Selective and membrane-permeable small molecule inhibitors of nicotinamide N-methyltransferase reverse high fat diet-induced obesity in mice
Neelakantan, Harshini, Vance, Virginia, Wetzel, Michael D., Wang, Hua-Yu Leo, McHardy, Stanton F., Finnerty, Celeste C., Hommel, Jonathan D., Watowich, Stanley J.
Published in Biochemical pharmacology (01.01.2018)
Published in Biochemical pharmacology (01.01.2018)
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Journal Article
Small molecule nicotinamide N-methyltransferase inhibitor activates senescent muscle stem cells and improves regenerative capacity of aged skeletal muscle
Neelakantan, Harshini, Brightwell, Camille R., Graber, Ted G., Maroto, Rosario, Wang, Hua-Yu Leo, McHardy, Stanton F., Papaconstantinou, John, Fry, Christopher S., Watowich, Stanley J.
Published in Biochemical pharmacology (01.05.2019)
Published in Biochemical pharmacology (01.05.2019)
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Journal Article
Digitoxin and a synthetic monosaccharide analog inhibit cell viability in lung cancer cells
Elbaz, Hosam A., Stueckle, Todd A., Wang, Hua-Yu Leo, O'Doherty, George A., Lowry, David T., Sargent, Linda M., Wang, Liying, Dinu, Cerasela Zoica, Rojanasakul, Yon
Published in Toxicology and applied pharmacology (01.01.2012)
Published in Toxicology and applied pharmacology (01.01.2012)
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Asymmetric Synthesis of CIDD-0072424 via an Enantioselective Nitro-Mannich Reaction: A Central Nervous System Penetrant, Selective Small Molecule Inhibitor of Protein Kinase C Epsilon
De Kraker, Harmannus, Wang, Hua-Yu Leo, Arman, Hadi D., Renteria, Rachel N., Fleischer, Caleb N., Messing, Robert O., McHardy, Stanton F.
Published in Journal of organic chemistry (05.04.2024)
Published in Journal of organic chemistry (05.04.2024)
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Journal Article
Selective and brain-penetrant lanosterol synthase inhibitors target glioma stem-like cells by inducing 24(S),25-epoxycholesterol production
Nguyen, Thu P., Wang, Wentian, Sternisha, Alex C., Corley, Chase D., Wang, Hua-Yu Leo, Wang, Xiaoyu, Ortiz, Francisco, Lim, Sang-Kyun, Abdullah, Kalil G., Parada, Luis F., Williams, Noelle S., McBrayer, Samuel K., McDonald, Jeffrey G., De Brabander, Jef K., Nijhawan, Deepak
Published in Cell chemical biology (16.02.2023)
Published in Cell chemical biology (16.02.2023)
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Journal Article
De novo synthesis of deoxy sugar via a Wharton rearrangement
Wang, Hua-Yu Leo, O'Doherty, George A.
Published in Chemical communications (Cambridge, England) (07.10.2011)
Published in Chemical communications (Cambridge, England) (07.10.2011)
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Journal Article
Modulators of Na/K-ATPase: a patent review
Wang, Hua-Yu Leo, O'Doherty, George A
Published in Expert opinion on therapeutic patents (01.06.2012)
Published in Expert opinion on therapeutic patents (01.06.2012)
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Journal Article
Monosaccharide digitoxin derivative sensitize human non-small cell lung cancer cells to anoikis through Mcl-1 proteasomal degradation
Pongrakhananon, Varisa, Stueckle, Todd A., Wang, Hua-Yu Leo, O’Doherty, George A., Dinu, Cerasela Zoica, Chanvorachote, Pithi, Rojanasakul, Yon
Published in Biochemical pharmacology (01.03.2014)
Published in Biochemical pharmacology (01.03.2014)
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Journal Article
Stereochemical Survey of Digitoxin Monosaccharides
Wang, Hua-Yu Leo, Xin, Wenjun, Zhou, Maoquan, Stueckle, Todd A, Rojanasakul, Yon, O'Doherty, George A
Published in ACS medicinal chemistry letters (13.01.2011)
Published in ACS medicinal chemistry letters (13.01.2011)
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Journal Article
C5′-Alkyl Substitution Effects on Digitoxigenin α-l-Glycoside Cancer Cytotoxicity
Wang, Hua-Yu Leo, Wu, Bulan, Zhang, Qi, Kang, Sang-Woo, Rojanasakul, Yon, O’Doherty, George A
Published in ACS medicinal chemistry letters (14.04.2011)
Published in ACS medicinal chemistry letters (14.04.2011)
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Journal Article
Structure–Activity Relationship Study of the Cleistriosides and Cleistetrosides for Antibacterial/Anticancer Activity
Shi, Pei, Silva, Michelle C, Wang, Hua-Yu Leo, Wu, Bulan, Akhmedov, Novruz G, Li, Miaosheng, Beuning, Penny J, O’Doherty, George A
Published in ACS medicinal chemistry letters (13.12.2012)
Published in ACS medicinal chemistry letters (13.12.2012)
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