Ogunjimi, Abiodun, Al-Hakim, Abdallah, Varelas, Xaralabos, Koszela, Joanna, Wasney, Gregory A., Vedadi, Masoud, Dhe-Paganon, Sirano, Cox, Sarah, Xu, Shuichan, Lopez-Girona, Antonia, Mercurio, Frank, Wrana, Jeff, Durocher, Daniel, Meloche, Sylvain, Webb, David R., Tyers, Mike, Sicheri, Frank
Published in Cell (24.06.2011)
Published in Cell (24.06.2011)
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Recognition and Specificity Determinants of the Human Cbx Chromodomains
Kaustov, Lilia, Ouyang, Hui, Amaya, Maria, Lemak, Alexander, Nady, Nataliya, Duan, Shili, Wasney, Gregory A., Li, Zhihong, Vedadi, Masoud, Schapira, Matthieu, Min, Jinrong, Arrowsmith, Cheryl H.
Published in The Journal of biological chemistry (07.01.2011)
Published in The Journal of biological chemistry (07.01.2011)
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Multivalency transforms SARS-CoV-2 antibodies into ultrapotent neutralizers
Rujas, Edurne, Kucharska, Iga, Tan, Yong Zi, Benlekbir, Samir, Cui, Hong, Zhao, Tiantian, Wasney, Gregory A, Budylowski, Patrick, Guvenc, Furkan, Newton, Jocelyn C, Sicard, Taylor, Semesi, Anthony, Muthuraman, Krithika, Nouanesengsy, Amy, Aschner, Clare Burn, Prieto, Katherine, Bueler, Stephanie A, Youssef, Sawsan, Liao-Chan, Sindy, Glanville, Jacob, Christie-Holmes, Natasha, Mubareka, Samira, Gray-Owen, Scott D, Rubinstein, John L, Treanor, Bebhinn, Julien, Jean-Philippe
Published in Nature communications (16.06.2021)
Published in Nature communications (16.06.2021)
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Delineating Structural Propensities of the 4E-BP2 Protein via Integrative Modeling and Clustering
Tsangaris, Thomas E., Smyth, Spencer, Gomes, Gregory-Neal W., Liu, Zi Hao, Milchberg, Moses, Bah, Alaji, Wasney, Gregory A., Forman-Kay, Julie D., Gradinaru, Claudiu C.
Published in The journal of physical chemistry. B (31.08.2023)
Published in The journal of physical chemistry. B (31.08.2023)
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Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5
Senisterra, Guillermo, Wu, Hong, Allali-Hassani, Abdellah, Wasney, Gregory A, Barsyte-Lovejoy, Dalia, Dombrovski, Ludmila, Dong, Aiping, Nguyen, Kong T, Smil, David, Bolshan, Yuri, Hajian, Taraneh, He, Hao, Seitova, Alma, Chau, Irene, Li, Fengling, Poda, Gennadiy, Couture, Jean-François, Brown, Peter J, Al-Awar, Rima, Schapira, Matthieu, Arrowsmith, Cheryl H, Vedadi, Masoud
Published in Biochemical journal (01.01.2013)
Published in Biochemical journal (01.01.2013)
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Structure and Mechanism of Staphylococcus aureus TarS, the Wall Teichoic Acid β-glycosyltransferase Involved in Methicillin Resistance
Sobhanifar, Solmaz, Worrall, Liam J, King, Dustin T, Wasney, Gregory A, Baumann, Lars, Gale, Robert T, Nosella, Michael, Brown, Eric D, Withers, Stephen G, Strynadka, Natalie C J
Published in PLoS pathogens (01.12.2016)
Published in PLoS pathogens (01.12.2016)
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Discovery of a 2,4-Diamino-7-aminoalkoxyquinazoline as a Potent and Selective Inhibitor of Histone Lysine Methyltransferase G9a
Liu, Feng, Chen, Xin, Allali-Hassani, Abdellah, Quinn, Amy M, Wasney, Gregory A, Dong, Aiping, Barsyte, Dalia, Kozieradzki, Ivona, Senisterra, Guillermo, Chau, Irene, Siarheyeva, Alena, Kireev, Dmitri B, Jadhav, Ajit, Herold, J. Martin, Frye, Stephen V, Arrowsmith, Cheryl H, Brown, Peter J, Simeonov, Anton, Vedadi, Masoud, Jin, Jian
