Use of a HEHEHE Purification Tag Instead of a Hexahistidine Tag Improves Biodistribution of Affibody Molecules Site-Specifically Labeled with Tc-99m, In-111 and I-125
Hofström, Camilla, Orlova, Anna, Altai, Mohamed, Wångsell, Fredrik, Gräslund, Torbjörn, Tolmachev, Vladimir
Published in Journal of medicinal chemistry (2011)
Published in Journal of medicinal chemistry (2011)
Get full text
Journal Article
Synthesis and evaluation of a new class of tertiary alcohol based BACE-1 inhibitors
Russo, Francesco, Wångsell, Fredrik, Sävmarker, Jonas, Jacobsson, Micael, Larhed, Mats
Published in Tetrahedron (28.11.2009)
Published in Tetrahedron (28.11.2009)
Get full text
Journal Article
Investigation of α-phenylnorstatine and α-benzylnorstatine as transition state isostere motifs in the search for new BACE-1 inhibitors
Wångsell, Fredrik, Nordeman, Patrik, Sävmarker, Jonas, Emanuelsson, Rikard, Jansson, Katarina, Lindberg, Jimmy, Rosenquist, Åsa, Samuelsson, Bertil, Larhed, Mats
Published in Bioorganic & medicinal chemistry (01.01.2011)
Published in Bioorganic & medicinal chemistry (01.01.2011)
Get full text
Journal Article
Synthesis of potent BACE-1 inhibitors incorporating a hydroxyethylene isostere as central core
Wångsell, Fredrik, Gustafsson, Karin, Kvarnström, Ingemar, Borkakoti, Neera, Edlund, Michael, Jansson, Katarina, Lindberg, Jimmy, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in European journal of medicinal chemistry (01.03.2010)
Published in European journal of medicinal chemistry (01.03.2010)
Get full text
Journal Article
Design and synthesis of BACE-1 inhibitors utilizing a tertiary hydroxyl motif as the transition state mimic
Wångsell, Fredrik, Russo, Francesco, Sävmarker, Jonas, Rosenquist, Åsa, Samuelsson, Bertil, Larhed, Mats
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Get full text
Journal Article
Synthesis and labeling of a piperazine-based library of 11C-labeled ligands for imaging of the vesicular acetylcholine transporter
Bergman, Sara, Estrada, Sergio, Hall, Håkan, Rahman, Rashidur, Blomgren, Andreas, Larhed, Mats, Svedberg, Marie, Thibblin, Alf, Wångsell, Fredrik, Antoni, Gunnar
Published in Journal of labelled compounds & radiopharmaceuticals (30.06.2014)
Published in Journal of labelled compounds & radiopharmaceuticals (30.06.2014)
Get full text
Journal Article
A3907, a systemic ASBT inhibitor, improves cholestasis in mice by multiorgan activity and shows translational relevance to humans
Caballero-Camino, Francisco J, Rodrigues, Pedro M, Wångsell, Fredrik, Agirre-Lizaso, Aloña, Olaizola, Paula, Izquierdo-Sanchez, Laura, Perugorria, Maria J, Bujanda, Luis, Angelin, Bo, Straniero, Sara, Wallebäck, Anna, Starke, Ingemar, Gillberg, Per-Göran, Strängberg, Ellen, Bonn, Britta, Mattsson, Jan P, Madsen, Martin R, Hansen, Henrik H, Lindström, Erik, Åkerblad, Peter, Banales, Jesus M
Published in Hepatology (Baltimore, Md.) (01.09.2023)
Published in Hepatology (Baltimore, Md.) (01.09.2023)
Get full text
Journal Article
Synthesis of novel potent hepatitis C virus NS3 protease inhibitors: Discovery of 4-hydroxy-cyclopent-2-ene-1,2-dicarboxylic acid as a N-acyl- l-hydroxyproline bioisostere
Thorstensson, Fredrik, Wångsell, Fredrik, Kvarnström, Ingemar, Vrang, Lotta, Hamelink, Elizabeth, Jansson, Katarina, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (2007)
Published in Bioorganic & medicinal chemistry (2007)
Get full text
Journal Article
Radical Functionalization of Unsaturated Amino Acids: Synthesis of Side-Chain-Fluorinated, Azido-Substituted, and Hydroxylated Amino Acids
Reeve, Philip A. P, Grabowska, Urszula, Oden, Lourdes Salvador, Wiktelius, Daniel, Wångsell, Fredrik, Jackson, Richard F. W
Published in ACS omega (30.06.2019)
Published in ACS omega (30.06.2019)
Get full text
Journal Article
OS-074-YI - A3907, a systemic ASBT inhibitor, improves cholestasis in mice by inhibiting multi-organ bile acid transport and shows translational relevance to human
