Longitudinal changes in EEG power, sleep cycles and behaviour in a tau model of neurodegeneration
Holton, C. M, Hanley, N, Shanks, E, Oxley, P, McCarthy, A, Eastwood, B. J, Murray, T. K, Nickerson, A, Wafford, K. A
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Published in Alzheimer's research & therapy (15.07.2020)
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A study of subunit selectivity, mechanism and site of action of the delta selective compound 2 (DS2) at human recombinant and rodent native GABA(A) receptors
Jensen, M L, Wafford, K A, Brown, A R, Belelli, D, Lambert, J J, Mirza, N R
Published in British journal of pharmacology (01.03.2013)
Published in British journal of pharmacology (01.03.2013)
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MRK-409 (MK-0343), a GABAA receptor subtype-selective partial agonist, is a non-sedating anxiolytic in preclinical species but causes sedation in humans
Atack, J R, Wafford, K A, Street, L J, Dawson, G R, Tye, S, Van Laere, K, Bormans, G, Sanabria-Bohórquez, S M, De Lepeleire, I, de Hoon, J N, Van Hecken, A, Burns, H D, McKernan, R M, Murphy, M G, Hargreaves, R J
Published in Journal of psychopharmacology (Oxford) (01.03.2011)
Published in Journal of psychopharmacology (Oxford) (01.03.2011)
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Differential effects of NMDA antagonists on high frequency and gamma EEG oscillations in a neurodevelopmental model of schizophrenia
Phillips, K.G., Cotel, M.C., McCarthy, A.P., Edgar, D.M., Tricklebank, M., O’Neill, M.J., Jones, M.W., Wafford, K.A.
Published in Neuropharmacology (01.03.2012)
Published in Neuropharmacology (01.03.2012)
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The role of K2P channels in anaesthesia and sleep
Steinberg, E. A., Wafford, K. A., Brickley, S. G., Franks, N. P., Wisden, W.
Published in Pflügers Archiv (01.05.2015)
Published in Pflügers Archiv (01.05.2015)
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Preclinical and clinical pharmacology of TPA023B, a GABAA receptor α2/α3 subtype-selective partial agonist
Atack, J R, Hallett, D J, Tye, S, Wafford, K A, Ryan, C, Sanabria-Bohórquez, S M, Eng, Wai-Si, Gibson, R E, Burns, H D, Dawson, G R, Carling, R W, Street, L J, Pike, A, De Lepeleire, I, Van Laere, K, Bormans, G, de Hoon, J N, Van Hecken, A, McKernan, R M, Murphy, M G, Hargreaves, R J
Published in Journal of psychopharmacology (Oxford) (01.03.2011)
Published in Journal of psychopharmacology (Oxford) (01.03.2011)
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Barbiturate interactions at the human GABAA receptor: dependence on receptor subunit combination
Thompson, S.A., Whiting, P.J., Wafford, K.A.
Published in British journal of pharmacology (01.02.1996)
Published in British journal of pharmacology (01.02.1996)
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Role of the beta subunit in determining the pharmacology of human gamma-aminobutyric acid type A receptors
HADINGHAM, K. L, WINGROVE, P. B, WHITING, P. J, WAFFORD, K. A, BAIN, C, KEMP, J. A, PALMER, K. J, WILSON, A. W, WILCOX, A. S, SIKELA, J. M, RAGAN, C. I
Published in Molecular pharmacology (01.12.1993)
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Published in Molecular pharmacology (01.12.1993)
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Novel compounds selectively enhance delta subunit containing GABA A receptors and increase tonic currents in thalamus
Wafford, K A, van Niel, M B, Ma, Q P, Horridge, E, Herd, M B, Peden, D R, Belelli, D, Lambert, J J
Published in Neuropharmacology (01.01.2009)
Published in Neuropharmacology (01.01.2009)
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Differentiating the role of gamma-aminobutyric acid type A (GABAA) receptor subtypes
Wafford, K A, Macaulay, A J, Fradley, R, O'Meara, G F, Reynolds, D S, Rosahl, T W
Published in Biochemical Society transactions (01.06.2004)
Published in Biochemical Society transactions (01.06.2004)
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Comparative Effects of LY3020371, a Potent and Selective Metabotropic Glutamate (mGlu) 2/3 Receptor Antagonist, and Ketamine, a Noncompetitive N -Methyl-d-Aspartate Receptor Antagonist in Rodents: Evidence Supporting the Use of mGlu2/3 Antagonists, for the Treatment of Depression
Witkin, J M, Mitchell, S N, Wafford, K A, Carter, G, Gilmour, G, Li, J, Eastwood, B J, Overshiner, C, Li, X, Rorick-Kehn, L, Rasmussen, K, Anderson, W H, Nikolayev, A, Tolstikov, V V, Kuo, M-S, Catlow, J T, Li, R, Smith, S C, Mitch, C H, Ornstein, P L, Swanson, S, Monn, J A
Published in The Journal of pharmacology and experimental therapeutics (01.04.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2017)
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Novel compounds selectively enhance δ subunit containing GABAA receptors and increase tonic currents in thalamus
Wafford, K.A., van Niel, M.B., Ma, Q.P., Horridge, E., Herd, M.B., Peden, D.R., Belelli, D., Lambert, J.J.
Published in Neuropharmacology (01.01.2009)
Published in Neuropharmacology (01.01.2009)
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The modulatory action of loreclezole at the gamma-aminobutyric acid type A receptor is determined by a single amino acid in the beta 2 and beta 3 subunit
Wingrove, P B, Wafford, K A, Bain, C, Whiting, P J
Published in Proceedings of the National Academy of Sciences - PNAS (10.05.1994)
Published in Proceedings of the National Academy of Sciences - PNAS (10.05.1994)
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A study of subunit selectivity, mechanism and site of action of the delta selective compound 2 (DS2) at human recombinant and rodent native GABAA receptors
Jensen, ML, Wafford, KA, Brown, AR, Belelli, D, Lambert, JJ, Mirza, NR
Published in British journal of pharmacology (01.03.2013)
Published in British journal of pharmacology (01.03.2013)
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Pharmacological characterization of a novel cell line expressing human alpha(4)beta(3)delta GABA(A) receptors
Brown, N, Kerby, J, Bonnert, T P, Whiting, P J, Wafford, K A
Published in British journal of pharmacology (01.08.2002)
Published in British journal of pharmacology (01.08.2002)
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