Published in Journal of medicinal chemistry (24.12.2009)
Published in Journal of medicinal chemistry (24.12.2009)
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An Allosteric Inhibitor of Protein Arginine Methyltransferase 3
Siarheyeva, Alena, Senisterra, Guillermo, Allali-Hassani, Abdellah, Dong, Aiping, Dobrovetsky, Elena, Wasney, Gregory A., Chau, Irene, Marcellus, Richard, Hajian, Taraneh, Liu, Feng, Korboukh, Ilia, Smil, David, Bolshan, Yuri, Min, Jinrong, Wu, Hong, Zeng, Hong, Loppnau, Peter, Poda, Gennadiy, Griffin, Carly, Aman, Ahmed, Brown, Peter J., Jin, Jian, Al-awar, Rima, Arrowsmith, Cheryl H., Schapira, Matthieu, Vedadi, Masoud
Published in Structure (London) (08.08.2012)
Published in Structure (London) (08.08.2012)
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Chemical Screening Methods to Identify Ligands That Promote Protein Stability, Protein Crystallization, and Structure Determination
Vedadi, Masoud, Niesen, Frank H., Allali-Hassani, Abdellah, Fedorov, Oleg Y., Finerty, Patrick J., Wasney, Gregory A., Yeung, Ron, Arrowsmith, Cheryl, Ball, Linda J., Berglund, Helena, Hui, Raymond, Marsden, Brian D., Nordlund, Pär, Sundstrom, Michael, Weigelt, Johan, Edwards, Aled M.
Published in Proceedings of the National Academy of Sciences - PNAS (24.10.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (24.10.2006)
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The Modular Structure of the Inner-Membrane Ring Component PrgK Facilitates Assembly of the Type III Secretion System Basal Body
Bergeron, Julien R.C., Worrall, Liam J., De, Soumya, Sgourakis, Nikolaos G., Cheung, Adrienne H., Lameignere, Emilie, Okon, Mark, Wasney, Gregory A., Baker, David, McIntosh, Lawrence P., Strynadka, Natalie C.J.
Published in Structure (London) (06.01.2015)
Published in Structure (London) (06.01.2015)
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Structure and mechanism of Staphylococcus aureus TarM, the wall teichoic acid α-glycosyltransferase
Sobhanifar, Solmaz, Worrall, Liam James, Gruninger, Robert J, Wasney, Gregory A, Blaukopf, Markus, Baumann, Lars, Lameignere, Emilie, Solomonson, Matthew, Brown, Eric D, Withers, Stephen G, Strynadka, Natalie C J
Published in Proceedings of the National Academy of Sciences - PNAS (10.02.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (10.02.2015)
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Protein Lysine Methyltransferase G9a Inhibitors: Design, Synthesis, and Structure Activity Relationships of 2,4-Diamino-7-aminoalkoxy-quinazolines
Liu, Feng, Chen, Xin, Allali-Hassani, Abdellah, Quinn, Amy M, Wigle, Tim J, Wasney, Gregory A, Dong, Aiping, Senisterra, Guillermo, Chau, Irene, Siarheyeva, Alena, Norris, Jacqueline L, Kireev, Dmitri B, Jadhav, Ajit, Herold, J. Martin, Janzen, William P, Arrowsmith, Cheryl H, Frye, Stephen V, Brown, Peter J, Simeonov, Anton, Vedadi, Masoud, Jin, Jian
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
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The Structure of a Type 3 Secretion System (T3SS) Ruler Protein Suggests a Molecular Mechanism for Needle Length Sensing
Bergeron, Julien R.C., Fernández, Lucia, Wasney, Gregory A., Vuckovic, Marija, Reffuveille, Fany, Hancock, Robert E.W., Strynadka, Natalie C.J.
