Discovery of potent and novel S-nitrosoglutathione reductase inhibitors devoid of cytochrome P450 activities
Sun, Xicheng, Qiu, Jian, Strong, Sarah A., Green, Louis S., Wasley, Jan W.F., Blonder, Joan P., Colagiovanni, Dorothy B., Mutka, Sarah C., Stout, Adam M., Richards, Jane P., Rosenthal, Gary J.
Published in Bioorganic & medicinal chemistry letters (01.10.2011)
Published in Bioorganic & medicinal chemistry letters (01.10.2011)
Get full text
Journal Article
Structure–activity relationship of pyrrole based S-nitrosoglutathione reductase inhibitors: Carboxamide modification
Sun, Xicheng, Qiu, Jian, Strong, Sarah A., Green, Louis S., Wasley, Jan W.F., Blonder, Joan P., Colagiovanni, Dorothy B., Stout, Adam M., Mutka, Sarah C., Richards, Jane P., Rosenthal, Gary J.
Published in Bioorganic & medicinal chemistry letters (15.03.2012)
Published in Bioorganic & medicinal chemistry letters (15.03.2012)
Get full text
Journal Article
Structure–activity relationships of pyrrole based S-nitrosoglutathione reductase inhibitors: Pyrrole regioisomers and propionic acid replacement
Sun, Xicheng, Qiu, Jian, Strong, Sarah A., Green, Louis S., Wasley, Jan W.F., Colagiovanni, Dorothy B., Mutka, Sarah C., Blonder, Joan P., Stout, Adam M., Richards, Jane P., Chun, Lawrence, Rosenthal, Gary J.
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Get full text
Journal Article
Discovery of S-Nitrosoglutathione Reductase Inhibitors: Potential Agents for the Treatment of Asthma and Other Inflammatory Diseases
Sun, Xicheng, Wasley, Jan W. F, Qiu, Jian, Blonder, Joan P, Stout, Adam M, Green, Louis S, Strong, Sarah A, Colagiovanni, Dorothy B, Richards, Jane P, Mutka, Sarah C, Chun, Lawrence, Rosenthal, Gary J
Published in ACS medicinal chemistry letters (12.05.2011)
Published in ACS medicinal chemistry letters (12.05.2011)
Get full text
Journal Article
trans-1-[(2-Phenylcyclopropyl)methyl]-4-arylpiperazines: Mixed Dopamine D2/D4 Receptor Antagonists as Potential Antipsychotic Agents
Zhang, Xiaoyan, Hodgetts, Kevin, Rachwal, Stanislaw, Zhao, He, Wasley, Jan W. F, Craven, Kimberly, Brodbeck, Robbin, Kieltyka, Andrzej, Hoffman, Diane, Bacolod, Maria D, Girard, Brian, Tran, Jennifer, Thurkauf, Andrew
Published in Journal of medicinal chemistry (19.10.2000)
Published in Journal of medicinal chemistry (19.10.2000)
Get full text
Journal Article
1H-pyrazolo-[3,4-c]cyclophepta[1,2-c]thiophenes: A unique structural class of dopamine D4 selective ligands
THURKAUF, Andrew, XI CHEN, SUOMING ZHANG, YANG GAO, KIELTYKA, Andrzej, WASLEY, Jan W. F, BRODBECK, Robbin, GREENLEE, William, GANGULY, Ashit, HE ZHAO
Published in Bioorganic & medicinal chemistry letters (01.09.2003)
Published in Bioorganic & medicinal chemistry letters (01.09.2003)
Get full text
Journal Article
beta.-Lapachone: synthesis of derivatives and activities in tumor models
Schaffner-Sabba, Karl, Schmidt-Ruppin, Karl H, Wehrli, Walter, Schuerch, Alfred R, Wasley, Jan W. F
Published in Journal of medicinal chemistry (01.08.1984)
Published in Journal of medicinal chemistry (01.08.1984)
Get full text
Journal Article
2-Phenyl-4(5)-[[4-(pyrimidin-2- yl)piperazin-1-yl]methyl]imidazole. A Highly Selective Antagonist at Cloned Human D4 Receptors
Thurkauf, Andrew, Yuan, Jun, Chen, Xi, He, Xiao Shu, Wasley, Jan W. F, Hutchison, Alan, Woodruff, Kristine H, Meade, Robin, Hoffman, Diane C, Donovan, Hilary, Jones-Hertzog, Deborah K
Published in Journal of medicinal chemistry (03.01.1997)
Published in Journal of medicinal chemistry (03.01.1997)
Get full text
Journal Article
1-Phenyl-3-(aminomethyl)pyrroles as Potential Antipsychotic Agents. Synthesis and Dopamine Receptor Binding
Thurkauf, Andrew, Yuan, Jun, Chen, Nathan, Wasley, Jan W. F, Meade, Robin, Woodruff, Kristine Harris, Huston, Kevin, Ross, Philip C
Published in Journal of medicinal chemistry (01.12.1995)
Published in Journal of medicinal chemistry (01.12.1995)
Get full text
Journal Article
Indoline and piperazine containing derivatives as a novel class of mixed D2/D4 receptor antagonists. Part 2: Asymmetric synthesis and biological evaluation
HE ZHAO, XIAOSHU HE, THURKAUF, Andrew, HOFFMAN, Diane, KIELTYKA, Andrzej, BRODBECK, Robbin, PRIMUS, Renee, WASLEY, Jan W. F
Published in Bioorganic & medicinal chemistry letters (01.11.2002)
Published in Bioorganic & medicinal chemistry letters (01.11.2002)
Get full text
Journal Article