Screening of a Custom-Designed Acid Fragment Library Identifies 1‑Phenylpyrroles and 1‑Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity
Mahy, William, Patel, Mikesh, Steadman, David, Woodward, Hannah L, Atkinson, Benjamin N, Svensson, Fredrik, Willis, Nicky J, Flint, Alister, Papatheodorou, Dimitra, Zhao, Yuguang, Vecchia, Luca, Ruza, Reinis R, Hillier, James, Frew, Sarah, Monaghan, Amy, Costa, Artur, Bictash, Magda, Walter, Magnus W, Jones, E. Yvonne, Fish, Paul V
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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Journal Article
Platinum catalysed hydrosilylation of propargylic alcohols
McAdam, Catherine A., McLaughlin, Mark G., Johnston, Adam J. S., Chen, Jun, Walter, Magnus W., Cook, Matthew J.
Published in Organic & biomolecular chemistry (21.07.2013)
Published in Organic & biomolecular chemistry (21.07.2013)
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Journal Article
Synthesis of mono Cytochrome P450 in a modified CHO-CPR cell-free protein production platform
Knauer, Jan Felix, Schulz, Christian, Zemella, Anne, Wüstenhagen, Doreen A, Walter, Ruben Magnus, Küpper, Jan-Heiner, Kubick, Stefan
Published in Scientific reports (13.01.2024)
Published in Scientific reports (13.01.2024)
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Journal Article
Biomimetic Synthesis of Pyrone-Derived Natural Products: Exploring Chemical Pathways from a Unique Polyketide Precursor
Eade, Serena J, Walter, Magnus W, Byrne, Colin, Odell, Barbara, Rodriguez, Raphaël, Baldwin, Jack E, Adlington, Robert M, Moses, John E
Published in Journal of organic chemistry (04.07.2008)
Published in Journal of organic chemistry (04.07.2008)
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Journal Article
Fast In Vitro Synthesis and Direct Labeling of Nanobodies for Prototyping in Microscopy Applications
Behrens, Lukas, Walter, Ruben Magnus, Cai, Weining, Ewers, Helge, van Bommel, Bas, Zemella, Anne
Published in ACS omega (20.08.2024)
Published in ACS omega (20.08.2024)
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Journal Article
Design and Synthesis of CNS-targeted Flavones and Analogues with Neuroprotective Potential Against H2O2- and Aβ1-42-Induced Toxicity in SH-SY5Y Human Neuroblastoma Cells
de Matos, Ana M., Martins, Alice, Man, Teresa, Evans, David, Walter, Magnus, Oliveira, Maria Conceição, López, Óscar, Fernandez-Bolaños, José G., Dätwyler, Philipp, Ernst, Beat, Macedo, M. Paula, Contino, Marialessandra, Colabufo, Nicola A., Rauter, Amélia P.
Published in Pharmaceuticals (Basel, Switzerland) (21.06.2019)
Published in Pharmaceuticals (Basel, Switzerland) (21.06.2019)
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Journal Article
Vesicle-based cell-free synthesis of short and long unspecific peroxygenases
Walter, Ruben Magnus, Zemella, Anne, Schramm, Marina, Kiebist, Jan, Kubick, Stefan
Published in Frontiers in bioengineering and biotechnology (01.11.2022)
Published in Frontiers in bioengineering and biotechnology (01.11.2022)
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Journal Article
Diastereoselective Synthesis of Cyclopropane Amino Acids Using Diazo Compounds Generated in Situ
Adams, Luke A, Aggarwal, Varinder K, Bonnert, Roger V, Bressel, Bettina, Cox, Russell J, Shepherd, Jon, de Vicente, Javier, Walter, Magnus, Whittingham, William G, Winn, Caroline L
Published in Journal of organic chemistry (28.11.2003)
Published in Journal of organic chemistry (28.11.2003)
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Journal Article
1-Aryl-3,4-dihydro-1H-quinolin-2-one derivatives, novel and selective norepinephrine reuptake inhibitors
Beadle, Christopher D, Boot, John, Camp, Nicholas P, Dezutter, Nancy, Findlay, Jeremy, Hayhurst, Lorna, Masters, John J, Penariol, Roberta, Walter, Magnus W
Published in Bioorganic & medicinal chemistry letters (15.10.2005)
Published in Bioorganic & medicinal chemistry letters (15.10.2005)
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Journal Article
Neurochemical and behavioral profiling of the selective GlyT1 inhibitors ALX5407 and LY2365109 indicate a preferential action in caudal vs. cortical brain areas
Perry, Kenneth W., Falcone, Julie F., Fell, Matthew J., Ryder, John W., Yu, Hong, Love, Patrick L., Katner, Jason, Gordon, Kimberly D., Wade, Mark R., Man, Teresa, Nomikos, George G., Phebus, Lee A., Cauvin, Annick J., Johnson, Kirk W., Jones, Carrie K., Hoffmann, Beth J., Sandusky, George E., Walter, Magnus W., Porter, Warren J., Yang, Lijuan, Merchant, Kalpana M., Shannon, Harlan E., Svensson, Kjell A.
