Heterocyclic ketones as inhibitors of histone deacetylase
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Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
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Methylpyrrole inhibitors of BET bromodomains
Hasvold, Lisa A., Sheppard, George S., Wang, Le, Fidanze, Steven D., Liu, Dachun, Pratt, John K., Mantei, Robert A., Wada, Carol K., Hubbard, Robbert, Shen, Yu, Lin, Xiaoyu, Huang, Xiaoli, Warder, Scott E., Wilcox, Denise, Li, Leiming, Buchanan, F. Greg, Smithee, Lauren, Albert, Daniel H., Magoc, Terrance J., Park, Chang H., Petros, Andrew M., Panchal, Sanjay C., Sun, Chaohong, Kovar, Peter, Soni, Nirupama B., Elmore, Steven W., Kati, Warren M., McDaniel, Keith F.
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
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Trifluoromethyl ketones as inhibitors of histone deacetylase
Frey, Robin R., Wada, Carol K., Garland, Robert B., Curtin, Michael L., Michaelides, Michael R., Li, Junling, Pease, Lori J., Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Murphy, Shannon S., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
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α-Keto amides as inhibitors of histone deacetylase
Wada, Carol K., Frey, Robin R., Ji, Zhiqin, Curtin, Michael L., Garland, Robert B., Holms, James H., Li, Junling, Pease, Lori J., Guo, Jun, Glaser, Keith B., Marcotte, Patrick A., Richardson, Paul L., Murphy, Shannon S., Bouska, Jennifer J., Tapang, Paul, Magoc, Terrance J., Albert, Daniel H., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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Phenoxyphenyl Sulfone N-Formylhydroxylamines (Retrohydroxamates) as Potent, Selective, Orally Bioavailable Matrix Metalloproteinase Inhibitors
Wada, Carol K, Holms, James H, Curtin, Michael L, Dai, Yujia, Florjancic, Alan S, Garland, Robert B, Guo, Yan, Heyman, H. Robin, Stacey, Jamie R, Steinman, Douglas H, Albert, Daniel H, Bouska, Jennifer J, Elmore, Ildiko N, Goodfellow, Carole L, Marcotte, Patrick A, Tapang, Paul, Morgan, Douglas W, Michaelides, Michael R, Davidsen, Steven K
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
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Biaryl Ether Retrohydroxamates as Potent, Long-lived, Orally Bioavailable MMP Inhibitors
Michaelides, Michael R., Dellaria, Joseph F., Gong, Jane, Holms, James H., Bouska, Jennifer J., Stacey, Jamie, Wada, Carol K., Heyman, H.Robin, Curtin, Michael L., Guo, Yan, Goodfellow, Carole L., Elmore, Ildiko B., Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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Journal Article
Discovery and characterization of the potent, selective and orally bioavailable MMP inhibitor ABT-770
Curtin, Michael L., Florjancic, Alan S., Heyman, H.Robin, Michaelides, Michael R., Garland, Robert B., Holms, James H., Steinman, Douglas H., Dellaria, Joseph F., Gong, Jane, Wada, Carol K., Guo, Yan, Elmore, Ildiko B., Tapang, Paul, Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Bouska, Jennifer J., Goodfellow, Carole L., Bauch, Joy L., Marsh, Kennan C., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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BROMODOMAIN INHIBITORS
HOLMS JAMES H, MANTEI ROBERT A, FIDANZE STEVEN D, HASVOLD LISA, WANG LE, DAI YUJIA, SHEPPARD GEORGE S, LIU DACHUN, KATI WARREN M, MCDANIEL KEITH F, MCCLELLAN WILLIAM J, WADA CAROL K, PRATT JOHN K
Year of Publication 24.09.2014
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Year of Publication 24.09.2014
Patent
THIENOPYRIDINE AND FUROPYRIDINE KINASE INHIBITORS
HEYMAN HOWARD R, RAFFERTY PAUL, MICHAELIDES MICHAEL R, CALDERWOOD DAVID J, HIRST GAVIN C, DAVIS HEATHER M, MUCKEY MELANIE A, DAVIDSEN STEVEN K, CURTIN MICHAEL L, WADA CAROL K, BETSCHMANN PATRICK, BURCHAT ANDREW F, HRNCIAR PETER, FREY ROBIN R
Year of Publication 15.11.2011
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Year of Publication 15.11.2011
Patent
Methylpyrrole inhibitors of BET bromodomains
Hasvold, Lisa A., Sheppard, George S., Wang, Le, Fidanze, Steven D., Liu, Dachun, Pratt, John K., Mantei, Robert A., Wada, Carol K., Hubbard, Robbert, Shen, Yu, Lin, Xiaoyu, Huang, Xiaoli, Warder, Scott E., Wilcox, Denise, Li, Leiming, Buchanan, F. Greg, Smithee, Lauren, Albert, Daniel H., Magoc, Terrance J., Park, Chang H., Petros, Andrew M., Panchal, Sanjay C., Sun, Chaohong, Kovar, Peter, Soni, Nirupama B., Elmore, Steven W., Kati, Warren M., McDaniel, Keith F.
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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Integrin α ν β 3 Targeted Gene Delivery Using RGD Peptidomimetic Conjugates with Copolymers of PEGylated Poly(ethylene imine)
Merkel, Olivia M., Germershaus, Oliver, Wada, Carol K., Tarcha, Peter J., Merdan, Thomas, Kissel, Thomas
Published in Bioconjugate chemistry (17.06.2009)
Published in Bioconjugate chemistry (17.06.2009)
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Journal Article
Integrin [alpha]^sub v^[beta]^sub 3^ Targeted Gene Delivery Using RGD Peptidomimetic Conjugates with Copolymers of PEGylated Poly(ethylene imine)
Merkel, Olivia M, Germershaus, Oliver, Wada, Carol K, Tarcha, Peter J, Merdan, Thomas, Kissel, Thomas
Published in Bioconjugate chemistry (17.06.2009)
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Published in Bioconjugate chemistry (17.06.2009)
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Integrin anb3 Targeted Gene Delivery Using RGD Peptidomimetic Conjugates with Copolymers of PEGylated Poly(ethylene imine)
Merkel, Olivia M, Germershaus, Oliver, Wada, Carol K, Tarcha, Peter J, Merdan, Thomas, Kissel, Thomas
Published in Bioconjugate chemistry (28.05.2009)
Published in Bioconjugate chemistry (28.05.2009)
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Journal Article
Integrin alphaVbeta3 targeted gene delivery using RGD peptidomimetic conjugates with copolymers of PEGylated poly(ethylene imine)
Merkel, Olivia M, Germershaus, Oliver, Wada, Carol K, Tarcha, Peter J, Merdan, Thomas, Kissel, Thomas
Published in Bioconjugate chemistry (01.06.2009)
Published in Bioconjugate chemistry (01.06.2009)
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Journal Article
BROMODOMAIN INHIBITORS
Fidanze, Steven D, Kati, Warren M, Sheppard, George S, Wada, Carol K, Wang, Le, McDaniel, Keith F, Holms, James H, Mantei, Robert A, Pratt, John K, McClellan, William J, Liu, Dachun, Dai, Yujia, Hasvold, Lisa
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
Patent