Discovery of 4-benzoyl-1-[(4-methoxy-1H-pyrrolo[2,3-b]lpyridin-3-yl)oxoacetyl]-2-(R)-methylpiperazine (BMS-378806): A novel HIV-1 attachment inhibitor that interferes with CD4-gp120 interactions
Wang, T, Zhang, ZX, Wallace, OB, Deshpande, M, Fang, HQ, Yang, Z, Zadjura, LM, Tweedie, DL, Huang, S, Zhao, F, Ranadive, S, Robinson, BS, Gong, YF, Riccardi, K, Spicer, TP, Deminie, C, Rose, R, Wang, HGH, Blair, WS, Shi, PY, Lin, PF, Colonno, RJ, Meanwell, NA
Published in Journal of medicinal chemistry (25.09.2003)
Published in Journal of medicinal chemistry (25.09.2003)
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Journal Article
Tetrahydroquinoline-Based selective estrogen receptor modulators (SERMs)
Wallace, Owen B, Lauwers, Kenneth S, Jones, Scott A, Dodge, Jeffrey A
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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Journal Article
A Selective Estrogen Receptor Modulator Designed for the Treatment of Uterine Leiomyoma with Unique Tissue Specificity for Uterus and Ovaries in Rats
Hummel, Conrad W, Geiser, Andrew G, Bryant, Henry U, Cohen, Ilene R, Dally, Robert D, Fong, Kin Chiu, Frank, Scott A, Hinklin, Ronald, Jones, Scott A, Lewis, George, McCann, Denis J, Rudmann, Daniel G, Shepherd, Timothy A, Tian, Hongqi, Wallace, Owen B, Wang, Minmin, Wang, Yong, Dodge, Jeffrey A
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
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Journal Article
A New Selective Estrogen Receptor Modulator with Potent Uterine Antagonist Activity, Agonist Activity in Bone, and Minimal Ovarian Stimulation
Geiser, Andrew G, Hummel, Conrad W, Draper, Michael W, Henck, Judith W, Cohen, Ilene R, Rudmann, Daniel G, Donnelly, Kevin B, Adrian, Mary D, Shepherd, Timothy A, Wallace, Owen B, McCann, Denis J, Oldham, Samuel W, Bryant, Henry U, Sato, Masahiko, Dodge, Jeffrey A
Published in Endocrinology (Philadelphia) (01.10.2005)
Published in Endocrinology (Philadelphia) (01.10.2005)
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Journal Article
A Selective Estrogen Receptor Modulator for the Treatment of Hot Flushes
Wallace, Owen B, Lauwers, Kenneth S, Dodge, Jeffrey A, May, Scott A, Calvin, Joel R, Hinklin, Ronald, Bryant, Henry U, Shetler, Pamela K, Adrian, Mary D, Geiser, Andrew G, Sato, Masahiko, Burris, Thomas P
Published in Journal of medicinal chemistry (09.02.2006)
Published in Journal of medicinal chemistry (09.02.2006)
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Journal Article
HIV-1 entry – an expanding portal for drug discovery
Blair, Wade S, Lin, Pin-Fang, Meanwell, Nicholas A, Wallace, Owen B
Published in Drug Discovery Today (01.05.2000)
Published in Drug Discovery Today (01.05.2000)
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Book Review
Journal Article
Benzothiophene and naphthalene derived constrained SERMs
Wallace, Owen B., Bryant, Henry U., Shetler, Pamela K., Adrian, Mary D., Geiser, Andrew G.
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
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Journal Article