Published in Neuropharmacology (01.10.2008)
Published in Neuropharmacology (01.10.2008)
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Journal Article
Discovery and SAR studies of novel GlyT1 inhibitors
Walter, Magnus W., Hoffman, Beth J., Gordon, Kimberly, Johnson, Kirk, Love, Patrick, Jones, Matthew, Man, Teresa, Phebus, Lee, Reel, Jon K., Rudyk, Helene C., Shannon, Harlan, Svensson, Kjell, Yu, Hong, Valli, Matthew J., Porter, Warren J.
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
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Journal Article
Discovery and structure–activity relationships of novel selective norepinephrine and dual serotonin/norepinephrine reuptake inhibitors
Boot, John, Cases, Manuel, Clark, Barry P., Findlay, Jeremy, Gallagher, Peter T., Hayhurst, Lorna, Man, Teresa, Montalbetti, Christian, Rathmell, Richard E., Rudyk, Hélène, Walter, Magnus W., Whatton, Maria, Wood, Virginia
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
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Journal Article
Discovery of novel and selective tertiary alcohol containing inhibitors of the norepinephrine transporter
Cases-Thomas, Manuel J., Masters, John J., Walter, Magnus W., Campbell, Gordon, Haughton, Louise, Gallagher, Peter T., Dobson, David R., Mancuso, Vincent, Bonnier, Benjamin, Giard, Thierry, Defrance, Thierry, Vanmarsenille, Michel, Ledgard, Andrew, White, Craig, Ouwerkerk-Mahadevan, Sivi, Brunelle, Francoise J., Dezutter, Nancy A., Herbots, Camy A., Lienard, Joel Y., Findlay, Jeremy, Hayhurst, Lorna, Boot, John, Thompson, Linda K., Hemrick-Luecke, Susan
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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Journal Article
Synthesis of 11C-labelled ( R)-OHDMI and CFMME and their evaluation as candidate radioligands for imaging central norepinephrine transporters with PET
Schou, Magnus, Pike, Victor W., Sóvágó, Judit, Gulyás, Balázs, Gallagher, Peter T., Dobson, David R., Walter, Magnus W., Rudyk, Helene, Farde, Lars, Halldin, Christer
Published in Bioorganic & medicinal chemistry (2007)
Published in Bioorganic & medicinal chemistry (2007)
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Journal Article
A Novel Oxidative Rearrangement of 6-Methoxypyran-2-ones
Eade, Serena J, Adlington, Robert M, Cowley, Andrew R, Walter, Magnus W, Baldwin, Jack E
Published in Organic letters (18.08.2005)
Published in Organic letters (18.08.2005)
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Journal Article
European Medicinal Chemistry Leaders in Industry (EMCL) – On the Status and Future of Medicinal Chemistry Research in Europe
Ali, Amjad, Bauser, Marcus, Bertrand, Sophie, Blackaby, Wesley, Boss, Christoph, Bossart, Martin, Hall, Adrian, Binch, Hayley, Czechtizky, Werngard, Gijsen, Harrie, Haning, Helmut, Hartung, Ingo V., Kilburn, Paul, Lassalle, Gilbert, Lücking, Ulrich, Mack, Jürgen, Missbach, Martin, Otsomaa, Leena, Torrens, Antoni, Wagner, Michael, Walter, Magnus, Weinstabl, Harald, Hijfte, Luc, Nussbaum, Franz
Published in ChemMedChem (03.07.2023)
Published in ChemMedChem (03.07.2023)
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Journal Article
1-Aryl-3,4-dihydro-1H-quinolin-2-one derivatives, novel and selective norepinephrine reuptake inhibitors
BEADLE, Christopher D, BOOT, John, CAMP, Nicholas P, DEZUTTER, Nancy, FINDLAY, Jeremy, HAYHURST, Lorna, MASTERS, John J, PENARIOL, Roberta, WALTER, Magnus W
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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Journal Article