Caballero, Francisco J., Rodrigues, Pedro Miguel, Lizaso, Aloña Agirre, Olaizola, Paula, Izquierdo-Sánchez, Laura, Perugorria, María Jesús, Bujanda, Luis, Angelin, Bo, Straniero, Sara, Wallebäck, Anna, Starke, Ingemar, Gillberg, Per-Göran, Strängberg, Ellen, Wangsell, Fredrik, Mattsson, Jan, Hansen, Henrik B., Lindström, Erik, Akerblad, Peter, Banales, Jesus Maria
Published in Journal of hepatology (01.06.2023)
Published in Journal of hepatology (01.06.2023)
Get full text
Journal Article
A3907, a systemic ASBT inhibitor, improves cholestasis in mice by inhibiting multi-organ bile acid transport and shows translational relevance to human
Caballero, Francisco J., Rodrigues, Pedro Miguel, Lizaso, Aloña Agirre, Olaizola, Paula, Izquierdo-Sánchez, Laura, Perugorria, María Jesús, Bujanda, Luis, Angelin, Bo, Straniero, Sara, Wallebäck, Anna, Starke, Ingemar, Gillberg, Per-Göran, Strängberg, Ellen, Wangsell, Fredrik, Mattsson, Jan, Hansen, Henrik B., Lindström, Erik, Akerblad, Peter, Banales, Jesus Maria
Published in JOURNAL OF HEPATOLOGY (01.06.2023)
Published in JOURNAL OF HEPATOLOGY (01.06.2023)
Get full text
Journal Article
Conference Proceeding
Use of a HEHEHE purification tag instead of a hexahistidine tag improves biodistribution of affibody molecules site-specifically labeled with (99m)Tc, (111)In, and (125)I
Hofstrom, Camilla, Orlova, Anna, Altai, Mohamed, Wangsell, Fredrik, Graslund, Torbjorn, Tolmachev, Vladimir
Published in Journal of medicinal chemistry (09.06.2011)
Published in Journal of medicinal chemistry (09.06.2011)
Get full text
Journal Article
Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: Use of cyclopentane and cyclopentene P2-motifs
Bäck, Marcus, Johansson, Per-Ola, Wångsell, Fredrik, Thorstensson, Fredrik, Kvarnström, Ingemar, Ayesa, Susana, Wähling, Horst, Pelcman, Mikael, Jansson, Katarina, Lindström, Stefan, Wallberg, Hans, Classon, Björn, Rydergård, Christina, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (15.11.2007)
Published in Bioorganic & medicinal chemistry (15.11.2007)
Get full text
Journal Article
메탈로-베타-락타마제 저해제로서의 1-아미노설포닐-2-카르복시피롤 유도체
KIRKHAM JAMES, APPELQVIST PIA, WALLBERG HANS, BUNT ADAM, WANGSELL FREDRIK, WILKINSON ANDREW, COOPER IAN, ORR DAVID, FINLAYSON JONATHAN
Year of Publication 25.07.2022
Get full text
Year of Publication 25.07.2022
Patent
항균 화합물
APPELQVIST PIA, WALLBERG HANS, BUNT ADAM, WANGSELL FREDRIK, WILKINSON ANDREW, COOPER IAN, ORR DAVID, FINLAYSON JONATHAN
Year of Publication 28.01.2021
Get full text
Year of Publication 28.01.2021
Patent
Synthesis and labeling of a piperazine-based library of C-11-labeled ligands for imaging of the vesicular acetylcholine transporter
Bergman, Sara, Estrada, Sergio, Hall, Hakan, Rahman, Rashidur, Blomgren, Andreas, Larhed, Mats, Svedberg, Marie, Thibblin, Alf, Wangsell, Fredrik, Antoni, Gunnar
Published in Journal of labelled compounds & radiopharmaceuticals (30.06.2014)
Published in Journal of labelled compounds & radiopharmaceuticals (30.06.2014)
Get full text
Journal Article
Synthesis and biological evaluation of a piperazine-based library of C-11-Labeled PET tracers for imaging of the vesicular acetylcholine transporter
Bergman, Sara, Blomgren, Andreas, Hall, Håkan, Larhed, Mats, Svedberg, Marie, Thibblin, Alf, Wangsell, Fredrik, Antoni, Gunnar
Published in Journal of labelled compounds & radiopharmaceuticals (2013)
Get full text
Published in Journal of labelled compounds & radiopharmaceuticals (2013)
Journal Article
Use of a HEHEHE Purification Tag Instead of a Hexahistidine Tag Improves Biodistribution of Affibody Molecules Site-Specifically Labeled with 99m Tc, 111 In, and 125 I
Hofström, Camilla, Orlova, Anna, Altai, Mohamed, Wångsell, Fredrik, Gräslund, Torbjörn, Tolmachev, Vladimir
Published in Journal of medicinal chemistry (09.06.2011)
Published in Journal of medicinal chemistry (09.06.2011)
Get full text
Journal Article
ANTIBACTERIAL COMPOUNDS
FINLAYSON, JONATHAN, COOPER, IAN, ORR, DAVID, WILKINSON, ANDREW, BUNT, ADAM, WALLBERG, HANS, WANGSELL, FREDRIK, APPELQVIST, PIA
Year of Publication 21.11.2019
Get full text
Year of Publication 21.11.2019
Patent