Published in The Journal of biological chemistry (22.01.2016)
Published in The Journal of biological chemistry (22.01.2016)
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Identification of a PGXPP degron motif in dishevelled and structural basis for its binding to the E3 ligase KLHL12
Chen, Zhuoyao, Wasney, Gregory A, Picaud, Sarah, Filippakopoulos, Panagis, Vedadi, Masoud, D'Angiolella, Vincenzo, Bullock, Alex N
Published in Open biology (01.06.2020)
Published in Open biology (01.06.2020)
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Polyphosphate suppresses complement via the terminal pathway
Wat, Jovian M., Foley, Jonathan H., Krisinger, Michael J., Ocariza, Linnette Mae, Lei, Victor, Wasney, Gregory A., Lameignere, Emilie, Strynadka, Natalie C., Smith, Stephanie A., Morrissey, James H., Conway, Edward M.
Published in Blood (30.01.2014)
Published in Blood (30.01.2014)
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Structural studies of the tandem Tudor domains of fragile X mental retardation related proteins FXR1 and FXR2
Adams-Cioaba, Melanie A, Guo, Yahong, Bian, ChuanBing, Amaya, Maria F, Lam, Robert, Wasney, Gregory A, Vedadi, Masoud, Xu, Chao, Min, Jinrong
Published in PloS one (02.11.2010)
Published in PloS one (02.11.2010)
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Small Molecule Inhibition of an Exopolysaccharide Modification Enzyme is a Viable Strategy To Block Pseudomonas aeruginosa Pel Biofilm Formation
Razvi, Erum, DiFrancesco, Benjamin R, Wasney, Gregory A, Morrison, Zachary A, Tam, John, Auger, Anick, Baker, Perrin, Alnabelseya, Noor, Rich, Jacquelyn D, Sivarajah, Piyanka, Whitfield, Gregory B, Harrison, Joe J, Melnyk, Roman A, Nitz, Mark, Howell, P Lynne
Published in Microbiology spectrum (15.06.2023)
Published in Microbiology spectrum (15.06.2023)
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Genome-scale protein expression and structural biology of Plasmodium falciparum and related Apicomplexan organisms
Vedadi, Masoud, Lew, Jocelyne, Artz, Jennifer, Amani, Mehrnaz, Zhao, Yong, Dong, Aiping, Wasney, Gregory A., Gao, Mian, Hills, Tanya, Brokx, Stephen, Qiu, Wei, Sharma, Sujata, Diassiti, Angelina, Alam, Zahoor, Melone, Michelle, Mulichak, Anne, Wernimont, Amy, Bray, James, Loppnau, Peter, Plotnikova, Olga, Newberry, Kate, Sundararajan, Emayavaram, Houston, Simon, Walker, John, Tempel, Wolfram, Bochkarev, Alexey, Kozieradzki, Ivona, Edwards, Aled, Arrowsmith, Cheryl, Roos, David, Kain, Kevin, Hui, Raymond
Published in Molecular and biochemical parasitology (01.01.2007)
Published in Molecular and biochemical parasitology (01.01.2007)
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A survey of proteins encoded by non-synonymous single nucleotide polymorphisms reveals a significant fraction with altered stability and activity
Allali-Hassani, Abdellah, Wasney, Gregory A, Chau, Irene, Hong, Bum Soo, Senisterra, Guillermo, Loppnau, Peter, Shi, Zhen, Moult, John, Edwards, Aled M, Arrowsmith, Cheryl H, Park, Hee Won, Schapira, Matthieu, Vedadi, Masoud
Published in Biochemical journal (15.11.2009)
Published in Biochemical journal (15.11.2009)
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